Efficacy of Chemokine Receptor Inhibition in Treating IL-36α-Induced Psoriasiform Inflammation
Campbell, James J, Ebsworth, Karen, Ertl, Linda S, McMahon, Jeffrey P, Wang, Yu, Yau, Simon, Mali, Venkat R, Chhina, Vicky, Kumamoto, Alice, Liu, Shirley, Dang, Ton, Newland, Dale, Charo, Israel F, Zhang, Penglie, Schall, Thomas J, Singh, Rajinder
Published in The Journal of immunology (1950) (15.03.2019)
Published in The Journal of immunology (1950) (15.03.2019)
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CCX559 is a potent, orally-administered small molecule PD-L1 inhibitor that induces anti-tumor immunity
Sullivan, Kathleen M C, Vilalta, Marta, Ertl, Linda S, Wang, Yu, Dunlap, Carolyn, Ebsworth, Karen, Zhao, Bin N, Li, Shijie, Zeng, Yibin, Miao, Zhenhua, Fan, Pingchen, Mali, Venkat, Lange, Christopher, McMurtrie, Darren, Yang, Ju, Lui, Rebecca, Scamp, Ryan, Chhina, Vicky, Kumamoto, Alice, Yau, Simon, Dang, Ton, Easterday, Ashton, Liu, Shirley, Miao, Shichang, Charo, Israel, Schall, Thomas J, Zhang, Penglie
Published in PloS one (07.06.2023)
Published in PloS one (07.06.2023)
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The Second Total Synthesis of Diazonamide A
Nicolaou, K. C., Bheema Rao, Paraselli, Hao, Junliang, Reddy, Mali Venkat, Rassias, Gerasimos, Huang, Xianhai, Chen, David Y.-K., Snyder, Scott A.
Published in Angewandte Chemie (International ed.) (17.04.2003)
Published in Angewandte Chemie (International ed.) (17.04.2003)
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Synthesis and Biological Evaluation of a Series of Liver-Selective Phosphonic Acid Thyroid Hormone Receptor Agonists and Their Prodrugs
Boyer, Serge H, Jiang, Hongjian, Jacintho, Jason D, Reddy, Mali Venkat, Li, Haiqing, Li, Wenyu, Godwin, Jennifer L, Schulz, William G, Cable, Edward E, Hou, Jinzhao, Wu, Rongrong, Fujitaki, James M, Hecker, Scott J, Erion, Mark D
Published in Journal of medicinal chemistry (27.11.2008)
Published in Journal of medicinal chemistry (27.11.2008)
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Cereblon-based Bifunctional Degrader of SOS1, BTX-6654, Targets Multiple KRAS Mutations and Inhibits Tumor Growth
Begovich, Kyle, Schoolmeesters, Angela, Rajapakse, Navin, Martinez-Terroba, Elena, Kumar, Maneesh, Shakya, Arvind, Lai, Chon, Greene, Steven, Whitefield, Brandon, Okano, Akinori, Mali, Venkat, Huang, Shenlin, Chourasia, Aparajita H, Fung, Leah
Published in Molecular cancer therapeutics (02.04.2024)
Published in Molecular cancer therapeutics (02.04.2024)
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Development of bifunctional CRBN-SOS1 degraders for treatment of mutant KRAS cancers
Begovich, Kyle, Schoolmeesters, Angela, Rajapakse, Navin, Kumar, Maneesh, Martinez-Terroba, Elena, Shakya, Arvind, Whitefield, Brandon, Mali, Venkat, Pagadala, Nataraj, Okano, Akinori, Huang, Shenlin, Chourasia, Aparajita Hoskote, Fung, Leah M.
Published in Journal of clinical oncology (01.06.2023)
Published in Journal of clinical oncology (01.06.2023)
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Abstract 6056: Identification of first-in-class, orally bioavailable SOS1 bifunctional degraders for the treatment of KRAS- and RTK-driven cancers
Begovich, Kyle, Schoolmeesters, Angela, Rajapakse, Navin, Martinez, Elena, Liu, Qiao, Shakya, Arvind, Okano, Akinori, Mali, Venkat, Huang, Shenlin, Chourasia, Aparajita, Fung, Leah
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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Targeting Chemokine Receptors CCR6 and CXCR2 in A Murine Model Of IL-36a-Induced Pustular Psoriasis
Campbell, James J, Ebsworth, Karen, Ertl, Linda, McMahon, Jeffrey P, Wang, Yu, Yau, Simon, Mali, Venkat R, Chhina, Vicky, Kumamoto, Alice, Liu, Shirley, Dang, Ton, Newland, Dale, Charo, Israel F, Zhang, Penglie, Schall, Thomas J, Singh, Rajinder
Published in The Journal of immunology (1950) (01.05.2019)
Published in The Journal of immunology (1950) (01.05.2019)
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Abstract 1745: Inhibition of chemokine receptor 2 (CCR2) with a small molecule antagonist enhances the effectiveness of checkpoint inhibition by altering the tumor microenvironment in mouse colorectal tumors: Reducing tumor size and increasing long term survival
Campbell, James J., Janson, Christine, Ertl, Linda, Li, Chris, Miao, Zhenhua, Krasinski, Antoni, Lui, Rebecca, Mali, Venkat, McMahon, Jeffrey, Zheng, Yibin, Wang, Yu, Zang, Xiaoping, Chhina, Vicky, Vilalta, Marta, Kumamoto, Alice, Dang, Ton, Liu, Shirley, Yao, Simon, Zhang, Penglie, Schall, Thomas J., Singh, Rajinder
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Year of Publication 14.12.2020
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Year of Publication 14.12.2020
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Year of Publication 22.09.2020
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PUNNA SREENIVAS, SINGH RAJINDER, YANG JU, ZHANG PENGLIE, ROTH HOWARD S, MCMURTRIE DARREN J, MALATHONG VIENGKHAM, MALI VENKAT REDDY
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Year of Publication 24.01.2022
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Year of Publication 24.01.2022
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PUNNA SREENIVAS, TANAKA HIROKO, FAN PINGCHEN, ZHANG PENGLIE, LANGE CHRISTOPHER W, ZENG YIBIN, MALATHONG VIENGKHAM, MALI VENKAT REDDY
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PUNNA SREENIVAS, FAN PINGCHEN, ZHANG PENGLIE, MIAO SHICHANG, STELLA VALENTINO J, SONG YANG, ZENG YIBIN, KRASINSKI ANTONI, MALI VENKAT REDDY
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Year of Publication 11.07.2019
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