Compuesto clorhidrato de (4a-r, 9a-s)-1-(1h-benzoimidazol-5-carbonil-2,3,4,4a,9,9a-hexahidro-1 h-inden[2,1-b] piridin-6-carbonitrilo y sus formas cristalinas i y ii, inhibidores de hsd 1; composicion farmaceutica; metodo para producir la forma cristalina i del compuesto; metodo para producir la forma cristalina ii del compuesto
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Year of Publication 08.11.2013
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Year of Publication 08.11.2013
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CRYSTALLINE FORMS OF HYDROCHLORIDE SALT OF (4A-R,9A-S)-1-(1H-BENZOIMIDAZOLE-5-CARBONYL)-2,3,4,4A,9,9A-HEXAHYDRO-1H-INDENO [2,1-B]PYRIDINE-6-CARBONITRILE AND THEIR USE AS HSD 1 INHIBITORS
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Year of Publication 11.09.2013
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Year of Publication 11.09.2013
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Crystalline forms of 1-chloro-4-(beta-D-glucopyranos-1-yl)-2-[4-ethynyl-benzyl)-benzene, methods for its preparation and the use thereof for preparing medicaments
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Year of Publication 13.08.2013
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Year of Publication 13.08.2013
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CRYSTALLINE FORMS OF HYDROCHLORIDE SALT OF (4A-R,9A-S) -1- (1H - BENZOIMIDAZOLE- 5 -CARBONYL) -2, 3, 4, 4A, 9, 9A - HEXAHYDRO -1H- INDENO [2, 1 -B] PYRIDINE- 6 -CARBONITRILE AND THEIR USE AS HSD 1 INHIBITORS
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Year of Publication 28.06.2013
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Year of Publication 28.06.2013
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CRYSTALLINE FORM OF 4-(BETA-D-GLUCOPYRANOS-1-YL)-1-METHYL-2-[4-((S)-TETRAHYDROFURAN-3-YLOXY)-BENZYL]-BENZENE, A METHOD FOR ITS PREPARATION AND THE USE THEREOF FOR PREPARING MEDICAMENTS
ECKHARDT MATTHIAS, MARTIN HANS-JUERGEN, HIMMELSBACH FRANK, BUTZ TANJA M
Year of Publication 16.12.2010
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Year of Publication 16.12.2010
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CRYSTALLINE COMPLEX OF 1-CYANO-2-(4-CYCLOPROPYL-BENZYL)-4-(β-D-GLUCOPYRANOS-1-YL)BENZENE, METHODS FOR ITS PREPARATION AND THE USE THEREOF FOR PREPARING MEDICAMENTSCRYSTALLINE COMPLEX OF 1-CYANO-2-(4-CYCLOPROPYL-BENZYL)-4-(β-D-GLUCOPYRANOS-1-YL)BENZENE, METHODS FOR ITS PREPARATION AND THE USE THEREOF FOR PREPARING MEDICAMENTS
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Year of Publication 30.12.2016
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Year of Publication 30.12.2016
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Crystalline forms of hydrochloride salt of (4a-R,9a-S) -1- (1h - benzoimidazole- 5 -carbonyl) -2, 3, 4, 4a, 9, 9a - hexahydro -1h- indeno [2, 1 -b] pyridine- 6 -carbonitrile and their use as HSD 1 inhibitors
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Year of Publication 02.05.2013
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Year of Publication 02.05.2013
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CRYSTALLINE FORMS OF HYDROCHLORIDE SALT OF (4A-R,9A-S) -1- (1H - BENZOIMIDAZOLE- 5 -CARBONYL) -2, 3, 4, 4A, 9, 9A - HEXAHYDRO -1H- INDENO [2, 1 -B] PYRIDINE- 6 -CARBONITRILE AND THEIR USE AS HSD 1 INHIBITORS (4A-R9A-S)-1-(1H--5-)-2344A99A--1H-[21-B] -6- HSD1
MARTIN SCHUEHLE M, HANS-JUERGEN MARTIN H-J, SANDRA SICK S, BING-SHIOU YANG B-S, MATTHIAS ECKHARDT M
Year of Publication 17.01.2014
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Year of Publication 17.01.2014
