Search Results - "MARIO G CARDOZO" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Synthesis and optimization of substituted furo[2,3-d]-pyrimidin-4-amines and 7H-pyrrolo[2,3-d]pyrimidin-4-amines as ACK1 inhibitors

Synthesis and optimization of substituted furo[2,3-d]-pyrimidin-4-amines and 7H-pyrrolo[2,3-d]pyrimidin-4-amines as ACK1 inhibitors

by Jiao, XianYun, Kopecky, David J., Liu, JinSong, Liu, JinQian, Jaen, Juan C., Cardozo, Mario G., Sharma, Rajiv, Walker, Nigel, Wesche, Holger, Li, Shyun, Farrelly, Ellyn, Xiao, Shou-Hua, Wang, Zhulun, Kayser, Frank
Published in Bioorganic & medicinal chemistry letters (01.10.2012)

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Journal Article

Observed bromodomain flexibility reveals histone peptide- and small molecule ligand-compatible forms of ATAD2

Observed bromodomain flexibility reveals histone peptide- and small molecule ligand-compatible forms of ATAD2

by Poncet-Montange, Guillaume, Zhan, Yanai, Bardenhagen, Jennifer P, Petrocchi, Alessia, Leo, Elisabetta, Shi, Xi, Lee, 4th, Gilbert R, Leonard, Paul G, Geck Do, Mary K, Cardozo, Mario G, Andersen, Jannik N, Palmer, Wylie S, Jones, Philip, Ladbury, John E
Published in Biochemical journal (01.03.2015)

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Discovery of potent and selective PKC-θ inhibitors

Discovery of potent and selective PKC-θ inhibitors

by Cywin, Charles L., Dahmann, Georg, Prokopowicz, Anthony S., Young, Erick R.R., Magolda, Ronald L., Cardozo, Mario G., Cogan, Derek A., DiSalvo, Darren, Ginn, John D., Kashem, Mohammed A., Wolak, John P., Homon, Carol A., Farrell, Thomas M., Grbic, Heather, Hu, Hanbo, Kaplita, Paul V., Liu, Lisa H., Spero, Denice M., Jeanfavre, Deborah D., O’Shea, Kathy M., White, Della M., Woska, Joseph R., Brown, Maryanne L.
Published in Bioorganic & medicinal chemistry letters (2007)

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Discovery of 2-Phenylamino-imidazo[4,5-h]isoquinolin-9-ones: A New Class of Inhibitors of Lck Kinase

Discovery of 2-Phenylamino-imidazo[4,5-h]isoquinolin-9-ones: A New Class of Inhibitors of Lck Kinase

by Snow, Roger J, Cardozo, Mario G, Morwick, Tina M, Busacca, Carl A, Dong, Yong, Eckner, Robert J, Jacober, Stephen, Jakes, Scott, Kapadia, Suresh, Lukas, Susan, Panzenbeck, Maret, Peet, Gregory W, Peterson, Jeffrey D, Prokopowicz, Anthony S, Sellati, Rosemarie, Tolbert, Robert M, Tschantz, Matt A, Moss, Neil
Published in Journal of medicinal chemistry (01.08.2002)

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Identification and optimization of N3,N6-diaryl-1H-pyrazolo[3,4-d]pyrimidine-3,6-diamines as a novel class of ACK1 inhibitors

Identification and optimization of N3,N6-diaryl-1H-pyrazolo[3,4-d]pyrimidine-3,6-diamines as a novel class of ACK1 inhibitors

by Kopecky, David J, Hao, Xiaolin, Chen, Yi, Fu, Jiasheng, Jiao, XianYun, Jaen, Juan C, Cardozo, Mario G, Liu, Jinsong, Wang, Zhulun, Walker, Nigel P C, Wesche, Holger, Li, Shyun, Farrelly, Ellyn, Xiao, Shou-Hua, Kayser, Frank
Published in Bioorganic & medicinal chemistry letters (15.12.2008)

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Journal Article

Optimization of 2-Phenylaminoimidazo[4,5-h]isoquinolin-9-ones: Orally Active Inhibitors of lck Kinase

