KEAP1의 조정제로서의 시클릭 시아노에논 유도체
CANDITO DAVID A, CHRISTIAN ALEC H, DI PIETRO ORNELLA, LIU PING, PALANI ANANDAN, ST GALLAY STEPHEN, ALTMAN MICHAEL, MANSOOR UMAR FARUK, LU MIN, SHAW DAVID MATTHEW, MENNIE KATRINA MARIE, REUTERSHAN MICHAEL H, MUSACCHIO ANDREW J
Year of Publication 24.03.2023
Get full text
Year of Publication 24.03.2023
Patent
아데노신 수용체 길항제로서의 7-, 8- 및 10-치환된 아미노 트리아졸로 퀴나졸린 유도체, 제약 조성물 및 그의 용도
WANG HUIJUN, SWAMINATHAN UMA, ALI AMJAD, LARSEN MATTHEW A, LIU PING, PAN JIANPING, DENG QIAOLIN, MANSOOR UMAR FARUK, LIU KUN, CUMMING JARED, DEMONG DUANE, ZHANG YONGLIAN, PLUMMER CHRISTOPHER W, SATHER AARON, GRAHAM THOMAS H, HENNESSY ELISABETH
Year of Publication 06.08.2021
Get full text
Year of Publication 06.08.2021
Patent
아데노신 수용체 길항제로서의 9-치환된 아미노 트리아졸로 퀴나졸린 유도체, 제약 조성물 및 그의 용도
WANG HUIJUN, SWAMINATHAN UMA, ALI AMJAD, LARSEN MATTHEW A, LIU PING, PAN JIANPING, DENG QIAOLIN, MANSOOR UMAR FARUK, LIU KUN, CUMMING JARED, DEMONG DUANE, PLUMMER CHRISTOPHER W, SATHER AARON, ZHANG YONGLIAN, GRAHAM THOMAS H, HOOVER ANDREW J, HENNESSY ELISABETH
Year of Publication 04.08.2021
Get full text
Year of Publication 04.08.2021
Patent
Continuous Flow Enables Metallaphotoredox Catalysis in a Medicinal Chemistry Setting: Accelerated Optimization and Library Execution of a Reductive Coupling between Benzylic Chlorides and Aryl Bromides
Brill, Zachary G, Ritts, Casey B, Mansoor, Umar Faruk, Sciammetta, Nunzio
Published in Organic letters (17.01.2020)
Published in Organic letters (17.01.2020)
Get full text
Journal Article
Continuous-Flow Solid-Phase Peptide Synthesis to Enable Rapid, Multigram Deliveries of Peptides
Ruhl, Kyle E., Di Maso, Michael J., Rose, Harrison B., Schultz, Danielle M., Lévesque, François, Grosser, Shane T., Silverman, Steven M., Li, Shasha, Sciammetta, Nunzio, Mansoor, Umar Faruk
Published in Organic process research & development (19.07.2024)
Published in Organic process research & development (19.07.2024)
Get full text
Journal Article
NOVEL COMPOUNDS THAT ARE ERK INHIBITORS
WITTER DAVID J, O'BOYLE BRENDAN, BOYCE CHRISTOPHER, KURUKULASURIYA RAVI, SLOMAN DAVID, TONG LING, SHINKRE BIDHAN A, THATAI JAYANTH THIRUVELLORE, SILIPHAIVANH PHIENG, FALCONE DANIELLE, MANSOOR UMAR FARUK, ZHOU WEI, KARUNAKARAN GANESH BABU, FEVRIER SALEM, LIPFORD KATHRYN, METHOT JOEY L, CHEN LEI, MALETIC MILANA M, HUANG XIANHAI, KOZLOWSKI JOSEPH, DANIELS MATTHEW H, LIM, JONG WON, WILSON KEVIN J, BAKSHI RAMAN KUMAR
Year of Publication 03.06.2015
Get full text
Year of Publication 03.06.2015
Patent
Discovery of novel spiro 1,3,4-thiadiazolines as potent, orally bioavailable and brain penetrant KSP inhibitors
Mansoor, Umar Faruk, Angeles, Angie R., Dai, Chaoyang, Yang, Liping, Vitharana, Dilrukshi, Basso, Andrea D., Gray, Kimberly, Tang, Huadong, Liu, Ming, Liang, Lianzhu, Allbritton, Omaira, Siddiqui, M. Arshad
Published in Bioorganic & medicinal chemistry (15.05.2015)
Published in Bioorganic & medicinal chemistry (15.05.2015)
Get full text
Journal Article
COMPOUNDS FOR INHIBITING KSP KINESIN ACTIVITY
CHENG CLIFF, SIDDIQUI ARSHAD M, ANGELES ANGIE R, MANSOOR UMAR FARUK, SHIPPS GERALD W. JR, HUANG XIAOHUA, DAI CHAOYANG, YANG LIPING, VITHARANA LALALNTHI DILRUKSHI
