How TCRs bind MHCs, peptides, and coreceptors
Rudolph, Markus G, Stanfield, Robyn L, Wilson, Ian A
Published in Annual Review of Immunology (01.01.2006)
Published in Annual Review of Immunology (01.01.2006)
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Journal Article
Using macromolecular phasing and refinement techniques for a small molecule gyrase inhibitor
Rudolph, Markus G., Guba, Wolfgang, Xuefei, Tan, Xu, Bruce
Published in Biophysical journal (10.02.2023)
Published in Biophysical journal (10.02.2023)
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Journal Article
Structural Basis for Allosteric Ligand Recognition in the Human CC Chemokine Receptor 7
Jaeger, Kathrin, Bruenle, Steffen, Weinert, Tobias, Guba, Wolfgang, Muehle, Jonas, Miyazaki, Takuya, Weber, Martin, Furrer, Antonia, Haenggi, Noemi, Tetaz, Tim, Huang, Chia-Ying, Mattle, Daniel, Vonach, Jean-Marie, Gast, Alain, Kuglstatter, Andreas, Rudolph, Markus G., Nogly, Przemyslaw, Benz, Joerg, Dawson, Roger J.P., Standfuss, Joerg
Published in Cell (22.08.2019)
Published in Cell (22.08.2019)
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Journal Article
D3R Grand Challenge 2: blind prediction of protein–ligand poses, affinity rankings, and relative binding free energies
Gaieb, Zied, Liu, Shuai, Gathiaka, Symon, Chiu, Michael, Yang, Huanwang, Shao, Chenghua, Feher, Victoria A., Walters, W. Patrick, Kuhn, Bernd, Rudolph, Markus G., Burley, Stephen K., Gilson, Michael K., Amaro, Rommie E.
Published in Journal of computer-aided molecular design (01.01.2018)
Published in Journal of computer-aided molecular design (01.01.2018)
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Journal Article
DNA-Encoded Library-Derived DDR1 Inhibitor Prevents Fibrosis and Renal Function Loss in a Genetic Mouse Model of Alport Syndrome
Richter, Hans, Satz, Alexander L, Bedoucha, Marc, Buettelmann, Bernd, Petersen, Ann C, Harmeier, Anja, Hermosilla, Ricardo, Hochstrasser, Remo, Burger, Dominique, Gsell, Bernard, Gasser, Rodolfo, Huber, Sylwia, Hug, Melanie N, Kocer, Buelent, Kuhn, Bernd, Ritter, Martin, Rudolph, Markus G, Weibel, Franziska, Molina-David, Judith, Kim, Jin-Ju, Santos, Javier Varona, Stihle, Martine, Georges, Guy J, Bonfil, R. Daniel, Fridman, Rafael, Uhles, Sabine, Moll, Solange, Faul, Christian, Fornoni, Alessia, Prunotto, Marco
Published in ACS chemical biology (18.01.2019)
Published in ACS chemical biology (18.01.2019)
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Journal Article
Discovery of a Series of Indane-Containing NBTIs with Activity against Multidrug-Resistant Gram-Negative Pathogens
Cumming, John G., Kreis, Lukas, Kühne, Holger, Wermuth, Roger, Vercruysse, Maarten, Kramer, Christian, Rudolph, Markus G., Xu, Zhiheng
Published in ACS medicinal chemistry letters (13.07.2023)
Published in ACS medicinal chemistry letters (13.07.2023)
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Journal Article
Structure of reverse gyrase with a minimal latch that supports ATP‐dependent positive supercoiling without specific interactions with the topoisomerase domain
Mhaindarkar, Vaibhav P., Rasche, René, Kümmel, Daniel, Rudolph, Markus G., Klostermeier, Dagmar
Published in Acta crystallographica. Section D, Biological crystallography. (01.06.2023)
Published in Acta crystallographica. Section D, Biological crystallography. (01.06.2023)
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Journal Article
TIP47 functions in the biogenesis of lipid droplets
Bulankina, Anna V, Deggerich, Anke, Wenzel, Dirk, Mutenda, Kudzai, Wittmann, Julia G, Rudolph, Markus G, Burger, Koert N.J, Höning, Stefan
Published in The Journal of cell biology (18.05.2009)
Published in The Journal of cell biology (18.05.2009)
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Journal Article
Discovery of a microbial transglutaminase enabling highly site-specific labeling of proteins
Steffen, Wojtek, Ko, Fu Chong, Patel, Jigar, Lyamichev, Victor, Albert, Thomas J., Benz, Jörg, Rudolph, Markus G., Bergmann, Frank, Streidl, Thomas, Kratzsch, Peter, Boenitz-Dulat, Mara, Oelschlaegel, Tobias, Schraeml, Michael