Optimization of 2-Phenylaminoimidazo[4,5-h]isoquinolin-9-ones: Orally Active Inhibitors of lck Kinase

by Goldberg, Daniel R, Butz, Tanja, Cardozo, Mario G, Eckner, Robert J, Hammach, Abdelhakim, Huang, Jessica, Jakes, Scott, Kapadia, Suresh, Kashem, Mohammed, Lukas, Susan, Morwick, Tina M, Panzenbeck, Maret, Patel, Usha, Pav, Susan, Peet, Gregory W, Peterson, Jeffrey D, Prokopowicz, Anthony S, Snow, Roger J, Sellati, Rosemarie, Takahashi, Hidenori, Tan, Jonathan, Tschantz, Matt A, Wang, Xiao-Jun, Wang, Yong, Wolak, John, Xiong, Pla, Moss, Neil
Published in Journal of medicinal chemistry (10.04.2003)

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Conformational analyses and molecular-shape comparisons of a series of indanone-benzylpiperidine inhibitors of acetylcholinesterase

Conformational analyses and molecular-shape comparisons of a series of indanone-benzylpiperidine inhibitors of acetylcholinesterase

by Cardozo, Mario G, Kawai, Takatoshi, Iimura, Youichi, Sugimoto, Hachiro, Yamanishi, Yoshiharu, Hopfinger, A. J
Published in Journal of medicinal chemistry (01.02.1992)

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Journal Article

A Novel Frequency Distribution Selection Method for Efficient Plate Layout of a Diverse Combinatorial Library

A Novel Frequency Distribution Selection Method for Efficient Plate Layout of a Diverse Combinatorial Library

by Graham, Edward T, Jacober, Stephen P, Cardozo, Mario G
Published in Journal of Chemical Information and Computer Sciences (01.11.2001)

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Journal Article

Quantitative structure-activity relationship. QSAR, analyses of the substituted indanone and benzylpiperidine rings of a series of indanone-benzylpiperidine inhibitors of acetylcholinesterase. [Erratum to document cited in CA116(9):83138p]

Quantitative structure-activity relationship. QSAR, analyses of the substituted indanone and benzylpiperidine rings of a series of indanone-benzylpiperidine inhibitors of acetylcholinesterase. [Erratum to document cited in CA116(9):83138p]

by Cardozo, Mario G, Iimura, Youichi, Sugimoto, Hachiro, Yamanishi, Yoshiharu, Hopfinger, A. J
Published in Journal of medicinal chemistry (01.12.1992)

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Journal Article

Quantitative structure-activity relationship. QSAR, analyses of the substituted indanone and benzylpiperidine rings of a series of indanone-benzylpiperidine inhibitors of acetylcholinesterase

Quantitative structure-activity relationship. QSAR, analyses of the substituted indanone and benzylpiperidine rings of a series of indanone-benzylpiperidine inhibitors of acetylcholinesterase

by Cardozo, Mario G, Iimura, Youichi, Sugimoto, Hachiro, Yamanishi, Yoshiharu, Hopfinger, A. J
Published in Journal of medicinal chemistry (01.02.1992)

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Journal Article

A model for the dynemicin-A cleavage of DNA using molecular dynamics simulation

A model for the dynemicin-A cleavage of DNA using molecular dynamics simulation

by Cardozo, M G, Hopfinger, A J
Published in Biopolymers (01.03.1993)

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Journal Article

Conformational analyses and molecular-shape comparisons of a series of indanone-benzylpiperidine inhibitors of acetylcholinesterase. [Erratum to document cited in CA116(11):98893e]

Conformational analyses and molecular-shape comparisons of a series of indanone-benzylpiperidine inhibitors of acetylcholinesterase. [Erratum to document cited in CA116(11):98893e]

by Cardozo, Mario G, Kawai, Takatoshi, Iimura, Youichi, Sugimoto, Hachiro, Yamanishi, Yoshiharu, Hopfinger, A. J
Published in Journal of medicinal chemistry (01.12.1992)

