Organocatalytic Enantioselective One-Pot Four-Component Ugi-Type Multicomponent Reaction for the Synthesis of Epoxy-tetrahydropyrrolo[3,4-b]pyridin-5-ones
Su, Yingpeng, Bouma, Marinus J., Alcaraz, Lilian, Stocks, Mike, Furber, Mark, Masson, Géraldine, Zhu, Jieping
Published in Chemistry : a European journal (01.10.2012)
Published in Chemistry : a European journal (01.10.2012)
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Anti-trypanosomal activity of non-peptidic nitrile-based cysteine protease inhibitors
Burtoloso, Antonio C B, de Albuquerque, Sérgio, Furber, Mark, Gomes, Juliana C, Gonçalez, Cristiana, Kenny, Peter W, Leitão, Andrei, Montanari, Carlos A, Quilles, Júnior, José Carlos, Ribeiro, Jean F R, Rocha, Josmar R
Published in PLoS neglected tropical diseases (21.02.2017)
Published in PLoS neglected tropical diseases (21.02.2017)
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NIK-IKK complex interaction controls NF-κB-dependent inflammatory activation of endothelium in response to LTβR ligation
Kucharzewska, Paulina, Maracle, Chrissta X, Jeucken, Kim C M, van Hamburg, Jan Piet, Israelsson, Elisabeth, Furber, Mark, Tas, Sander W, Olsson, Henric K
Published in Journal of cell science (01.04.2019)
Published in Journal of cell science (01.04.2019)
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Chiral Phosphoric Acid-Catalyzed Enantioselective Three- Component Aza-Diels-Alder Reactions of Aminopyrroles and Aminopyrazoles
Brioche, Julien, Courant, Thibaut, Alcaraz, Lilian, Stocks, Michael, Furber, Mark, Zhu, Jieping, Masson, Géraldine
Published in Advanced synthesis & catalysis (26.05.2014)
Published in Advanced synthesis & catalysis (26.05.2014)
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Cathepsin C Inhibitors: Property Optimization and Identification of a Clinical Candidate
Furber, Mark, Tiden, Anna-Karin, Gardiner, Philip, Mete, Antonio, Ford, Rhonan, Millichip, Ian, Stein, Linda, Mather, Andrew, Kinchin, Elizabeth, Luckhurst, Christopher, Barber, Simon, Cage, Peter, Sanganee, Hitesh, Austin, Rupert, Chohan, Kamaldeep, Beri, Raj, Thong, Bob, Wallace, Alan, Oreffo, Victor, Hutchinson, Ray, Harper, Steve, Debreczeni, Judit, Breed, Jason, Wissler, Lisa, Edman, Karl
Published in Journal of medicinal chemistry (27.03.2014)
Published in Journal of medicinal chemistry (27.03.2014)
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Journal Article
Chiral Phosphoric Acid-Catalyzed Enantioselective Three- Component Aza-Diels-Alder Reactions of Aminopyrroles and Aminopyrazoles
Brioche, Julien, Courant, Thibaut, Alcaraz, Lilian, Stocks, Michael, Furber, Mark, Zhu, Jieping, Masson, Géraldine
Published in Advanced synthesis & catalysis (26.05.2014)
Published in Advanced synthesis & catalysis (26.05.2014)
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The Discovery of MMP7 Inhibitors Exploiting a Novel Selectivity Trigger
Edman, Karl, Furber, Mark, Hemsley, Paul, Johansson, Cristian, Pairaudeau, Garry, Petersen, Jens, Stocks, Michael, Tervo, Anu, Ward, Alison, Wells, Edward, Wissler, Lisa
Published in ChemMedChem (02.05.2011)
Published in ChemMedChem (02.05.2011)
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Discovery of isoindoline and tetrahydroisoquinoline derivatives as potent, selective PPARδ agonists
Luckhurst, Christopher A., Stein, Linda A., Furber, Mark, Webb, Nicola, Ratcliffe, Marianne J., Allenby, Gary, Botterell, Sara, Tomlinson, Wendy, Martin, Barrie, Walding, Andrew
