NanoLuc Complementation Reporter Optimized for Accurate Measurement of Protein Interactions in Cells
Dixon, Andrew S, Schwinn, Marie K, Hall, Mary P, Zimmerman, Kris, Otto, Paul, Lubben, Thomas H, Butler, Braeden L, Binkowski, Brock F, Machleidt, Thomas, Kirkland, Thomas A, Wood, Monika G, Eggers, Christopher T, Encell, Lance P, Wood, Keith V
Published in ACS chemical biology (19.02.2016)
Published in ACS chemical biology (19.02.2016)
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Journal Article
NanoBRETA Novel BRET Platform for the Analysis of Protein–Protein Interactions
Machleidt, Thomas, Woodroofe, Carolyn C, Schwinn, Marie K, Méndez, Jacqui, Robers, Matthew B, Zimmerman, Kris, Otto, Paul, Daniels, Danette L, Kirkland, Thomas A, Wood, Keith V
Published in ACS chemical biology (21.08.2015)
Published in ACS chemical biology (21.08.2015)
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Journal Article
Quantitative, Wide-Spectrum Kinase Profiling in Live Cells for Assessing the Effect of Cellular ATP on Target Engagement
Vasta, James D., Corona, Cesear R., Wilkinson, Jennifer, Zimprich, Chad A., Hartnett, James R., Ingold, Morgan R., Zimmerman, Kristopher, Machleidt, Thomas, Kirkland, Thomas A., Huwiler, Kristin G., Ohana, Rachel Friedman, Slater, Michael, Otto, Paul, Cong, Mei, Wells, Carrow I., Berger, Benedict-Tilman, Hanke, Thomas, Glas, Carina, Ding, Ke, Drewry, David H., Huber, Kilian V.M., Willson, Timothy M., Knapp, Stefan, Müller, Susanne, Meisenheimer, Poncho L., Fan, Frank, Wood, Keith V., Robers, Matthew B.
Published in Cell chemical biology (15.02.2018)
Published in Cell chemical biology (15.02.2018)
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Journal Article
Application of BRET to monitor ligand binding to GPCRs
Stoddart, Leigh A, Johnstone, Elizabeth K M, Wheal, Amanda J, Goulding, Joëlle, Robers, Matthew B, Machleidt, Thomas, Wood, Keith V, Hill, Stephen J, Pfleger, Kevin D G
Published in Nature methods (01.07.2015)
Published in Nature methods (01.07.2015)
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Journal Article
Engineered Luciferase Reporter from a Deep Sea Shrimp Utilizing a Novel Imidazopyrazinone Substrate
Hall, Mary P, Unch, James, Binkowski, Brock F, Valley, Michael P, Butler, Braeden L, Wood, Monika G, Otto, Paul, Zimmerman, Kristopher, Vidugiris, Gediminas, Machleidt, Thomas, Robers, Matthew B, Benink, Hélène A, Eggers, Christopher T, Slater, Michael R, Meisenheimer, Poncho L, Klaubert, Dieter H, Fan, Frank, Encell, Lance P, Wood, Keith V
Published in ACS chemical biology (16.11.2012)
Published in ACS chemical biology (16.11.2012)
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Journal Article
Monitoring phosphorylation and acetylation of CRISPR-mediated HiBiT-tagged endogenous proteins
Alves, Juliano, Schwinn, Marie, Machleidt, Thomas, Goueli, Said A., Cali, James J., Zegzouti, Hicham
Published in Scientific reports (25.01.2024)
Published in Scientific reports (25.01.2024)
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Journal Article
Simultaneous inhibition of DNA-PK and Polϴ improves integration efficiency and precision of genome editing
Wimberger, Sandra, Akrap, Nina, Firth, Mike, Brengdahl, Johan, Engberg, Susanna, Schwinn, Marie K., Slater, Michael R., Lundin, Anders, Hsieh, Pei-Pei, Li, Songyuan, Cerboni, Silvia, Sumner, Jonathan, Bestas, Burcu, Schiffthaler, Bastian, Magnusson, Björn, Di Castro, Silvio, Iyer, Preeti, Bohlooly-Y, Mohammad, Machleidt, Thomas, Rees, Steve, Engkvist, Ola, Norris, Tyrell, Cadogan, Elaine B., Forment, Josep V., Šviković, Saša, Akcakaya, Pinar, Taheri-Ghahfarokhi, Amir, Maresca, Marcello
Published in Nature communications (14.08.2023)
Published in Nature communications (14.08.2023)
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Exploiting an Asp-Glu "switch" in glycogen synthase kinase 3 to design paralog-selective inhibitors for use in acute myeloid leukemia
