Getting a Handle on Neuropharmacology by Targeting Receptor-Associated Proteins
Maher, Michael P., Matta, Jose A., Gu, Shenyan, Seierstad, Mark, Bredt, David S.
Published in Neuron (Cambridge, Mass.) (06.12.2017)
Published in Neuron (Cambridge, Mass.) (06.12.2017)
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Journal Article
Molecular determinants of ASIC1 modulation by divalent cations
Liu, Yi, Ma, Jichun, DesJarlais, Renee L, Hagan, Rebecca, Rech, Jason, Liu, Changlu, Miller, Robyn, Schoellerman, Jeffrey, Luo, Jinquan, Letavic, Michael, Grasberger, Bruce, Maher, Michael P
Published in Scientific reports (28.01.2024)
Published in Scientific reports (28.01.2024)
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Journal Article
Development of phenotypic assays for identifying novel blockers of L-type calcium channels in neurons
Hagan, Rebecca, Rex, Elizabeth, Woody, David, Milewski, Monika, Glaza, Thomas, Maher, Michael P, Liu, Yi
Published in Scientific reports (11.01.2021)
Published in Scientific reports (11.01.2021)
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Journal Article
Characterization of voltage-gated sodium-channel blockers by electrical stimulation and fluorescence detection of membrane potential
González, Jesús E, Huang, Chien-Jung, Harootunian, Alec, Maher, Michael P, Quan, Catherine, Raj, Christopher D, McCormack, Ken, Numann, Randal, Negulescu, Paul A
Published in Nature biotechnology (01.04.2006)
Published in Nature biotechnology (01.04.2006)
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Journal Article
Pharmacology and Antitussive Efficacy of 4-(3-Trifluoromethyl-pyridin-2-yl)-piperazine-1-carboxylic Acid (5-Trifluoromethyl-pyridin-2-yl)-amide (JNJ17203212), a Transient Receptor Potential Vanilloid 1 Antagonist in Guinea Pigs
Bhattacharya, Anindya, Scott, Brian P, Nasser, Nadia, Ao, Hong, Maher, Michael P, Dubin, Adrienne E, Swanson, Devin M, Shankley, Nigel P, Wickenden, Alan D, Chaplan, Sandra R
Published in The Journal of pharmacology and experimental therapeutics (01.11.2007)
Published in The Journal of pharmacology and experimental therapeutics (01.11.2007)
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Journal Article
Characterization of 2-(2,6-dichloro-benzyl)-thiazolo[5,4- d]pyrimidin-7-yl]-(4-trifluoromethyl-phenyl)-amine (JNJ-39729209) as a novel TRPV1 antagonist
Maher, Michael P., Bhattacharya, Anindya, Ao, Hong, Swanson, Nadia, Wu, Nyan-Tsz, Freedman, Jamie, Kansagara, Mena, Scott, Brian, Li, Dong H., Eckert, William A., Liu, Yi, Sepassi, Kia, Rizzolio, Michele, Fitzgerald, Anne, Liu, Jing, Branstetter, Bryan J., Rech, Jason C., Lebsack, Alec D., Breitenbucher, J. Guy, Wickenden, Alan D., Chaplan, Sandra R.
Published in European journal of pharmacology (01.08.2011)
Published in European journal of pharmacology (01.08.2011)
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Journal Article
High-throughput-compatible assays using a genetically-encoded calcium indicator
Wu, Nyantsz, Nishioka, Walter K, Derecki, Noël C, Maher, Michael P
Published in Scientific reports (03.09.2019)
Published in Scientific reports (03.09.2019)
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Journal Article
Discovery and Characterization of AMPA Receptor Modulators Selective for TARP-γ8
Maher, Michael P, Wu, Nyantsz, Ravula, Suchitra, Ameriks, Michael K, Savall, Brad M, Liu, Changlu, Lord, Brian, Wyatt, Ryan M, Matta, Jose A, Dugovic, Christine, Yun, Sujin, Ver Donck, Luc, Steckler, Thomas, Wickenden, Alan D, Carruthers, Nicholas I, Lovenberg, Timothy W
Published in The Journal of pharmacology and experimental therapeutics (01.05.2016)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2016)
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Journal Article
Recent advances in the biology and medicinal chemistry of TRPA1
Rech, Jason C, Eckert, William A, Maher, Michael P, Banke, Tue, Bhattacharya, Anindya, Wickenden, Alan D
Published in Future medicinal chemistry (01.05.2010)
Published in Future medicinal chemistry (01.05.2010)
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Journal Article
Targeting the Ion Channel Kv1.3 with Scorpion Venom Peptides Engineered for Potency, Selectivity, and Half-life
Edwards, Wilson, Fung-Leung, Wai-Ping, Huang, Chichi, Chi, Ellen, Wu, Nancy, Liu, Yi, Maher, Michael P., Bonesteel, Rachelle, Connor, Judith, Fellows, Ross, Garcia, Elena, Lee, Jerry, Lu, Lu, Ngo, Karen, Scott, Brian, Zhou, Hong, Swanson, Ronald V., Wickenden, Alan D.