Published in The Journal of biological chemistry (22.09.2017)
Published in The Journal of biological chemistry (22.09.2017)
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Journal Article
A Real-World Perspective on Molecular Design
Kuhn, Bernd, Guba, Wolfgang, Hert, Jérôme, Banner, David, Bissantz, Caterina, Ceccarelli, Simona, Haap, Wolfgang, Körner, Matthias, Kuglstatter, Andreas, Lerner, Christian, Mattei, Patrizio, Neidhart, Werner, Pinard, Emmanuel, Rudolph, Markus G, Schulz-Gasch, Tanja, Woltering, Thomas, Stahl, Martin
Published in Journal of medicinal chemistry (12.05.2016)
Published in Journal of medicinal chemistry (12.05.2016)
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Journal Article
A high quality, industrial data set for binding affinity prediction: performance comparison in different early drug discovery scenarios
Tosstorff, Andreas, Rudolph, Markus G., Cole, Jason C., Reutlinger, Michael, Kramer, Christian, Schaffhauser, Hervé, Nilly, Agnès, Flohr, Alexander, Kuhn, Bernd
Published in Journal of computer-aided molecular design (01.10.2022)
Published in Journal of computer-aided molecular design (01.10.2022)
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Journal Article
Details Matter in Structure-based Drug Design
Kuhn, Bernd, Peters, Jens-Uwe, Rudolph, Markus G, Mohr, Peter, Stahl, Martin, Tosstorff, Andreas
Published in Chimia (01.08.2023)
Published in Chimia (01.08.2023)
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Journal Article
Ligand channel in pharmacologically stabilized rhodopsin
Mattle, Daniel, Kuhn, Bernd, Aebi, Johannes, Bedoucha, Marc, Kekilli, Demet, Grozinger, Nathalie, Alker, Andre, Rudolph, Markus G., Schmid, Georg, Schertler, Gebhard F. X., Hennig, Michael, Standfuss, Jörg, Dawson, Roger J. P.
Published in Proceedings of the National Academy of Sciences - PNAS (03.04.2018)
Published in Proceedings of the National Academy of Sciences - PNAS (03.04.2018)
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Journal Article
Structure of the Acid-sensing ion channel 1 in complex with the gating modifier Psalmotoxin 1
Dawson, Roger J.P., Benz, Jörg, Stohler, Peter, Tetaz, Tim, Joseph, Catherine, Huber, Sylwia, Schmid, Georg, Hügin, Daniela, Pflimlin, Pascal, Trube, Gerd, Rudolph, Markus G., Hennig, Michael, Ruf, Armin
Published in Nature communications (03.07.2012)
Published in Nature communications (03.07.2012)
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Journal Article
Small molecule AX-024 reduces T cell proliferation independently of CD3ϵ/Nck1 interaction, which is governed by a domain swap in the Nck1-SH3.1 domain
Richter, Kirsten, Rufer, Arne C., Muller, Magali, Burger, Dominique, Casagrande, Fabio, Grossenbacher, Tabea, Huber, Sylwia, Hug, Melanie N., Koldewey, Philipp, D'Osualdo, Andrea, Schlatter, Daniel, Stoll, Theodor, Rudolph, Markus G.
Published in The Journal of biological chemistry (05.06.2020)
Published in The Journal of biological chemistry (05.06.2020)
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Journal Article
Chemoproteomic discovery of a covalent allosteric inhibitor of WRN helicase
Baltgalvis, Kristen A., Lamb, Kelsey N., Symons, Kent T., Wu, Chu-Chiao, Hoffman, Melissa A., Snead, Aaron N., Song, Xiaodan, Glaza, Thomas, Kikuchi, Shota, Green, Jason C., Rogness, Donald C., Lam, Betty, Rodriguez-Aguirre, Maria E., Woody, David R., Eissler, Christie L., Rodiles, Socorro, Negron, Seth M., Bernard, Steffen M., Tran, Eileen, Pollock, Jonathan, Tabatabaei, Ali, Contreras, Victor, Williams, Heather N., Pastuszka, Martha K., Sigler, John J., Pettazzoni, Piergiorgio, Rudolph, Markus G., Classen, Moritz, Brugger, Doris, Claiborne, Christopher, Plancher, Jean-Marc, Cuartas, Isabel, Seoane, Joan, Burgess, Laurence E., Abraham, Robert T., Weinstein, David S., Simon, Gabriel M., Patricelli, Matthew P., Kinsella, Todd M.
Published in Nature (London) (09.05.2024)
Published in Nature (London) (09.05.2024)
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