Novel Small Molecule Tyrosine Kinase 2 Pseudokinase Ligands Block Cytokine-Induced TYK2-Mediated Signaling Pathways
Zhou, Yu, Li, Xin, Shen, Ru, Wang, Xiangzhu, Zhang, Fan, Liu, Suxing, Li, Di, Liu, Jian, Li, Puhui, Yan, Yinfa, Dong, Ping, Zhang, Zhigao, Wu, Heping, Zhuang, Linghang, Chowdhury, Rasheduzzaman, Miller, Matthew, Issa, Mena, Mao, Yuchang, Chen, Hongli, Feng, Jun, Li, Jing, Bai, Chang, He, Feng, Tao, Weikang
Published in Frontiers in immunology (20.05.2022)
Published in Frontiers in immunology (20.05.2022)
Get full text
Journal Article
Discovery of SHR5428 as a selective and noncovalent inhibitor of CDK7
Jia, Minqiang, Wang, Weimin, Chen, Gang, Wu, Ting, Zhang, Ting, Zhou, Qian, Yin, Junzhao, Li, Jie, Li, Xun, Mao, Yuchang, Feng, Jun, Hu, Min, Li, Xin, He, Feng
Published in Bioorganic & medicinal chemistry letters (01.09.2023)
Published in Bioorganic & medicinal chemistry letters (01.09.2023)
Get full text
Journal Article
Discovery of 2‑(Ortho-Substituted Benzyl)-Indole Derivatives as Potent and Orally Bioavailable RORγ Agonists with Antitumor Activity
Lu, Biao, Liu, Dong, Gui, Bin, Gou, Jun, Dong, Huaide, Hu, Qiyue, Feng, Jun, Mao, Yuchang, Shen, Xiaodong, Wang, Shenglan, Zhang, Caihua, Shen, Ru, Yan, Yinfa, Chen, Lei, Wang, Huiyun, Li, Di, Zhang, Jiayin, Zhang, Minsheng, Zhang, Rumin, Bai, Chang, He, Feng, Tao, Weikang, Liu, Suxing
Published in Journal of medicinal chemistry (28.10.2021)
Published in Journal of medicinal chemistry (28.10.2021)
Get full text
Journal Article
Discovery of spiro amide SHR902275: A potent, selective, and efficacious RAF inhibitor targeting RAS mutant cancers
Zhao, Peng, Zhuang, Linghang, Wang, Xiangzhu, Huang, Song, Wu, Heping, Zhou, Yu, Yan, Yuna, Zhang, Fan, Shen, Ru, Li, Jing, Liu, Suxing, Zhang, Rumin, Dong, Ping, Mao, Yuchang, Fan, Yuanmin, He, Chunyong, Sun, Jiakang, Zhang, Lei, Hu, Qiyue, Wan, Hong, Feng, Jun, Bai, Chang, He, Feng, Tao, Weikang
Published in European journal of medicinal chemistry (15.01.2022)
Published in European journal of medicinal chemistry (15.01.2022)
Get full text
Journal Article
Discovery of SHR2415, a Novel Pyrrole-Fused Urea Scaffold ERK1/2 Inhibitor
Li, Xin, Dong, Ping, Zhang, Ting, Cai, Guodong, Chen, Yang, Dong, Huaide, Yang, Fang, Zhang, Lei, Mao, Yuchang, Feng, Jun, Bai, Chang, He, Feng, Tao, Weikang
Published in ACS medicinal chemistry letters (14.04.2022)
Published in ACS medicinal chemistry letters (14.04.2022)
Get full text
Journal Article
Discovery of SHR5133, a Highly Potent and Novel HBV Capsid Assembly Modulator
Li, Xin, Zhang, Zhigao, Chen, Yang, Wang, Bin, Yang, Guimei, Xu, Xiangbin, Yechao, Baihui, Bai, Dongdong, Feng, Binqiang, Mao, Yuchang, Feng, Jun, Bai, Chang, He, Feng, Tao, Weikang
Published in ACS medicinal chemistry letters (10.03.2022)
Published in ACS medicinal chemistry letters (10.03.2022)
Get full text
Journal Article
Abstract 3146: HRA00130-C004, a novel anti-DLL3 ADC with bystander effect, high DAR and favorable safety profiles
Yao, Qingqing, Xue, Changding, Xu, Zhibin, You, Lingfeng, Xue, Zhendong, Mao, Yuchang, Lin, Sophie, Feng, Jun, Zhang, Zhe, Ye, Xin, Hu, Min, He, Feng
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Get full text
Journal Article
Abstract 7279: Discovery of SHR1127, an orally bioavailable, highly potent and selective KRAS G12D inhibitor
Li, Xin, Shen, Feng, Zhang, Limin, Wang, Wei, Kong, Luyao, Bao, Yong, Mao, Yuchang, Wang, Zaiyong, Lin, Sophie, Zhang, Zhe, Feng, Jun, Hu, Min, He, Feng
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Get full text
Journal Article
Abstract 3145: HRA00242-C004, a novel anti-PSMA ADC with high DAR reveals potent in vitro and in vivo anti-tumor efficacy
Lin, Guang, Zhang, Haoying, Xu, Zhibin, You, Lingfeng, Xue, Zhendong, Mao, Yuchang, Yang, Xiaoying, Hu, Bing, Lin, Sophie, Feng, Jun, Zhang, Zhe, Ye, Xin, Hu, Min, He, Feng
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Get full text
Journal Article
Abstract LB031: SHR-A1811, a novel anti-HER2 ADC with superior bystander effect, optimal DAR and favorable safety profiles
Zhang, Ting, You, Lingfeng, Xu, Jianyan, Yin, Junzhao, Qu, Bolei, Mao, Yuchang, Fu, Beibei, Cao, Dan, Zhao, Linda, Feng, Jun, Hu, Min, He, Feng
Published in Cancer research (Chicago, Ill.) (14.04.2023)
Published in Cancer research (Chicago, Ill.) (14.04.2023)
Get full text
Journal Article
Discovery of Isoindoline Amide Derivatives as Potent and Orally Bioavailable ADAMTS-4/5 Inhibitors for the Treatment of Osteoarthritis
Zhao, Peng, Liu, Dong, Song, Chunying, Li, Di, Zhang, Xinzhu, Horecny, Ivana, Zhang, Fengqi, Yan, Yuna, Zhuang, Linghang, Li, Jing, Liu, Suxing, Mao, Yuchang, Feng, Jun, Liu, Jian, Tao, Weikang
Published in ACS pharmacology & translational science (08.07.2022)
Published in ACS pharmacology & translational science (08.07.2022)
Get full text
Journal Article
Medicine for improving bioavailability of atorvastatin
WANG YINGJIE, SHEN ZHIJIE, WANG XIAOLONG, WANG BAIYANG, MAO YUCHANG, HU ZHUOHAN
Year of Publication 13.08.2014
Get full text
Year of Publication 13.08.2014
Patent
Medicine for improving bioavailability of atorvastatin
WANG YINGJIE, SHEN ZHIJIE, WANG XIAOLONG, WANG BAIYANG, MAO YUCHANG, HU ZHUOHAN
Year of Publication 09.01.2013
Get full text
Year of Publication 09.01.2013
Patent