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Genome-wide localization of small molecules
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Published in Nature biotechnology (01.01.2014)
Published in Nature biotechnology (01.01.2014)
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Catalytic site remodelling of the DOT1L methyltransferase by selective inhibitors
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Published in Nature communications (18.12.2012)
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Selective inhibition of CDK7 reveals high-confidence targets and new models for TFIIH function in transcription
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Biased Multicomponent Reactions to Develop Novel Bromodomain Inhibitors
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Structure-Guided DOT1L Probe Optimization by Label-Free Ligand Displacement
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7,9-Diaryl-1,6,8-trioxaspiro[4.5]dec-3-en-2-ones: Readily accessible and highly potent anticancer compounds
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Published in Bioorganic & medicinal chemistry letters (15.08.2014)
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Published in Nature communications (01.05.2013)
Published in Nature communications (01.05.2013)
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시클린-의존성 키나제 7 (CDK7)의 억제제
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Year of Publication 01.10.2021
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Year of Publication 01.10.2021
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시클린-의존성 키나제 7 (CDK7)의 억제제
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Year of Publication 09.04.2019
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7CDK7 INHIBITORS OF CYCLIN-DEPENDENT KINASE 7 CDK7
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Year of Publication 09.01.2017
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INHIBITORS OF TRANSCRIPTION FACTORS AND USES THEREOF
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Year of Publication 29.03.2016
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Year of Publication 29.03.2016
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Abstract 3230: Genome-wide localization of anti-cancer drugs
Anders, Lars, Guenther, Matthew G., Qi, Jun, Fan, Zi Peng, Marineau, Jason J., Rahl, Peter B., Lovén, Jakob, Sigova, Alla A., Smith, William B., Lee, Tong Ihn, Bradner, James E., Young, Richard A.
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Published in Cancer research (Chicago, Ill.) (01.10.2014)
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Genome-wide determination of drug localization
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Published in Nature biotechnology (15.12.2013)
Published in Nature biotechnology (15.12.2013)
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Correction: Corrigendum: Catalytic site remodelling of the DOT1L methyltransferase by selective inhibitors
Yu, Wenyu, Chory, Emma J., Wernimont, Amy K., Tempel, Wolfram, Scopton, Alex, Federation, Alexander, Marineau, Jason J., Qi, Jun, Barsyte-Lovejoy, Dalia, Yi, Joanna, Marcellus, Richard, Iacob, Roxana E., Engen, John R., Griffin, Carly, Aman, Ahmed, Wienholds, Erno, Li, Fengling, Pineda, Javier, Estiu, Guillermina, Shatseva, Tatiana, Hajian, Taraneh, Al-awar, Rima, Dick, John E., Vedadi, Masoud, Brown, Peter J., Arrowsmith, Cheryl H., Bradner, James E., Schapira, Matthieu
Published in Nature communications (21.05.2013)
Published in Nature communications (21.05.2013)
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