Comparison of high pressure homogenization and stirred bead milling for the production of nano-crystalline suspensions
Nakach, Mostafa, Authelin, Jean-René, Perrin, Marc-Antoine, Lakkireddy, Harivardhan Reddy
Published in International journal of pharmaceutics (25.08.2018)
Published in International journal of pharmaceutics (25.08.2018)
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Journal Article
Crystal structure determination of the elusive paracetamol Form III
Perrin, Marc-Antoine, Neumann, Marcus A, Elmaleh, Hagit, Zaske, Lionel
Published in Chemical communications (Cambridge, England) (01.01.2009)
Published in Chemical communications (Cambridge, England) (01.01.2009)
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Journal Article
Differential Water Thermodynamics Determine PI3K-Beta/Delta Selectivity for Solvent-Exposed Ligand Modifications
Robinson, Daniel, Bertrand, Thomas, Carry, Jean-Christophe, Halley, Frank, Karlsson, Andreas, Mathieu, Magali, Minoux, Hervé, Perrin, Marc-Antoine, Robert, Benoit, Schio, Laurent, Sherman, Woody
Published in Journal of chemical information and modeling (23.05.2016)
Published in Journal of chemical information and modeling (23.05.2016)
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Journal Article
Rimonabant Dimorphism and Its Pressure–Temperature Phase Diagram: A Delicate Case of Overall Monotropic Behavior
Perrin, Marc-Antoine, Bauer, Michel, Barrio, Maria, Tamarit, Josep-Lluís, Céolin, René, Rietveld, Ivo B.
Published in Journal of pharmaceutical sciences (01.07.2013)
Published in Journal of pharmaceutical sciences (01.07.2013)
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Journal Article
Polymorphism of Progesterone: Relative Stabilities of the Orthorhombic Phases I and II Inferred from Topological and Experimental Pressure-Temperature Phase Diagrams
Barrio, Maria, Espeau, Philippe, Lluis Tamarit, Josep, Perrin, Marc-Antoine, Veglio, Nestor, Ceolin, René
Published in Journal of pharmaceutical sciences (01.05.2009)
Published in Journal of pharmaceutical sciences (01.05.2009)
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Journal Article
Polymorphism of paracetamol: Relative stabilities of the monoclinic and orthorhombic phases inferred from topological pressure‐temperature and temperature‐volume phase diagrams
Espeau, Philippe, Céolin, René, Tamarit, Josep‐Lluis, Perrin, Marc‐Antoine, Gauchi, Jean‐Pierre, Leveiller, Franck
Published in Journal of pharmaceutical sciences (01.03.2005)
Published in Journal of pharmaceutical sciences (01.03.2005)
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Journal Article
Liquid-Liquid Miscibility Gaps and Hydrate Formation in Drug-Water Binary Systems: Pressure-Temperature Phase Diagram of Lidocaine and Pressure-Temperature-Composition Phase Diagram of the Lidocaine-Water System
Ceolin, René, Barrio, Maria, Tamarit, Josep-Lluis, Veglio, Nestor, Perrin, Marc-Antoine, Espeau, Philippe
Published in Journal of pharmaceutical sciences (01.06.2010)
Published in Journal of pharmaceutical sciences (01.06.2010)
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Journal Article
Rhodium(III)-Catalyzed C–H Activation/Heterocyclization as a Macrocyclization Strategy. Synthesis of Macrocyclic Pyridones
Krieger, Jean-Philippe, Lesuisse, Dominique, Ricci, Gino, Perrin, Marc-Antoine, Meyer, Christophe, Cossy, Janine
Published in Organic letters (19.05.2017)
Published in Organic letters (19.05.2017)
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Journal Article
Overall Monotropic Behavior of a Metastable Phase of Biclotymol, 2,2′-Methylenebis(4-Chloro-3-Methyl-Isopropylphenol), Inferred From Experimental and Topological Construction of the Related P-T State Diagram
Céolin, René, Tamarit, Josep-Lluis, Barrio, Maria, López, David O., Nicolaï, Béatrice, Veglio, Nestor, Perrin, Marc-Antoine, Espeau, Philippe
Published in Journal of pharmaceutical sciences (01.09.2008)
