Ligands for Glutamate Receptors: Design and Therapeutic Prospects
Bräuner-Osborne, Hans, Egebjerg, Jan, Nielsen, Elsebet Ø, Madsen, Ulf, Krogsgaard-Larsen, Povl
Published in Journal of medicinal chemistry (13.07.2000)
Published in Journal of medicinal chemistry (13.07.2000)
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Bioisosteric Modifications of 2-Arylureidobenzoic Acids: Selective Noncompetitive Antagonists for the Homomeric Kainate Receptor Subtype GluR5
Valgeirsson, Jon, Nielsen, Elsebet Ø, Peters, Dan, Mathiesen, Claus, Kristensen, Anders S, Madsen, Ulf
Published in Journal of medicinal chemistry (30.12.2004)
Published in Journal of medicinal chemistry (30.12.2004)
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Design, Synthesis, and Pharmacology of a Highly Subtype-Selective GluR1/2 Agonist, (RS)-2-Amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)propionic Acid (Cl-HIBO)
Bjerrum, Esben J, Kristensen, Anders S, Pickering, Darryl S, Greenwood, Jeremy R, Nielsen, Birgitte, Liljefors, Tommy, Schousboe, Arne, Bräuner-Osborne, Hans, Madsen, Ulf
Published in Journal of medicinal chemistry (22.05.2003)
Published in Journal of medicinal chemistry (22.05.2003)
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The AMPA Receptor Binding Site: Focus on Agonists and Competitive Antagonists
Stensbol, Tine, Madsen, Ulf, Krogsgaard-Larsen, Povl
Published in Current pharmaceutical design (01.05.2002)
Published in Current pharmaceutical design (01.05.2002)
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Novel 1-Hydroxyazole Bioisosteres of Glutamic Acid. Synthesis, Protolytic Properties, and Pharmacology
Stensbøl, Tine B, Uhlmann, Peter, Morel, Sandrine, Eriksen, Birgitte L, Felding, Jakob, Kromann, Hasse, Hermit, Mette B, Greenwood, Jeremy R, Braüner-Osborne, Hans, Madsen, Ulf, Junager, Finn, Krogsgaard-Larsen, Povl, Begtrup, Mikael, Vedsø, Per
Published in Journal of medicinal chemistry (03.01.2002)
Published in Journal of medicinal chemistry (03.01.2002)
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(S)-Homo-AMPA, a Specific Agonist at the mGlu6 Subtype of Metabotropic Glutamic Acid Receptors
Ahmadian, Haleh, Nielsen, Birgitte, Bräuner-Osborne, Hans, Johansen, Tommy N, Stensbøl, Tine B, Sløk, Frank A, Sekiyama, Naohiro, Nakanishi, Shigetada, Krogsgaard-Larsen, Povl, Madsen, Ulf
Published in Journal of medicinal chemistry (24.10.1997)
Published in Journal of medicinal chemistry (24.10.1997)
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Partial Agonism and Antagonism of the Ionotropic Glutamate Receptor iGLuR5
Hald, Helle, Naur, Peter, Pickering, Darryl S., Sprogøe, Desiree, Madsen, Ulf, Timmermann, Daniel B., Ahring, Philip K., Liljefors, Tommy, Schousboe, Arne, Egebjerg, Jan, Gajhede, Michael, Kastrup, Jette Sandholm
Published in The Journal of biological chemistry (31.08.2007)
Published in The Journal of biological chemistry (31.08.2007)
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N-Methyl-d-aspartic Acid Receptor Agonists: Resolution, Absolute Stereochemistry, and Pharmacology of the Enantiomers of 2-Amino-2-(3-hydroxy-5-methyl-4-isoxazolyl)acetic Acid
Madsen, Ulf, Frydenvang, Karla, Ebert, Bjarke, Johansen, Tommy N, Brehm, Lotte, Krogsgaard-Larsen, Povl
Published in Journal of medicinal chemistry (05.01.1996)
Published in Journal of medicinal chemistry (05.01.1996)
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Synthesis of new isoxazoline-based acidic amino acids and investigation of their affinity and selectivity profile at ionotropic glutamate receptors
Pinto, Andrea, Conti, Paola, Grazioso, Giovanni, Tamborini, Lucia, Madsen, Ulf, Nielsen, Birgitte, De Micheli, Carlo
Published in European journal of medicinal chemistry (01.02.2011)
Published in European journal of medicinal chemistry (01.02.2011)
