Optimization of Thienopyrrole‐Based Finger‐Loop Inhibitors of the Hepatitis C Virus NS5B Polymerase
Martin Hernando, Jose Ignacio, Ontoria, Jesus Maria, Malancona, Savina, Attenni, Barbara, Fiore, Fabrizio, Bonelli, Fabio, Koch, Uwe, Di Marco, Stefania, Colarusso, Stefania, Ponzi, Simona, Gennari, Nadia, Vignetti, Sue Ellen, del Rosario Rico Ferreira, Maria, Habermann, Jörg, Rowley, Michael, Narjes, Frank
Published in ChemMedChem (05.10.2009)
Published in ChemMedChem (05.10.2009)
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The Discovery of Novel Antimalarial Aminoxadiazoles as a Promising Nonendoperoxide Scaffold
Sandoval, Elena, Lafuente-Monasterio, María José, Almela, María J, Castañeda, Pablo, Jiménez Díaz, María Belén, Martínez-Martínez, María S, Vidal, Jaume, Angulo-Barturen, Íñigo, Bamborough, Paul, Burrows, Jeremy, Cammack, Nicholas, Chaparro, María J, Coterón, José M, de Cozar, Cristina, Crespo, Benigno, Díaz, Beatriz, Drewes, Gerard, Fernández, Esther, Ferrer-Bazaga, Santiago, Fraile, María Teresa, Gamo, Francisco J, Ghidelli-Disse, Sonja, Gómez, Rubén, Haselden, John, Huss, Sophie, León, María Luisa, de Mercado, Jaime, Macdonald, Simon J. F, Martín Hernando, José Ignacio, Prats, Sara, Puente, Margarita, Rodríguez, Anne, de la Rosa, Juan C, Rueda, Lourdes, Selenski, Carolyn, Willis, Paul, Wilson, David M, Witty, Michael, Calderón, Félix
Published in Journal of medicinal chemistry (24.08.2017)
Published in Journal of medicinal chemistry (24.08.2017)
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Journal Article
Correction to The Discovery of Novel Antimalarial Aminoxadiazoles as a Promising Nonendoperoxide Scaffold
Sandoval, Elena, Lafuente-Monasterio, María José, Almela, María J., Castañeda, Pablo, Jiménez Díaz, María Belén, Martínez-Martínez, María S., Vidal, Jaume, Angulo-Barturen, Íñigo, Bamborough, Paul, Burrows, Jeremy, Cammack, Nicholas, Chaparro, María J., Coterón, José M., de Cozar, Cristina, Crespo, Benigno, Díaz, Beatriz, Drewes, Gerard, Fernández, Esther, Ferrer-Bazaga, Santiago, Fraile, María Teresa, Gamo, Francisco J., Ghidelli-Disse, Sonja, Gómez, Rubén, Haselden, John, Huss, Sophie, León, María Luisa, de Mercado, Jaime, Macdonald, Simon J. F., Martín Hernando, José Ignacio, Prats, Sara, Puente, Margarita, Rodríguez, Anne, de la Rosa, Juan C., Rueda, Lourdes, Selenski, Carolyn, Willis, Paul, Wilson, David M., Witty, Michael, Calderón, Félix
Published in Journal of medicinal chemistry (14.12.2017)
Published in Journal of medicinal chemistry (14.12.2017)
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Identification of MK-5710 ((8aS)-8a-methyl-1,3-dioxo-2-[(1S,2R)-2-phenylcyclopropyl]-N-(1-phenyl-1H-pyrazol-5-yl)hexahydroimid azo[1,5-a]pyrazine-7(1H)-carboxamide), a potent smoothened antagonist for use in Hedgehog pathway dependent malignancies, Part 1
Malancona, Savina, Altamura, Sergio, Filocamo, Gessica, Kinzel, Olaf, Hernando, Jose Ignacio Martin, Rowley, Michael, Scarpelli, Rita, Steinkühler, Christian, Jones, Philip
Published in Bioorganic & medicinal chemistry letters (01.08.2011)
Published in Bioorganic & medicinal chemistry letters (01.08.2011)
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Journal Article
Identification of MK-5710 ((8aS)-8a-methyl-1,3-dioxo-2-[(1S,2R)-2-phenylcyclo- propyl]-N-(1-phenyl-1H-pyrazol-5-yl)hexahydro-imidazo[1,5-a]pyrazine-7(1H)-carboxamide), a potent smoothened antagonist for use in Hedgehog pathway dependent malignancies, Part 2