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ARYL-AND HETEROARYLCARBONYL DERIVATIVES OF HEXAHYDROINDENOPYRIDINE AND OCTAHYDROBENZOQUINOLINE
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Year of Publication 21.06.2012
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Year of Publication 21.06.2012
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CRYSTALLINE FORMS OF HYDROCHLORIDE SALT OF (4A-R,9A-S) -1- (1H - BENZOIMIDAZOLE- 5 -CARBONYL) -2, 3, 4, 4A, 9, 9A - HEXAHYDRO -1H- INDENO [2, 1 -B] PYRIDINE- 6 -CARBONITRILE AND THEIR USE AS HSD 1 INHIBITORS
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Year of Publication 10.05.2012
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Year of Publication 10.05.2012
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CRYSTALLINE FORMS OF HYDROCHLORIDE SALT OF (4A-R,9A-S) -1- (1H - BENZOIMIDAZOLE- 5 -CARBONYL) -2, 3, 4, 4A, 9, 9A - HEXAHYDRO -1H- INDENO [2, 1 -B] PYRIDINE- 6 -CARBONITRILE AND THEIR USE AS HSD 1 INHIBITORS
YANG, BING-SHIOU, SICK, SANDRA, ECKHARDT, MATTHIAS, MARTIN, HANS-JUERGEN, SCHUEHLE, MARTIN
Year of Publication 10.05.2012
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Year of Publication 10.05.2012
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CRYSTALLINE FORM OF 4-(ß-D-GLUCOPYRANOS-1-YL)-1-METHYL-2-[4-((S)-TETRAHYDROFURAN-3-YLOXY)-BENZYL]-BENZENE, A METHOD FOR ITS PREPARATION AND THE USE THEREOF FOR PREPARING MEDICAMENTS
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Year of Publication 12.08.2009
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Year of Publication 12.08.2009
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CRYSTALLINE FORM OF 4-(.BETA.-D-GLUCOPYRANOS-1-YL)-1-METHYL-2-[4-((S)-TETRAHYDROFURAN-3-YLOXY)-BENZYL]-BENZENE, A METHOD FOR ITS PREPARATION AND THE USE THEREOF FOR PREPARING MEDICAMENTS
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Year of Publication 02.05.2008
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Year of Publication 02.05.2008
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CRYSTALLINE FORM OF 4-(ß-D-GLUCOPYRANOS-1-YL)-1-METHYL-2-[4-((S)-TETRAHYDROFURAN-3-YLOXY)-BENZYL]-BENZENE, A METHOD FOR ITS PREPARATION AND THE USE THEREOF FOR PREPARING MEDICAMENTS
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Year of Publication 02.05.2008
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Year of Publication 02.05.2008
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Year of Publication 15.01.2011
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Year of Publication 15.01.2011
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ΚΡΥΣΤΑΛΛΙΚΕΣ ΜΟΡΦΕΣ ΥΔΡΟΧΛΩΡΙΚΟΥ ΑΛΑΤΟΣ (4Α-R,9Α-S)-1-(1Η-ΒΕΝΖΟΪΜΙΔΑΖΟΛΟ-5-ΚΑΡΒΟΝΥΛ)2,3,4,4Α,9,9Α-ΕΞΑΫΔΡΟ-1Η-ΙΝΔΕΝΟ[2,1-Β]ΠΥΡΙΔΙΝΟ-6-ΚΑΡΒΟΝΙΤΡΙΛΙΟΥ ΚΑΙ ΧΡΗΣΗ ΤΟΥΣ ΩΣ ΑΝΑΣΤΟΛΕΙΣ ΤΗΣ HSD 1
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Year of Publication 25.01.2017
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Year of Publication 25.01.2017
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CRYSTALLINE FORMS OF 1-CHLORO-4-(ß-D-GLUCOPYRANOS-1-YL)-2-(4-ETHYNYL-BENZYL)-BENZENE, METHODS FOR ITS PREPARATION AND THE USE THEREOF FOR PREPARING MEDICAMENTS
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Year of Publication 15.12.2010
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Year of Publication 15.12.2010
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Crystalline forms of 1-chloro-4-(β-D-glucopyranos-1-yl)-2-[4-
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Year of Publication 25.05.2010
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Year of Publication 25.05.2010
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