A new mild method for the synthesis of amidines
Lange, Udo E.W., Schäfer, Bernd, Baucke, Dorit, Buschmann, Ernst, Mack, Helmut
Published in Tetrahedron letters (24.09.1999)
Published in Tetrahedron letters (24.09.1999)
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Journal Article
Discovery of ABT-957: 1-Benzyl-5-oxopyrrolidine-2-carboxamides as selective calpain inhibitors with enhanced metabolic stability
Jantos, Katja, Kling, Andreas, Mack, Helmut, Hornberger, Wilfried, Moeller, Achim, Nimmrich, Volker, Lao, Yanbin, Nijsen, Marjoleen
Published in Bioorganic & medicinal chemistry letters (01.08.2019)
Published in Bioorganic & medicinal chemistry letters (01.08.2019)
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Journal Article
Rho kinase, a promising drug target for neurological disorders
Mueller, Bernhard K, Mack, Helmut, Teusch, Nicole
Published in Nature reviews. Drug discovery (01.05.2005)
Published in Nature reviews. Drug discovery (01.05.2005)
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Journal Article
Discovery of Novel and Highly Selective Inhibitors of Calpain for the Treatment of Alzheimer’s Disease: 2‑(3-Phenyl‑1H‑pyrazol-1-yl)-nicotinamides
Kling, Andreas, Jantos, Katja, Mack, Helmut, Hornberger, Wilfried, Drescher, Karla, Nimmrich, Volker, Relo, Ana, Wicke, Karsten, Hutchins, Charles W, Lao, Yanbin, Marsh, Kennan, Moeller, Achim
Published in Journal of medicinal chemistry (24.08.2017)
Published in Journal of medicinal chemistry (24.08.2017)
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Journal Article
Inhibition of Rho kinase (ROCK) increases neurite outgrowth on chondroitin sulphate proteoglycan in vitro and axonal regeneration in the adult optic nerve in vivo
Lingor, Paul, Teusch, Nicole, Schwarz, Katrin, Mueller, Reinhold, Mack, Helmut, Bähr, Mathias, Mueller, Bernhard K
Published in Journal of neurochemistry (01.10.2007)
Published in Journal of neurochemistry (01.10.2007)
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Journal Article
서브미크론 표면-개질된 금속 산화물 입자
SHARMA MEGHA, GIASUDDIN ABUL BASHAR MOHAMMAD, MACK HELMUT, RUBERU THANTHIRIGE PURNIMA A
Year of Publication 30.05.2024
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Year of Publication 30.05.2024
Patent
Identification of Selective Dual ROCK1 and ROCK2 Inhibitors Using Structure-Based Drug Design
Hobson, Adrian D, Judge, Russell A, Aguirre, Ana L, Brown, Brian S, Cui, Yifang, Ding, Ping, Dominguez, Eric, DiGiammarino, Enrico, Egan, David A, Freiberg, Gail M, Gopalakrishnan, Sujatha M, Harris, Christopher M, Honore, Marie P, Kage, Karen L, Kapecki, Nicolas J, Ling, Christopher, Ma, Junli, Mack, Helmut, Mamo, Mulugeta, Maurus, Stefan, McRae, Bradford, Moore, Nigel S, Mueller, Bernhard K, Mueller, Reinhold, Namovic, Marian T, Patel, Kaushal, Pratt, Steve D, Putman, C. Brent, Queeney, Kara L, Sarris, Kathy K, Schaffter, Lisa M, Stoll, Vincent, Vasudevan, Anil, Wang, Lei, Wang, Lu, Wirthl, William, Yach, Kimberly
Published in Journal of medicinal chemistry (27.12.2018)
Published in Journal of medicinal chemistry (27.12.2018)
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Journal Article
Mitigating the Metabolic Liability of Carbonyl Reduction: Novel Calpain Inhibitors with P1′ Extension
Kling, Andreas, Jantos, Katja, Mack, Helmut, Hornberger, Wilfried, Backfisch, Gisela, Lao, Yanbin, Nijsen, Marjoleen, Rendenbach-Mueller, Beatrice, Moeller, Achim
Published in ACS medicinal chemistry letters (08.03.2018)
Published in ACS medicinal chemistry letters (08.03.2018)
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Journal Article
A-1048400 is a novel, orally active, state-dependent neuronal calcium channel blocker that produces dose-dependent antinociception without altering hemodynamic function in rats
Scott, Victoria E., Vortherms, Timothy A., Niforatos, Wende, Swensen, Andrew M., Neelands, Torben, Milicic, Ivan, Banfor, Patricia N., King, Andrew, Zhong, Chengmin, Simler, Gricelda, Zhan, Cenchen, Bratcher, Natalie, Boyce-Rustay, Janel M., Zhu, Chang Z., Bhatia, Pramila, Doherty, George, Mack, Helmut, Stewart, Andrew O., Jarvis, Michael F.
Published in Biochemical pharmacology (01.02.2012)
Published in Biochemical pharmacology (01.02.2012)
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Journal Article
HETEROCYCLIC COMPOUNDS AND THEIR USE AS GLYCOGEN SYNTHASE KINASE-3 INHIBITORS
MARCEL VAN GAALEN, MACK HELMUT, MARGARETHA HENRICA MARIA BAKKER, SEAN COLM TURNER, CAROLIN HOFT, WILFRIED HORNBERGER
Year of Publication 13.07.2017
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Year of Publication 13.07.2017
Patent
Discovery of diphenyl lactam derivatives as N-type calcium channel blockers
Doherty, George A., Bhatia, Pramila, Vortherms, Timothy A., Marsh, Kennan C., Wetter, Jill M., Mack, Helmut, Scott, Victoria E., Jarvis, Michael F., Stewart, Andrew O.
Published in Bioorganic & medicinal chemistry letters (15.02.2012)
Published in Bioorganic & medicinal chemistry letters (15.02.2012)
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Journal Article
CARBOXAMIDE COMPOUNDS AND THEIR USE AS CALPAIN INHIBITORS IV
MACK HELMUT, GISELA BACKFISCH, LAO YANBIN, KLING ANDREAS, ACHIM MOELLER, KATJA JANTOS, WILFRIED HORNBERGER, MARJOLEEN NIJSEN
Year of Publication 28.04.2016
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Year of Publication 28.04.2016
Patent
CARBOXAMIDE COMPOUNDS AND THEIR USE AS CALPAIN INHIBITORS
SEEMANN DIETMAR, NIMMRICH VOLKER, MACK HELMUT, KLING ANDREAS, MOELLER ACHIM, HORNBERGER WILFRIED, LUBISCH WILFRIED
Year of Publication 05.08.2015
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Year of Publication 05.08.2015
Patent
CARBOXAMIDE COMPOUNDS AND THEIR USE AS CALPAIN INHIBITORS
SEEMANN DIETMAR, NIMMRICH VOLKER, MACK HELMUT, KLING ANDREAS, MOELLER ACHIM, HORNBERGER WILFRIED, LUBISCH WILFRIED
Year of Publication 05.08.2015
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Year of Publication 05.08.2015
Patent