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Pharmacological characterization and modeling of the binding sites of novel 1,3-bis(pyridinylethynyl)benzenes as metabotropic glutamate receptor 5-selective negative allosteric modulators
Mølck, Christina, Harpsøe, Kasper, Gloriam, David E, Clausen, Rasmus P, Madsen, Ulf, Pedersen, Lars Ø, Jimenez, Hermogenes N, Nielsen, Søren M, Mathiesen, Jesper M, Bräuner-Osborne, Hans
Published in Molecular pharmacology (01.11.2012)
Published in Molecular pharmacology (01.11.2012)
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Structural Proof of a Dimeric Positive Modulator Bridging Two Identical AMPA Receptor-Binding Sites
Kaae, Birgitte H., Harpsøe, Kasper, Kastrup, Jette S., Sanz, Alberto Contreras, Pickering, Darryl S., Metzler, Bjørn, Clausen, Rasmus P., Gajhede, Michael, Sauerberg, Per, Liljefors, Tommy, Madsen, Ulf
Published in Chemistry & biology (01.11.2007)
Published in Chemistry & biology (01.11.2007)
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Design, synthesis and in vitro pharmacology of GluK1 and GluK3 antagonists. Studies towards the design of subtype-selective antagonists through 2-carboxyethyl-phenylalanines with substituents interacting with non-conserved residues in the GluK binding sites
Sköld, Niklas, Nielsen, Birgitte, Olsen, Jacob, Han, Liwei, Olsen, Lars, Madsen, Ulf, Kristensen, Jesper L., Pickering, Darryl S., Johansen, Tommy N.
Published in Bioorganic & medicinal chemistry (01.10.2014)
Published in Bioorganic & medicinal chemistry (01.10.2014)
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Analogues of 3-Hydroxyisoxazole-Containing Glutamate Receptor Ligands Based on the 3-Hydroxypyrazole-Moiety: Design, Synthesis and Pharmacological Characterization
Jørgensen, Lars, Nielsen, Birgitte, Pickering, Darryl S., Kristensen, Anders S., Frydenvang, Karla, Madsen, Ulf, Clausen, Rasmus P.
Published in Neurochemical research (01.10.2014)
Published in Neurochemical research (01.10.2014)
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Partial agonism and antagonism of the ionotropic glutamate receptor iGLuR5: structures of the ligand-binding core in complex with domoic acid and 2-amino-3-[5-tert-butyl-3-(phosphonomethoxy)-4-isoxazolyl]propionic acid
Hald, Helle, Naur, Peter, Pickering, Darryl S, Sprogøe, Desiree, Madsen, Ulf, Timmermann, Daniel B, Ahring, Philip K, Liljefors, Tommy, Schousboe, Arne, Egebjerg, Jan, Gajhede, Michael, Kastrup, Jette Sandholm
Published in The Journal of biological chemistry (31.08.2007)
Published in The Journal of biological chemistry (31.08.2007)
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Synthesis and Pharmacological Characterization at Glutamate Receptors of the Four Enantiopure Isomers of Tricholomic Acid
Pinto, Andrea, Conti, Paola, Amici, Marco De, Tamborini, Lucia, Madsen, Ulf, Nielsen, Birgitte, Christesen, Thomas, Bräuner-Osborne, Hans, Micheli, Carlo De
Published in Journal of medicinal chemistry (10.04.2008)
Published in Journal of medicinal chemistry (10.04.2008)
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Cognitive enhancing effects of an AMPA receptor positive modulator on place learning in mice
Malá, Hana, Chen, Yuxia, Worm, Vivi Hu, Kure, Julie, Kaae, Birgitte H., Madsen, Ulf, Badolo, Lassina, Pickering, Darryl S., Mogensen, Jesper
Published in Behavioural brain research (2012)
Published in Behavioural brain research (2012)
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Synthesis and pharmacological evaluation of novel conformationally constrained homologues of glutamic acid
Conti, Paola, Caligiuri, Antonio, Pinto, Andrea, Roda, Gabriella, Tamborini, Lucia, Nielsen, Birgitte, Madsen, Ulf, Frydenvang, Karla, Colombo, Alessio, De Micheli, Carlo
Published in European journal of medicinal chemistry (01.08.2007)
Published in European journal of medicinal chemistry (01.08.2007)
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