Pyrazolo[1',5':1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones as selective human A1 adenosine receptor ligands
GIOVANNONI, Maria Paola, VERGELLI, Claudia, GAVALDA, Amadeu, CILIBRIZZI, Agostino, CROCETTI, Letizia, BIANCALANI, Claudio, GRAZIANO, Alessia, DAL PIAZ, Vittorio, LOZA, Maria Isabel, CADAVID, Maria Isabel, DIAZ, José Luis
Published in Bioorganic & medicinal chemistry (15.11.2010)
Published in Bioorganic & medicinal chemistry (15.11.2010)
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Synthesis, enantioresolution, and activity profile of chiral 6-methyl-2,4-disubs-tituted pyridazin-3(2H)-ones as potent N-formyl peptide receptor agonists
Cilibrizzi, Agostino, Schepetkin, Igor A., Bartolucci, Gianluca, Crocetti, Letizia, Piaz, Vittorio Dal, Giovannoni, Maria Paola, Graziano, Alessia, Kirpotina, Liliya N., Quinn, Mark T., Vergelli, Claudia
Published in Bioorganic & medicinal chemistry (27.04.2012)
Published in Bioorganic & medicinal chemistry (27.04.2012)
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Pyrazolo[1',5':1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones as selective human A(1) adenosine receptor ligands
Giovannoni, Maria Paola, Vergelli, Claudia, Cilibrizzi, Agostino, Crocetti, Letizia, Biancalani, Claudio, Graziano, Alessia, Dal Piaz, Vittorio, Loza, Maria Isabel, Cadavid, Maria Isabel, Díaz, José Luis, Gavaldà, Amadeu
Published in Bioorganic & medicinal chemistry (15.11.2010)
Published in Bioorganic & medicinal chemistry (15.11.2010)
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4-Amino-5-substituted-3(2H)-pyridazinones as Orally Active Antinociceptive Agents: Synthesis and Studies on the Mechanism of Action
Giovannoni, Maria Paola, Cesari, Nicoletta, Vergelli, Claudia, Graziano, Alessia, Biancalani, Claudio, Biagini, Pierfrancesco, Ghelardini, Carla, Vivoli, Elisa, Dal Piaz, Vittorio
Published in Journal of medicinal chemistry (09.08.2007)
Published in Journal of medicinal chemistry (09.08.2007)
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Pyrazolo[1',5':1,6]pyrimido[4,5-d]pyridazin-4(3 H)-ones as selective human A sub(1) adenosine receptor ligands
Giovannoni, Maria Paola, Vergelli, Claudia, Cilibrizzi, Agostino, Crocetti, Letizia, Biancalani, Claudio, Graziano, Alessia, Piaz, Vittorio Dal, Loza, Maria Isabel, Cadavid, Maria Isabel, Diaz, Jose Luis, Gavalda, Amadeu
Published in Bioorganic & medicinal chemistry (15.11.2010)
Published in Bioorganic & medicinal chemistry (15.11.2010)
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4-Amino-5-vinyl-3(2 H)-pyridazinones and analogues as potent antinociceptive agents: Synthesis, SARs, and preliminary studies on the mechanism of action
Vergelli, Claudia, Giovannoni, Maria Paola, Pieretti, Stefano, Giannuario, Amalia Di, Piaz, Vittorio Dal, Biagini, Pierfrancesco, Biancalani, Claudio, Graziano, Alessia, Cesari, Nicoletta
Published in Bioorganic & medicinal chemistry (15.08.2007)
Published in Bioorganic & medicinal chemistry (15.08.2007)
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Journal Article
Pyrazolo[1′,5′:1,6]pyrimido[4,5- d]pyridazin-4(3 H)-ones as selective human A 1 adenosine receptor ligands
Giovannoni, Maria Paola, Vergelli, Claudia, Cilibrizzi, Agostino, Crocetti, Letizia, Biancalani, Claudio, Graziano, Alessia, Piaz, Vittorio Dal, Loza, Maria Isabel, Cadavid, Maria Isabel, Díaz, José Luis, Gavaldà, Amadeu
Published in Bioorganic & medicinal chemistry (2010)
Published in Bioorganic & medicinal chemistry (2010)
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New Pyrazolo[1',5':1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones Fluoroderivatives as Human A1 Adenosine Receptor Ligands
Graziano, Alessia, Giovannoni, Maria Paola, Cilibrizzi, Agostino, Crocetti, Letizia, Piaz, Vittorio Dal, Vergelli, Claudia, Trincavelli, Maria Letizia, Martini, Claudia, Giacomelli, Chiara
Published in Acta chimica Slovenica (01.09.2012)