Year of Publication 02.07.2010
Get full text
Year of Publication 02.07.2010
Patent
KDM5 INHIBITORS
FISCHER, Christian, MANSOOR, Umar Faruk, SILIPHAIVANH, Phieng, GUNAYDIN, Hakan
Year of Publication 18.03.2020
Get full text
Year of Publication 18.03.2020
Patent
9-substituted amino triazolo quinazoline derivatives as adenosine receptor antagonists, pharmaceutical compositions and their use
Swaminathan, Uma, Liu, Ping, Mansoor, Umar Faruk, Plummer, Christopher W, Wang, Huijun, Deng, Qiaolin, Sather, Aaron, Liu, Kun, Hoover, Andrew J, Ali, Amjad, Hennessy, Elisabeth, Pan, Jianping, DeMong, Duane, Graham, Thomas H, Larsen, Matthew A, Cumming, Jared, Zhang, Yonglian
Year of Publication 13.08.2024
Get full text
Year of Publication 13.08.2024
Patent
KDM5 INHIBITORS
Fischer, Christian, Gunaydin, Hakan, Siliphaivanh, Phieng, MANSOOR, UMAR FARUK
Year of Publication 13.02.2020
Get full text
Year of Publication 13.02.2020
Patent
ADENOSINE A2A AND A2B RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITIONS AND USE THEREOF
MORENO, Jesus, ALI, Amjad, PLUMMER, Christopher W, DEMONG, Duane E, CUMMING, Jared N, SATHER, Aaron C, HENNESSY, Elisabeth T, JOHNSON, Rebecca Elizabeth, LARSEN, Matthew A, KAPLAN, William P, LI, Derun, MANSOOR, Umar Faruk, DENG, Qiaolin
Year of Publication 06.06.2024
Get full text
Year of Publication 06.06.2024
Patent
9-SUBSTITUTED AMINO TRIAZOLO QUINAZOLINE DERIVATIVES AS ADENOSINE RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITIONS AND THEIR USE
SATHER, AARON, LARSEN, MATTHEW A, HENNESSY, ELISABETH, HOOVER, ANDREW J, ZHANG, YONGLIAN, MANSOOR, UMAR FARUK, ALI, AMJAD, DENG, QIAOLIN, LIU, PING, CUMMING, JARED, GRAHAM, THOMAS H, DEMONG, DUANE, PAN, JIANPING, SWAMINATHAN, UMA, LIU, KUN, PLUMMER, CHRISTOPHER W, WANG, HUIJUN
Year of Publication 07.05.2024
Get full text
Year of Publication 07.05.2024
Patent
ADENOSINE A2A AND A2B RECEPTOR DUAL ANTAGONISTS FOR IMMUNO-ONCOLOGY
Swaminathan, Uma, Hennessy, Elisabeth T, Mansoor, Umar Faruk, Wu, Heping, Ye, Yingchun, Kelly, Joseph M, Yu, Younong, Lo, Michael Man-Chu, Cumming, Jared N, Ali, Amjad, DeMong, Duane, Kuang, Rongze, Graham, Thomas H, Moreno, Jesus, De Lera Ruiz, Manuel
Year of Publication 07.03.2024
Get full text
Year of Publication 07.03.2024
Patent
KDM5 INHIBITORS
FISCHER, Christian, MANSOOR, Umar Faruk, SILIPHAIVANH, Phieng, GUNAYDIN, Hakan
Year of Publication 21.08.2019
Get full text
Year of Publication 21.08.2019
Patent
Cyclic cyanoenone derivatives as modulators of KEAP1
LU, Min, PALANI, Anandan, SHAW, David Matthew, MUSACCHIO, Andrew J, ALTMAN, Michael, CANDITO, David A, REUTERSHAN, Michael H, DI PIETRO, Ornella, ST-GALLAY, Stephen, MENNIE, Katrina Marie, CHRISTIAN, Alec H, LIU, Ping, MANSOOR, Umar Faruk
Year of Publication 08.02.2024
Get full text
Year of Publication 08.02.2024
Patent
Cyclic cyanoenone derivatives as modulators of KEAP1
LU, Min, PALANI, Anandan, SHAW, David Matthew, MUSACCHIO, Andrew J, ALTMAN, Michael, CANDITO, David A, REUTERSHAN, Michael H, DI PIETRO, Ornella, ST-GALLAY, Stephen, MENNIE, Katrina Marie, CHRISTIAN, Alec H, LIU, Ping, MANSOOR, Umar Faruk
Year of Publication 07.12.2023
Get full text
Year of Publication 07.12.2023
Patent