Published in The Journal of biological chemistry (15.08.2014)
Published in The Journal of biological chemistry (15.08.2014)
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Journal Article
Discovery of Imidazo[1,2‑a]pyrazines and Pyrazolo[1,5‑c]pyrimidines as TARP γ‑8 Selective AMPAR Negative Modulators
Savall, Brad M, Wu, Dongpei, Swanson, Devin M, Seierstad, Mark, Wu, Nyantsz, Vives Martinez, Jorge, García Olmos, Beatriz, Lord, Brian, Coe, Kevin, Koudriakova, Tatiana, Lovenberg, Timothy W, Carruthers, Nicholas I, Maher, Michael P, Ameriks, Michael K
Published in ACS medicinal chemistry letters (14.03.2019)
Published in ACS medicinal chemistry letters (14.03.2019)
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Journal Article
Lead Optimization of 5‑Aryl Benzimidazolone- and Oxindole-Based AMPA Receptor Modulators Selective for TARP γ‑8
Ravula, Suchitra, Savall, Brad M, Wu, Nyantsz, Lord, Brian, Coe, Kevin, Wang, Kai, Seierstad, Mark, Swanson, Devin M, Ziff, Jeannie, Nguyen, Minh, Leung, Perry, Rynberg, Ray, La, David, Pippel, Daniel J, Koudriakova, Tatiana, Lovenberg, Timothy W, Carruthers, Nicholas I, Maher, Michael P, Ameriks, Michael K
Published in ACS medicinal chemistry letters (09.08.2018)
Published in ACS medicinal chemistry letters (09.08.2018)
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Journal Article
pH-Insensitive FRET voltage dyes
Maher, Michael P, Wu, Nyan-Tsz, Ao, Hong
Published in Journal of biomolecular screening (01.08.2007)
Published in Journal of biomolecular screening (01.08.2007)
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Journal Article
Discovery and synthesis of 6,7,8,9-tetrahydro-5H-pyrimido-[4,5-d]azepines as novel TRPV1 antagonists
HAWRYLUK, Natalie A, MERIT, Jeffrey E, FREEDMAN, Jamie M, SCOTT, Brian P, WICKENDEN, Alan D, CHAPLAN, Sandra R, BREITENBUCHER, J. Guy, LEBSACK, Alec D, BRANSTETTER, Bryan J, HACK, Michael D, SWANSON, Nadia, HONG AO, MAHER, Michael P, BHATTACHARYA, Anindya, QI WANG
Published in Bioorganic & medicinal chemistry letters (01.12.2010)
Published in Bioorganic & medicinal chemistry letters (01.12.2010)
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Journal Article
Identification and synthesis of 2,7-diamino-thiazolo[5,4- d]pyrimidine derivatives as TRPV1 antagonists
Lebsack, Alec D., Branstetter, Bryan J., Hack, Michael D., Xiao, Wei, Peterson, Matthew L., Nasser, Nadia, Maher, Michael P., Ao, Hong, Bhattacharya, Anindya, Kansagara, Mena, Scott, Brian P., Luo, Lin, Rynberg, Raymond, Rizzolio, Michele, Chaplan, Sandra R., Wickenden, Alan D., Guy Breitenbucher, J.
Published in Bioorganic & medicinal chemistry letters (2009)
Published in Bioorganic & medicinal chemistry letters (2009)
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Journal Article
1,2-Diamino-ethane-substituted-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepines as TRPV1 antagonists with improved properties
LEBSACK, Alec D, RECH, Jason C, HONG AO, MAHER, Michael P, HERRMANN, Michelle, FREEDMAN, Jamie, SCOTT, Brian P, LIN LUO, BHATTACHARYA, Anindya, QI WANG, CHAPLAN, Sandra R, WICKENDEN, Alan D, BRANSTETTER, Bryan J, BREITENBUCHER, J. Guy, HAWRYLUK, Natalie A, MERIT, Jeffrey E, ALLISON, Brett, RYNBERG, Raymond, BUMA, Johnathan, RIZZOLIO, Michele, SWANSON, Nadia
Published in Bioorganic & medicinal chemistry letters (01.12.2010)
Published in Bioorganic & medicinal chemistry letters (01.12.2010)
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Journal Article
HCN channels as targets for drug discovery
Maher, Michael P, Wu, Nyan-Tsz, Guo, Hong-Qing, Dubin, Adrienne E, Chaplan, Sandra R, Wickenden, Alan D
Published in Combinatorial chemistry & high throughput screening (01.01.2009)
Published in Combinatorial chemistry & high throughput screening (01.01.2009)
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Journal Article
The neurochip: a new multielectrode device for stimulating and recording from cultured neurons
Maher, MichaelP, Pine, Jerome, Wright, John, Tai, Yu-Chong
Published in Journal of neuroscience methods (01.02.1999)
Published in Journal of neuroscience methods (01.02.1999)
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