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Journal Article

Identification and optimization of N super(3),N super(6)-diaryl-1H- pyrazolo[3,4-d]pyrimidine-3,6-diamines as a novel class of ACK1 inhibitors

Identification and optimization of N super(3),N super(6)-diaryl-1H- pyrazolo[3,4-d]pyrimidine-3,6-diamines as a novel class of ACK1 inhibitors

by Kopecky, David J, Hao, Xiaolin, Chen, Yi, Fu, Jiasheng, Jiao, XianYun, Jaen, Juan C, Cardozo, Mario G, Liu, Jinsong, Wang, Zhulun, Walker, Nigel PC, Wesche, Holger, Li, Shyun, Farrelly, Ellyn, Xiao, Shou-Hua, Kayser, Frank
Published in Bioorganic & medicinal chemistry (01.12.2008)

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Journal Article

Identification and optimization of N 3, N 6-diaryl-1 H-pyrazolo[3,4- d]pyrimidine-3,6-diamines as a novel class of ACK1 inhibitors

Identification and optimization of N 3, N 6-diaryl-1 H-pyrazolo[3,4- d]pyrimidine-3,6-diamines as a novel class of ACK1 inhibitors

by Kopecky, David J., Hao, Xiaolin, Chen, Yi, Fu, Jiasheng, Jiao, XianYun, Jaen, Juan C., Cardozo, Mario G., Liu, Jinsong, Wang, Zhulun, Walker, Nigel P.C., Wesche, Holger, Li, Shyun, Farrelly, Ellyn, Xiao, Shou-Hua, Kayser, Frank
Published in Bioorganic & medicinal chemistry letters (2008)

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Journal Article

LRRK2 INHIBITORS

LRRK2 INHIBITORS

by SWEENEY, Zachary K, GUO, Zuojun, MOREAU, Robert J, TULLY, David C, CARDOZO, Mario G
Year of Publication 16.11.2023

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Patent

LRRK2 INHIBITORS

LRRK2 INHIBITORS

by GUO, Zuojun, MOREAU, Robert J, TULLY, David C, CARDOZO, Mario G, RAJAPAKSA, Naomi S, RAO, Meera
Year of Publication 16.11.2023

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Patent

Identification and optimization of N3,N6-diaryl-lH-pyrazolo[3,4-d] pyrimidine-3,6-diamines as a novel class of ACK1 inhibitors

Identification and optimization of N3,N6-diaryl-lH-pyrazolo[3,4-d] pyrimidine-3,6-diamines as a novel class of ACK1 inhibitors

by KOPECKY, David J, XIAOLIN HAO, WESCHE, Holger, LI, Shyun, FARRELLY, Ellyn, XIAO, Shou-Hua, KAYSER, Frank, YI CHEN, JIASHENG FU, XIANYUN JIAO, JAEN, Juan C, CARDOZO, Mario G, JINSONG LIU, ZHULUN WANG, WALKER, Nigel P. C
Published in Bioorganic & medicinal chemistry letters (2008)

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Journal Article

Molecular modelling of ligand–DNA intercalation interactions

Molecular modelling of ligand–DNA intercalation interactions

by Hopfinger, A. J., Cardozo, Mario G., Kawakami, Y.
Published in Journal of the Chemical Society. Faraday transactions (1995)

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Journal Article

IMIDAZO(1,2-A)PYRIDINE DERIVATIVES AS RIPK2 INHIBITORS

IMIDAZO(1,2-A)PYRIDINE DERIVATIVES AS RIPK2 INHIBITORS

by SWEENEY, Zachary K, GUO, Zuojun, THEDE, Kai, CARDOZO, Mario G, TULLY, David C, MOREAU, Robert Joseph, RAJAPAKSA, Naomi S, GRESSIES, Steffen, RAO, Meera
Year of Publication 14.12.2023

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Patent

LRRK2 inhibitors

LRRK2 inhibitors

by MOREAU, ROBERT J, GUO, ZUOJUN, RAO, MEERA, TULLY, DAVID C, RAJAPAKSA, NAOMI S, CARDOZO, MARIO G
Year of Publication 01.03.2024

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Patent

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