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Published in Acta chimica Slovenica (01.09.2012)
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New pyrazolo[1′,5′:1,6]pyrimido[4,5- d]pyridazin-4(3 H)-ones as potent and selective PDE5 inhibitors
Feixas, Joan, Giovannoni, Maria Paola, Vergelli, Claudia, Gavaldà, Amadeu, Cesari, Nicoletta, Graziano, Alessia, Piaz, Vittorio Dal
Published in Bioorganic & medicinal chemistry letters (02.05.2005)
Published in Bioorganic & medicinal chemistry letters (02.05.2005)
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Alpha2-agonists as analgesic agents
Giovannoni, Maria Paola, Ghelardini, Carla, Vergelli, Claudia, Dal Piaz, Vittorio
Published in Medicinal research reviews (01.03.2009)
Published in Medicinal research reviews (01.03.2009)
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Design, synthesis and evaluation of N-benzoylindazole derivatives and analogues as inhibitors of human neutrophil elastase
CROCETTI, Letizia, GIOVANNONI, Maria Paola, SCHEPETKIN, Igor A, QUINN, Mark T, KHLEBNIKOV, Andrei I, CILIBRIZZI, Agostino, DAL PIAZ, Vittorio, GRAZIANO, Alessia, VERGELLI, Claudia
Published in Bioorganic & medicinal chemistry (2011)
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Published in Bioorganic & medicinal chemistry (2011)
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Novel Heterocyclic-Fused Pyridazinones as Potent and Selective Phosphodiesterase IV Inhibitors
Dal Piaz, Vittorio, Giovannoni, Maria Paola, Castellana, Carla, Palacios, José Maria, Beleta, Jorge, Doménech, Teresa, Segarra, Victor
Published in Journal of medicinal chemistry (09.05.1997)
Published in Journal of medicinal chemistry (09.05.1997)
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4-Amino-3(2 H)-pyridazinones bearing arylpiperazinylalkyl groups and related compounds: synthesis and antinociceptive activity
Piaz, Vittorio Dal, Vergelli, Claudia, Giovannoni, Maria Paola, Scheideler, Mark A, Petrone, Giuseppe, Zaratin, Paola
Published in Farmaco (Società chimica italiana : 1989) (01.11.2003)
Published in Farmaco (Società chimica italiana : 1989) (01.11.2003)
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5,6-Diphenylpyridazine Derivatives as Acyl-CoA:Cholesterol Acyltransferase Inhibitors
Giovannoni, Maria Paola, Piaz, Vittorio Dal, Kwon, Byoung-Mog, Kim, Mi-Kyung, Kim, Young-Kook, Toma, Lucio, Barlocco, Daniela, Bernini, Franco, Canavesi, Monica
Published in Journal of medicinal chemistry (22.11.2001)
Published in Journal of medicinal chemistry (22.11.2001)
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Repurposing strategies on pyridazinone-based series by pharmacophore- and structure-driven screening
Floresta, Giuseppe, Crocetti, Letizia, Giovannoni, Maria Paola, Biagini, Pierfrancesco, Cilibrizzi, Agostino
Published in Journal of Enzyme Inhibition and Medicinal Chemistry (01.01.2020)
Published in Journal of Enzyme Inhibition and Medicinal Chemistry (01.01.2020)
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Heterocyclic-fused 3(2H)-pyridazinones as potent and selective PDE IV inhibitors: Further structure-activity relationships and molecular modelling studies
Piaz, Vittorio Dal, Giovannoni, Maria Paola, Castellana, Carla, Palacios, José Maria, Beleta, Jorge, Doménech, Teresa, Segarra, Victor
Published in European journal of medicinal chemistry (01.10.1998)
Published in European journal of medicinal chemistry (01.10.1998)
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Synthesis and Evaluation of Some Pyrazolo[3,4-d]pyridazinones and Analogues as PDE 5 Inhibitors Potentially Useful as Peripheral Vasodilator Agents
Piaz, Vittorio Dal, Castellana, Maria Carla, Vergelli, Claudia, Giovannoni, Maria Paola, Gavaldà, Amadeu, Segarra, Victor, Beleta, Jorge, Ryder, Hamish, Palacios, Josè Maria
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2002)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2002)
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