Small molecule proteostasis regulators that reprogram the ER to reduce extracellular protein aggregation
Plate, Lars, Cooley, Christina B, Chen, John J, Paxman, Ryan J, Gallagher, Ciara M, Madoux, Franck, Genereux, Joseph C, Dobbs, Wesley, Garza, Dan, Spicer, Timothy P, Scampavia, Louis, Brown, Steven J, Rosen, Hugh, Powers, Evan T, Walter, Peter, Hodder, Peter, Wiseman, R Luke, Kelly, Jeffery W
Published in eLife (20.07.2016)
Published in eLife (20.07.2016)
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Journal Article
Development of Functionally Selective, Small Molecule Agonists at Kappa Opioid Receptors
Zhou, Lei, Lovell, Kimberly M., Frankowski, Kevin J., Slauson, Stephen R., Phillips, Angela M., Streicher, John M., Stahl, Edward, Schmid, Cullen L., Hodder, Peter, Madoux, Franck, Cameron, Michael D., Prisinzano, Thomas E., Aubé, Jeffrey, Bohn, Laura M.
Published in The Journal of biological chemistry (20.12.2013)
Published in The Journal of biological chemistry (20.12.2013)
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Journal Article
Advanced Development of Primary Pancreatic Organoid Tumor Models for High-Throughput Phenotypic Drug Screening
Hou, Shurong, Tiriac, Hervé, Sridharan, Banu Priya, Scampavia, Louis, Madoux, Franck, Seldin, Jan, Souza, Glauco R., Watson, Donald, Tuveson, David, Spicer, Timothy P.
Published in SLAS discovery (01.07.2018)
Published in SLAS discovery (01.07.2018)
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Journal Article
Inhibition of Adrenocortical Carcinoma Cell Proliferation by Steroidogenic Factor-1 Inverse Agonists
Doghman, Mabrouka, Cazareth, Julie, Douguet, Dominique, Madoux, Franck, Hodder, Peter, Lalli, Enzo
Published in The journal of clinical endocrinology and metabolism (01.06.2009)
Published in The journal of clinical endocrinology and metabolism (01.06.2009)
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Journal Article
Discovery of an enzyme and substrate selective inhibitor of ADAM10 using an exosite-binding glycosylated substrate
Madoux, Franck, Dreymuller, Daniela, Pettiloud, Jean-Phillipe, Santos, Radleigh, Becker-Pauly, Christoph, Ludwig, Andreas, Fields, Gregg B, Bannister, Thomas, Spicer, Timothy P, Cudic, Mare, Scampavia, Louis D, Minond, Dmitriy
Published in Scientific reports (05.12.2016)
Published in Scientific reports (05.12.2016)
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Journal Article
Identification of verrucarin a as a potent and selective steroid receptor coactivator-3 small molecule inhibitor
Yan, Fei, Yu, Yang, Chow, Dar-Chone, Palzkill, Timothy, Madoux, Franck, Hodder, Peter, Chase, Peter, Griffin, Patrick R, O'Malley, Bert W, Lonard, David M
Published in PloS one (01.04.2014)
Published in PloS one (01.04.2014)
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Journal Article
Selective Targeting of Extracellular Insulin-Degrading Enzyme by Quasi-Irreversible Thiol-Modifying Inhibitors
Abdul-Hay, Samer O, Bannister, Thomas D, Wang, Hui, Cameron, Michael D, Caulfield, Thomas R, Masson, Amandine, Bertrand, Juliette, Howard, Erin A, McGuire, Michael P, Crisafulli, Umberto, Rosenberry, Terrone R, Topper, Caitlyn L, Thompson, Caroline R, Schürer, Stephan C, Madoux, Franck, Hodder, Peter, Leissring, Malcolm A
Published in ACS chemical biology (18.12.2015)
Published in ACS chemical biology (18.12.2015)
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Journal Article
Potent, Selective and Cell Penetrant Inhibitors of SF-1 by Functional Ultra-High-Throughput Screening
Madoux, Franck, Li, Xiaolin, Chase, Peter, Zastrow, Gina, Cameron, Michael D, Conkright, Juliana J, Griffin, Patrick R, Thacher, Scott, Hodder, Peter
Published in Molecular pharmacology (01.06.2008)
Published in Molecular pharmacology (01.06.2008)
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Journal Article
Bufalin Is a Potent Small-Molecule Inhibitor of the Steroid Receptor Coactivators SRC-3 and SRC-1
YING WANG, LONARD, David M, HODDER, Peter, CHASE, Peter, GRIFFIN, Patrick R, SUOLING ZHOU, LAN LIAO, JIANMING XU, O'MALLEY, Bert W, YANG YU, CHOW, Dar-Chone, PALZKILL, Timothy G, JIN WANG, RUOGU QI, MATZUK, Alexander J, XIANZHOU SONG, MADOUX, Franck
Published in Cancer research (Chicago, Ill.) (01.03.2014)
Published in Cancer research (Chicago, Ill.) (01.03.2014)
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Journal Article
A novel three-dimensional high-throughput screening approach identifies inducers of a mutant KRAS selective lethal phenotype
Kota, Smitha, Hou, Shurong, Guerrant, William, Madoux, Franck, Troutman, Scott, Fernandez-Vega, Virneliz, Alekseeva, Nina, Madala, Neeharika, Scampavia, Louis, Kissil, Joseph, Spicer, Timothy P
Published in Oncogene (01.08.2018)
Published in Oncogene (01.08.2018)
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Journal Article
Small-molecule proteostasis regulators for protein conformational diseases
Calamini, Barbara, Silva, Maria Catarina, Madoux, Franck, Hutt, Darren M, Khanna, Shilpi, Chalfant, Monica A, Saldanha, S Adrian, Hodder, Peter, Tait, Bradley D, Garza, Dan, Balch, William E, Morimoto, Richard I
Published in Nature chemical biology (25.12.2011)
Published in Nature chemical biology (25.12.2011)
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Journal Article
Endogenous and Synthetic ABHD5 Ligands Regulate ABHD5-Perilipin Interactions and Lipolysis in Fat and Muscle
Sanders, Matthew A., Madoux, Franck, Mladenovic, Ljiljana, Zhang, Huamei, Ye, Xiangqun, Angrish, Michelle, Mottillo, Emilio P., Caruso, Joseph A., Halvorsen, Geoff, Roush, William R., Chase, Peter, Hodder, Peter, Granneman, James G.
