Discovery of a Selective Inhibitor of Oncogenic B-Raf Kinase with Potent Antimelanoma Activity
Tsai, James, Lee, John T., Wang, Weiru, Zhang, Jiazhong, Cho, Hanna, Mamo, Shumeye, Bremer, Ryan, Gillette, Sam, Kong, Jun, Haass, Nikolas K., Sproesser, Katrin, Li, Ling, Smalley, Keiran S. M., Fong, Daniel, Zhu, Yong-Liang, Marimuthu, Adhirai, Nguyen, Hoa, Lam, Billy, Liu, Jennifer, Cheung, Ivana, Rice, Julie, Suzuki, Yoshihisa, Luu, Catherine, Settachatgul, Calvin, Shellooe, Rafe, Cantwell, John, Kim, Sung-Hou, Schlessinger, Joseph, Zhang, Kam Y. J., West, Brian L., Powell, Ben, Habets, Gaston, Zhang, Chao, Ibrahim, Prabha N., Hirth, Peter, Artis, Dean R., Herlyn, Meenhard, Bollag, Gideon
Published in Proceedings of the National Academy of Sciences - PNAS (26.02.2008)
Published in Proceedings of the National Academy of Sciences - PNAS (26.02.2008)
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Journal Article
Design, Synthesis, and Crystal Structure of Hydroxyethyl Secondary Amine-Based Peptidomimetic Inhibitors of Human β-Secretase
Maillard, Michel C, Hom, Roy K, Benson, Timothy E, Moon, Joseph B, Mamo, Shumeye, Bienkowski, Michael, Tomasselli, Alfredo G, Woods, Danielle D, Prince, D. Bryan, Paddock, Donna J, Emmons, Thomas L, Tucker, John A, Dappen, Michael S, Brogley, Louis, Thorsett, Eugene D, Jewett, Nancy, Sinha, Sukanto, John, Varghese
Published in Journal of medicinal chemistry (22.02.2007)
Published in Journal of medicinal chemistry (22.02.2007)
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Journal Article
Design and Synthesis of Hydroxyethylene-Based Peptidomimetic Inhibitors of Human β-Secretase
Hom, Roy K, Gailunas, Andrea F, Mamo, Shumeye, Fang, Larry Y, Tung, Jay S, Walker, Donald E, Davis, David, Thorsett, Eugene D, Jewett, Nancy E, Moon, Joseph B, John, Varghese
Published in Journal of medicinal chemistry (01.01.2004)
Published in Journal of medicinal chemistry (01.01.2004)
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Journal Article
Design of Substrate-Based Inhibitors of Human β-Secretase
Tung, Jay S, Davis, David L, Anderson, John P, Walker, Don E, Mamo, Shumeye, Jewett, Nancy, Hom, Roy K, Sinha, Sukanto, Thorsett, Eugene D, John, Varghese
Published in Journal of medicinal chemistry (17.01.2002)
Published in Journal of medicinal chemistry (17.01.2002)
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Journal Article
Design and Synthesis of Statine-Based Cell-Permeable Peptidomimetic Inhibitors of Human β-Secretase
Hom, Roy K, Fang, Larry Y, Mamo, Shumeye, Tung, Jay S, Guinn, Ashley C, Walker, Don E, Davis, David L, Gailunas, Andrea F, Thorsett, Eugene D, Sinha, Sukanto, Knops, Jeroen E, Jewett, Nancy E, Anderson, John P, John, Varghese
Published in Journal of medicinal chemistry (08.05.2003)
Published in Journal of medicinal chemistry (08.05.2003)
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Journal Article
PYRROLO[2,3-B]PYRIDINE DERIVATIVES AS KINASE MODULATORS
ZHU HONGYAO, MAMO SHUMEYE, SPEVAK WAYNE, CHO HANNA, SHI SHENGHUA, IBRAHIM PRABHA N, GILLETTE SAM
Year of Publication 09.09.2009
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Year of Publication 09.09.2009
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