Structure-guided design of a selective inhibitor of the methyltransferase KMT9 with cellular activity
Wang, Sheng, Klein, Sebastian O, Urban, Sylvia, Staudt, Maximilian, Barthes, Nicolas P F, Willmann, Dominica, Bacher, Johannes, Sum, Manuela, Bauer, Helena, Peng, Ling, Rennar, Georg A, Gratzke, Christian, Schüle, Katrin M, Zhang, Lin, Einsle, Oliver, Greschik, Holger, MacLeod, Calum, Thomson, Christopher G, Jung, Manfred, Metzger, Eric, Schüle, Roland
Published in Nature communications (02.01.2024)
Published in Nature communications (02.01.2024)
Get full text
Journal Article
A restricted role for TYK2 catalytic activity in human cytokine responses revealed by novel TYK2-selective inhibitors
Sohn, Sue J, Barrett, Kathy, Van Abbema, Anne, Chang, Christine, Kohli, Pawan Bir, Kanda, Hidenobu, Smith, Janice, Lai, Yingjie, Zhou, Aihe, Zhang, Birong, Yang, Wenqian, Williams, Karen, Macleod, Calum, Hurley, Christopher A, Kulagowski, Janusz J, Lewin-Koh, Nicholas, Dengler, Hart S, Johnson, Adam R, Ghilardi, Nico, Zak, Mark, Liang, Jun, Blair, Wade S, Magnuson, Steven, Wu, Lawren C
Published in The Journal of immunology (1950) (01.09.2013)
Published in The Journal of immunology (1950) (01.09.2013)
Get full text
Journal Article
Synthesis of 2-Substituted Benzofurans and Indoles Using Functionalized Titanium Benzylidene Reagents on Solid Phase
Macleod, Calum, McKiernan, Gordon J, Guthrie, Emma J, Farrugia, Louis J, Hamprecht, Dieter W, Macritchie, Jackie, Hartley, Richard C
Published in Journal of organic chemistry (24.01.2003)
Published in Journal of organic chemistry (24.01.2003)
Get full text
Journal Article
Discovery of GDC-0077 (Inavolisib), a Highly Selective Inhibitor and Degrader of Mutant PI3Kα
Hanan, Emily J., Braun, Marie-Gabrielle, Heald, Robert A., MacLeod, Calum, Chan, Connie, Clausen, Saundra, Edgar, Kyle A., Eigenbrot, Charles, Elliott, Richard, Endres, Nicholas, Friedman, Lori S., Gogol, Emily, Gu, Xiao-Hui, Thibodeau, Rebecca Hong, Jackson, Philip S., Kiefer, James R., Knight, Jamie D., Nannini, Michelle, Narukulla, Raman, Pace, Amanda, Pang, Jodie, Purkey, Hans E., Salphati, Laurent, Sampath, Deepak, Schmidt, Stephen, Sideris, Steve, Song, Kyung, Sujatha-Bhaskar, Swathi, Ultsch, Mark, Wallweber, Heidi, Xin, Jianfeng, Yeap, SiewKuen, Young, Amy, Zhong, Yu, Staben, Steven T.
Published in Journal of medicinal chemistry (22.12.2022)
Published in Journal of medicinal chemistry (22.12.2022)
Get full text
Journal Article
Plastic bag politics: modifying consumer behaviour for sustainable development
Ritch, Elaine, Brennan, Carol, MacLeod, Calum
Published in International journal of consumer studies (01.03.2009)
Published in International journal of consumer studies (01.03.2009)
Get full text
Journal Article
Organising a collaborative online hackathon for cutting‐edge climate research
Thomas, James, Stone, Emma J., Mitchell, Dann M., Seviour, William, Barnes, Clair, Bloomfield, Hannah, Crook, Julia, Jones, Hayley, MacLeod, Calum
Published in Weather (01.06.2022)
Published in Weather (01.06.2022)
Get full text
Journal Article
Identification of an imidazopyridine scaffold to generate potent and selective TYK2 inhibitors that demonstrate activity in an in vivo psoriasis model
Liang, Jun, Van Abbema, Anne, Balazs, Mercedesz, Barrett, Kathy, Berezhkovsky, Leo, Blair, Wade S., Chang, Christine, Delarosa, Donnie, DeVoss, Jason, Driscoll, Jim, Eigenbrot, Charles, Goodacre, Simon, Ghilardi, Nico, MacLeod, Calum, Johnson, Adam, Bir Kohli, Pawan, Lai, Yingjie, Lin, Zhonghua, Mantik, Priscilla, Menghrajani, Kapil, Nguyen, Hieu, Peng, Ivan, Sambrone, Amy, Shia, Steven, Smith, Jan, Sohn, Sue, Tsui, Vickie, Ultsch, Mark, Williams, Karen, Wu, Lawren C., Yang, Wenqian, Zhang, Birong, Magnuson, Steven
Published in Bioorganic & medicinal chemistry letters (15.09.2017)
Published in Bioorganic & medicinal chemistry letters (15.09.2017)
Get full text
Journal Article
Mitigation of Acetylcholine Esterase Activity in the 1,7-Diazacarbazole Series of Inhibitors of Checkpoint Kinase 1