Published in Journal of pharmaceutical sciences (01.09.2008)
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Journal Article
Total Synthesis of (+)-Oxo-tomaymycin
Benedetti, Françoise, Perrin, Marc-Antoine, Bosc, Sebastien, Chouteau, Franck, Champion, Nicolas, Bigot, Antony
Published in Organic process research & development (15.05.2020)
Published in Organic process research & development (15.05.2020)
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Journal Article
Ring Expansion of Cyclic β-Amino Alcohols Induced by Diethylaminosulfur Trifluoride: Synthesis of Cyclic Amines with a Tertiary Fluorine at C3
Anxionnat, Bruno, Robert, Benoit, George, Pascal, Ricci, Gino, Perrin, Marc-Antoine, Gomez Pardo, Domingo, Cossy, Janine
Published in Journal of organic chemistry (20.07.2012)
Published in Journal of organic chemistry (20.07.2012)
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Journal Article
Imidazopyrazinones (IPYs): Non-Quinolone Bacterial Topoisomerase Inhibitors Showing Partial Cross-Resistance with Quinolones
Jeannot, Frédéric, Taillier, Thomas, Despeyroux, Pierre, Renard, Stéphane, Rey, Astrid, Mourez, Michaël, Poeverlein, Christoph, Khichane, Imène, Perrin, Marc-Antoine, Versluys, Stéphanie, Stavenger, Robert A, Huang, Jianzhong, Germe, Thomas, Maxwell, Anthony, Cao, Sha, Huseby, Douglas L, Hughes, Diarmaid, Bacqué, Eric
Published in Journal of medicinal chemistry (26.04.2018)
Published in Journal of medicinal chemistry (26.04.2018)
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Journal Article
Discovery and Optimization of Pyrimidone Indoline Amide PI3Kβ Inhibitors for the Treatment of Phosphatase and Tensin Homologue (PTEN)-Deficient Cancers
Certal, Victor, Carry, Jean-Christophe, Halley, Frank, Virone-Oddos, Angela, Thompson, Fabienne, Filoche-Rommé, Bruno, El-Ahmad, Youssef, Karlsson, Andreas, Charrier, Véronique, Delorme, Cécile, Rak, Alexey, Abecassis, Pierre-Yves, Amara, Céline, Vincent, Loïc, Bonnevaux, Hélène, Nicolas, Jean-Paul, Mathieu, Magali, Bertrand, Thomas, Marquette, Jean-Pierre, Michot, Nadine, Benard, Tsiala, Perrin, Marc-Antoine, Lemaitre, Olivier, Guerif, Stephane, Perron, Sébastien, Monget, Sylvie, Gruss-Leleu, Florence, Doerflinger, Gilles, Guizani, Houlfa, Brollo, Maurice, Delbarre, Laurence, Bertin, Luc, Richepin, Patrick, Loyau, Véronique, Garcia-Echeverria, Carlos, Lengauer, Christoph, Schio, Laurent
Published in Journal of medicinal chemistry (13.02.2014)
Published in Journal of medicinal chemistry (13.02.2014)
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Journal Article
Revisiting the Blind Tests in Crystal Structure Prediction: Accurate Energy Ranking of Molecular Crystals
Asmadi, Aldi, Neumann, Marcus A, Kendrick, John, Girard, Pascale, Perrin, Marc-Antoine, Leusen, Frank J. J
Published in The journal of physical chemistry. B (24.12.2009)
Published in The journal of physical chemistry. B (24.12.2009)
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Journal Article
Crystal Structures and Phase Relationships of 2 Polymorphs of 1,4-Diazabicyclo[3.2.2]nonane-4-Carboxylic Acid 4-Bromophenyl Ester Fumarate, A Selective α-7 Nicotinic Receptor Partial Agonist
Robert, Benoît, Perrin, Marc-Antoine, Barrio, Maria, Tamarit, Josep-Lluis, Coquerel, Gérard, Ceolin, René, Rietveld, Ivo B.
Published in Journal of pharmaceutical sciences (01.01.2016)
Published in Journal of pharmaceutical sciences (01.01.2016)
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Journal Article
Solid-State Properties and Dehydration Behavior of the Active Pharmaceutical Ingredient Potassium Guaiacol-4-sulfonate
Mahé, Nathalie, Nicolaï, Béatrice, Barrio, Maria, Perrin, Marc-Antoine, Do, Bernard, Tamarit, Josep-Lluis, Céolin, René, Rietveld, Ivo B
Published in Crystal growth & design (03.07.2013)
Published in Crystal growth & design (03.07.2013)
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