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
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Journal Article
Discovery of Potent and Selective Adamantane-Based Small-Molecule P2X 7 Receptor Antagonists/Interleukin-1β Inhibitors
Furber, Mark, Alcaraz, Lilian, Bent, Janice E., Beyerbach, Armin, Bowers, Keith, Braddock, Martin, Caffrey, Moya V., Cladingboel, David, Collington, John, Donald, David K., Fagura, Malbinder, Ince, Frank, Kinchin, Elizabeth C., Laurent, Celine, Lawson, Mandy, Luker, Timothy J., Mortimore, Michael M. P., Pimm, Austen D., Riley, Robert J., Roberts, Nicola, Robertson, Mark, Theaker, Jill, Thorne, Philip V., Weaver, Richard, Webborn, Peter, Willis, Paul
Published in Journal of medicinal chemistry (29.11.2007)
Published in Journal of medicinal chemistry (29.11.2007)
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Journal Article
Discovery of potent and selective adamantane-based small-molecule P2X(7) receptor antagonists/interleukin-1 beta,6 inhibitors
Furber, Mark, Alcaraz, Lilian, Bent, Janice E., Beyerbach, Armin, Bowers, Keith, Braddock, Martin, Caffrey, Moya V., Cladingboel, David, Collington, John, Donald, David K., Fagura, Malbinder, Ince, Frank, Kinchin, Elizabeth C., Laurent, Celine, Lawson, Mandy, Luker, Timothy J., Mortimore, Michael M. P., Pimm, Austen D., Riley, Robert J., Roberts, Nicola, Robertson, Mark, Theaker, Jill, Thorne, Philip V., Weaver, Richard, Webborn, Peter, Willis, Paul
Published in Journal of medicinal chemistry (29.11.2007)
Published in Journal of medicinal chemistry (29.11.2007)
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A Palladium-Catalyzed Synthesis of Amidines from Aryl Halides
Saluste, C. Gustaf, Whitby, Richard J., Furber, Mark
Published in Angewandte Chemie (International ed.) (17.11.2000)
Published in Angewandte Chemie (International ed.) (17.11.2000)
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Journal Article
Synthesis and biological evaluation of N-alkylated 8-oxybenz[c]azepine derivatives as selective PPARδ agonists
Luckhurst, Christopher A., Ratcliffe, Marianne, Stein, Linda, Furber, Mark, Botterell, Sara, Laughton, David, Tomlinson, Wendy, Weaver, Richard, Chohan, Kamaldeep, Walding, Andrew
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
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Journal Article
Discovery and evolution of phenoxypiperidine hydroxyamide dual CCR3/H-1 antagonists. Part II: Optimising in vivo clearance
Furber, Mark, Alcaraz, Lilian, Luckhurst, Christopher, Bahl, Ash, Beaton, Haydn, Bowers, Keith, Collington, John, Denton, Rebecca, Donald, David, Kinchin, Elizabeth, MacDonald, Cathy, Rigby, Aaron, Riley, Rob, Soars, Matt, Springthorpe, Brian, Webborn, Peter
Published in Bioorganic & medicinal chemistry letters (15.12.2012)
Published in Bioorganic & medicinal chemistry letters (15.12.2012)
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Journal Article
Discovery and evolution of phenoxypiperidine hydroxyamide dual CCR3/H-1 antagonists. Part I
Furber, Mark, Alcaraz, Lilian, Luckhurst, Christopher, Bahl, Ash, Beaton, Haydn, Bowers, Keith, Collington, John, Denton, Rebecca, Donald, David, Kinchin, Elizabeth, MacDonald, Cathy, Rigby, Aaron, Riley, Rob, Soars, Matt, Springthorpe, Brian, Webborn, Peter
Published in Bioorganic & medicinal chemistry letters (15.12.2012)
Published in Bioorganic & medicinal chemistry letters (15.12.2012)
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