Gazzard, Lewis, Williams, Karen, Chen, Huifen, Axford, Lorraine, Blackwood, Elizabeth, Burton, Brenda, Chapman, Kerry, Crackett, Peter, Drobnick, Joy, Ellwood, Charles, Epler, Jennifer, Flagella, Michael, Gancia, Emanuela, Gill, Matthew, Goodacre, Simon, Halladay, Jason, Hewitt, Joanne, Hunt, Hazel, Kintz, Samuel, Lyssikatos, Joseph, Macleod, Calum, Major, Sarah, Médard, Guillaume, Narukulla, Raman, Ramiscal, Judi, Schmidt, Stephen, Seward, Eileen, Wiesmann, Christian, Wu, Ping, Yee, Sharon, Yen, Ivana, Malek, Shiva
Published in Journal of medicinal chemistry (25.06.2015)
Published in Journal of medicinal chemistry (25.06.2015)
Get full text
Journal Article
The acute management of ankle fractures (Augment) study: A prospective trainee led national collaborative audit of the Boast 12 guidelines
Stedman, Tobias, Kumar, Vish, Shin, Je Song, Haines, Samuel, Monsell, Fergal, Dewar, Greg, Kozhikunnath, Arun, Rai, Praveen, Tadros, John, Black, Jonathon, Rae, Fraser, Tan, Harriet, Smith, Ben, Chuter, Graham, Javed, Omar, Ho, Beatrice, Williams, Mark, Bull, Eleanor, Hassan, Abdul Rahman, Howe, Thomas, Knapper, Thomas, Fleming, Tom, Fowler, Tim, Grice, John, Taylor, Alexander, Al-Kaisi, Kahlan, Paavana, Thumri, Goh, En Lin, Costa, Matthew, Harris, Maredudd, Siddiqui, Nashat, White, Andrew, Chawla, Amit, Dalwai, Ramesh, Dixit, Anurag, Papachristou, Athanasios, Tweedie, Blair, Drake, Benjamin, Khan, Sameer, Ward, Alex, Madhvani, Kiran, Naveed, Umna, Chahal, Gurdip, Watts, Anna, Blundell, Chris, Harrison, Peter, Wright, Jake, Lesko, Laszlo, Osman, Khabab, Hartley, Laura, Marsh, Alastair, Lloyd, Adam, Fananapazir, Leila, Hartshorn, Rebecca, Divecha, Hiren, Peiris, Kennedy, James, Rogers, Sophie, Hodhody, Ghazal, Jones, Matt, Davies-Jones, Gareth, Kay, Robert, Elbana, Husam, Cash, Thomas, Studnicka, Katarzyna, Bux, Mohammed, McLauchlan, George, Stirling, Scott, Rossiter, Daniel, Anibueze, Chukwudubem, To, Christopher, Gyimah, Dominic Ayi, Fagg, James, Stanger, Sophie, Al-Sukaini, Ahmad, Venkatesan, Mohanraj, McKerron, Sally, Abdelaziz, Ahmed, Toh, Eugene, Balai, Edward, Lowdon, Hamish, Davda, Kinner, Solari, Francesca, Hill, Daniel, Anderson, Kerry, Forder, Justin, Bikkannavar, Pratik, Erotocritou, Marios, Singh, Saumya, Cadwallader, Craig, Latif, Javed, Baid, Roshni, Khatri, Khushboo, Zafeiris, Konstantinos, Charalambides, Charalambos, Taylor, Isabel, Qulaghassi, Mahdi, Onubogu, Ifeanyi Kem, Oliver, Matthew, Williams, James
Published in The surgeon (Edinburgh) (01.10.2021)
Published in The surgeon (Edinburgh) (01.10.2021)
Get full text
Journal Article
BENZOXAZEPIN OXAZOLIDINONE COMPOUNDS AND METHODS OF USE
BRAUN MARIE GABRIELLE, ELLIOTT RICHARD, MACLEOD CALUM, STABEN STEVEN T, HANAN EMILY, HEALD ROBERT ANDREW
Year of Publication 28.08.2019
Get full text
Year of Publication 28.08.2019
Patent
Trigger finger as the first presentation of Dupuytren’s disease
Jamal, Bilal, Bell, Sarah, Milne, Alistair, MacLeod, Calum
Published in European orthopaedics and traumatology (08.06.2015)
Published in European orthopaedics and traumatology (08.06.2015)
Get full text
Journal Article
융합된 티오펜 유도체 및 이의 용도
MACHIN PETER, MELDRUM ERIC, MALAGU KARINE FABIENNE, PROISY NICOLAS, WINSHIP PAUL COLIN MICHAEL, LANARO ROBERTA, MACLEOD CALUM, CHAMBERS MARK, VESEY DAVID RICHARD, DE CHASSEY BENOIT
Year of Publication 18.12.2020
Get full text
Year of Publication 18.12.2020
Patent
NIK 억제제로서의 신규 치환 아자인돌린 유도체
GROSS GERHARD MAX, JACOBY EDGAR, KULAGOWSKI JANUSZ JOZEF, QUEROLLE OLIVIER ALEXIS GEORGES, MACLEOD CALUM, MEERPOEL LIEVEN, HYND GEORGE, PONCELET VIRGINIE SOPHIE, MANN SAMUEL EDWARD, STANSFIELD IAN
Year of Publication 09.03.2020
Get full text
Year of Publication 09.03.2020
Patent
벤즈옥사제핀 옥사졸리디논 화합물 및 사용 방법
BRAUN MARIE GABRIELLE, ELLIOTT RICHARD, MACLEOD CALUM, STABEN STEVEN T, HANAN EMILY, HEALD ROBERT ANDREW
Year of Publication 17.01.2018
Get full text
Year of Publication 17.01.2018
Patent
NEW THIENOPYRIMIDINE DERIVATIVES AS NIK INHIBITORS
MACLEOD CALUM, PRICE STEPHEN COLIN, MONTANA JOHN GARY, TISSELLI PATRIZIA, HYND GEORGE, MANN SAMUEL EDWARD
Year of Publication 14.06.2017
Get full text
Year of Publication 14.06.2017
Patent