Kinzel, Olaf, Alfieri, Anna, Altamura, Sergio, Brunetti, Mirko, Bufali, Simone, Colaceci, Fabrizio, Ferrigno, Federica, Filocamo, Gessica, Fonsi, Massimiliano, Gallinari, Paola, Malancona, Savina, Hernando, Jose Ignacio Martin, Monteagudo, Edith, Orsale, Maria Vittoria, Palumbi, Maria Cecilia, Pucci, Vincenzo, Rowley, Michael, Sasso, Romina, Scarpelli, Rita, Steinkühler, Christian, Jones, Philip
Published in Bioorganic & medicinal chemistry letters (01.08.2011)
Published in Bioorganic & medicinal chemistry letters (01.08.2011)
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Journal Article
Influence of the substitution pattern on the Pb(OAc) 4 mediated oxidative cleavage of steroidal 1,2-diols
Martı́n Hernando, José Ignacio, Rico Ferreira, Maria del Rosario, Candela Lena, José Ignacio, Toupet, Loı̈c, Birlirakis, Nicolas, Arseniyadis, Siméon
Published in Tetrahedron: asymmetry (15.10.1999)
Published in Tetrahedron: asymmetry (15.10.1999)
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Journal Article
Development of Chemical Entities Endowed with Potent Fast-Killing Properties against Plasmodium falciparum Malaria Parasites
Matralis, Alexios N, Malik, Adnan, Penzo, Maria, Moreno, Inmaculada, Almela, Maria J, Camino, Isabel, Crespo, Benigno, Saadeddin, Anas, Ghidelli-Disse, Sonja, Rueda, Lourdes, Calderon, Felix, Osborne, Simon A, Drewes, Gerard, Böesche, Markus, Fernández-Álvaro, Elena, Martin Hernando, Jose Ignacio, Baker, David A
Published in Journal of medicinal chemistry (24.10.2019)
Published in Journal of medicinal chemistry (24.10.2019)
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Journal Article
Studies towards the taxoid diterpene ABC-ring system: practical access to highly functionalized enantiomerically pure analogues of major group representatives
Martı́n Hernando, José Ignacio, del Rosario Rico Ferreira, Maria, Candela Lena, José Ignacio, Birlirakis, Nicolas, Arseniyadis, Siméon
Published in Tetrahedron: asymmetry (10.03.2000)
Published in Tetrahedron: asymmetry (10.03.2000)
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Journal Article
Modified steroids: Pb(OAc) 4 mediated one-pot multistage transformations of steroidal unsaturated 1,2-diols
del Rosario Rico Ferreira, Maria, Martı́n Hernando, José Ignacio, Candela Lena, José Ignacio, Quı́lez del Moral, José, Arseniyadis, Siméon
Published in Tetrahedron: asymmetry (23.04.1999)
Published in Tetrahedron: asymmetry (23.04.1999)
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Advanced taxoids from Hajos-Parrish ketone and isophorone by the transmetallation (C11-C12)-aldol (C1-C2) approach
Ferreira, MDR, Hernando, JIM, Lena, JIC, Birlirakis, N, Arseniyadis, S
Published in Synlett (01.01.2000)
Published in Synlett (01.01.2000)
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A rapid entry into major groups of taxoids
Ignacio Martı́n Hernando, José, del Rosario Rico Ferreira, Maria, Ignacio Candela Lena, José, Birlirakis, Nicolas, Arseniyadis, Siméon
Published in Tetrahedron letters (05.02.2000)
Published in Tetrahedron letters (05.02.2000)
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Journal Article
Stereoselective synthesis of an A-seco-taxoid subunit using the Aldol-annelation-fragmentation strategy
Arseniyadis, Siméon, del Rosario Rico Ferreira, María, Quílez del Moral, José, Ignacio Martín Hernando, José, Potier, Pierre, Toupet, Loïc
Published in Tetrahedron letters (01.10.1998)
Published in Tetrahedron letters (01.10.1998)
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Year of Publication 21.03.2022
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Year of Publication 23.02.2022
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Year of Publication 23.02.2022
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