Published in Cell metabolism (03.11.2015)
Published in Cell metabolism (03.11.2015)
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Journal Article
A 1536-Well 3D Viability Assay to Assess the Cytotoxic Effect of Drugs on Spheroids
Madoux, Franck, Tanner, Allison, Vessels, Michelle, Willetts, Lynsey, Hou, Shurong, Scampavia, Louis, Spicer, Timothy P.
Published in SLAS discovery (01.06.2017)
Published in SLAS discovery (01.06.2017)
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Journal Article
A Novel 3-dimensional High Throughput Screening Approach Identifies Inducers of a Mutant KRAS Selective Lethal Phenotype
Kota, Smitha, Hou, Shurong, Guerrant, William, Madoux, Franck, Troutman, Scott, Fernandez-Vega, Virneliz, Alekseeva, Nina, Madala, Neeharika, Scampavia, Louis, Kissil, Joseph, Spicer, Timothy P.
Published in Oncogene (10.05.2018)
Published in Oncogene (10.05.2018)
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Journal Article
Casein Kinase 1δ-dependent Wee1 Protein Degradation
Penas, Clara, Ramachandran, Vimal, Simanski, Scott, Lee, Choogon, Madoux, Franck, Rahaim, Ronald J., Chauhan, Ruchi, Barnaby, Omar, Schurer, Stephan, Hodder, Peter, Steen, Judith, Roush, William R., Ayad, Nagi G.
Published in The Journal of biological chemistry (04.07.2014)
Published in The Journal of biological chemistry (04.07.2014)
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Journal Article
First-in-Class Inhibitors of Sulfur Metabolism with Bactericidal Activity against Non-Replicating M. tuberculosis
Palde, Prakash B., Bhaskar, Ashima, Pedró Rosa, Laura E., Madoux, Franck, Chase, Peter, Gupta, Vinayak, Spicer, Timothy, Scampavia, Louis, Singh, Amit, Carroll, Kate S.
Published in ACS chemical biology (15.01.2016)
Published in ACS chemical biology (15.01.2016)
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Journal Article
A FluoPol-ABPP PAD2 High-Throughput Screen Identifies the First Calcium Site Inhibitor Targeting the PADs
Lewallen, Daniel M, Bicker, Kevin L, Madoux, Franck, Chase, Peter, Anguish, Lynne, Coonrod, Scott, Hodder, Peter, Thompson, Paul R
Published in ACS chemical biology (18.04.2014)
Published in ACS chemical biology (18.04.2014)
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Journal Article
Identification of small-molecule inhibitors of the colorectal cancer oncogene Krüppel-like factor 5 expression by ultrahigh-throughput screening
Bialkowska, Agnieszka B, Crisp, Melissa, Bannister, Thomas, He, Yuanjun, Chowdhury, Sarwat, Schürer, Stephan, Chase, Peter, Spicer, Timothy, Madoux, Franck, Tian, Chenlu, Hodder, Peter, Zaharevitz, Daniel, Yang, Vincent W
Published in Molecular cancer therapeutics (01.11.2011)
Published in Molecular cancer therapeutics (01.11.2011)
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Journal Article
Development of high throughput screening assays and pilot screen for inhibitors of metalloproteases meprin α and β
Madoux, Franck, Tredup, Claudia, Spicer, Timothy P., Scampavia, Louis, Chase, Peter S., Hodder, Peter S., Fields, Gregg B., Becker-Pauly, Christoph, Minond, Dmitriy
Published in Biopolymers (01.09.2014)
Published in Biopolymers (01.09.2014)
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