Wagner, Florence F, Benajiba, Lina, Campbell, Arthur J, Weïwer, Michel, Sacher, Joshua R, Gale, Jennifer P, Ross, Linda, Puissant, Alexandre, Alexe, Gabriela, Conway, Amy, Back, Morgan, Pikman, Yana, Galinsky, Ilene, DeAngelo, Daniel J, Stone, Richard M, Kaya, Taner, Shi, Xi, Robers, Matthew B, Machleidt, Thomas, Wilkinson, Jennifer, Hermine, Olivier, Kung, Andrew, Stein, Adam J, Lakshminarasimhan, Damodharan, Hemann, Michael T, Scolnick, Edward, Zhang, Yan-Ling, Pan, Jen Q, Stegmaier, Kimberly, Holson, Edward B
Published in Science translational medicine (07.03.2018)
Published in Science translational medicine (07.03.2018)
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Journal Article
Identification of a new JNK inhibitor targeting the JNK-JIP interaction site
Stebbins, John L, De, Surya K, Machleidt, Thomas, Becattini, Barbara, Vazquez, Jesus, Kuntzen, Christian, Chen, Li-Hsing, Cellitti, Jason F, Riel-Mehan, Megan, Emdadi, Aras, Solinas, Giovanni, Karin, Michael, Pellecchia, Maurizio
Published in Proceedings of the National Academy of Sciences - PNAS (28.10.2008)
Published in Proceedings of the National Academy of Sciences - PNAS (28.10.2008)
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Journal Article
An Integrated Approach toward NanoBRET Tracers for Analysis of GPCR Ligand Engagement
Killoran, Michael P., Levin, Sergiy, Boursier, Michelle E., Zimmerman, Kristopher, Hurst, Robin, Hall, Mary P., Machleidt, Thomas, Kirkland, Thomas A., Friedman Ohana, Rachel
Published in Molecules (Basel, Switzerland) (12.05.2021)
Published in Molecules (Basel, Switzerland) (12.05.2021)
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Journal Article
5,5-Dialkylluciferins are thermal stable substrates for bioluminescence-based detection systems
Shi, Ce, Killoran, Michael P, Hall, Mary P, Otto, Paul, Wood, Monika G, Strauss, Ethan, Encell, Lance P, Machleidt, Thomas, Wood, Keith V, Kirkland, Thomas A
Published in PloS one (14.12.2020)
Published in PloS one (14.12.2020)
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Journal Article
Luciferase Calibrants Enable Absolute Quantitation of Bioluminescence Power
Klein, Mark A., Lazarev, Sergey, Gervasi, Charles, Cowan, Cristopher, Machleidt, Thomas, Friedman Ohana, Rachel
Published in ACS measurement science au (20.12.2023)
Published in ACS measurement science au (20.12.2023)
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Journal Article
Development of a rapid, simple, and sensitive point-of-care technology platform utilizing ternary NanoLuc
Torio, Emily A., Ressler, Valerie T., Kincaid, Virginia A., Hurst, Robin, Hall, Mary P., Encell, Lance P., Zimmerman, Kristopher, Forsyth, Stuart K., Rehrauer, William M., Accola, Molly A., Hsu, Chia-Chang, Machleidt, Thomas, Dart, Melanie L.
Published in Frontiers in microbiology (26.10.2022)
Published in Frontiers in microbiology (26.10.2022)
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Journal Article
Design, Synthesis, and Structure−Activity Relationship of Substrate Competitive, Selective, and in Vivo Active Triazole and Thiadiazole Inhibitors of the c-Jun N-Terminal Kinase
De, Surya K, Stebbins, John L, Chen, Li-Hsing, Riel-Mehan, Megan, Machleidt, Thomas, Dahl, Russell, Yuan, Hongbin, Emdadi, Aras, Barile, Elisa, Chen, Vida, Murphy, Ria, Pellecchia, Maurizio
Published in Journal of medicinal chemistry (09.04.2009)
Published in Journal of medicinal chemistry (09.04.2009)
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Journal Article
Identification of known drugs targeting the endoplasmic reticulum stress response
Bi, Kun, Nishihara, Kana, Machleidt, Thomas, Hermanson, Spencer, Wang, Jun, Sakamuru, Srilatha, Huang, Ruili, Xia, Menghang
Published in Analytical and bioanalytical chemistry (01.07.2015)
Published in Analytical and bioanalytical chemistry (01.07.2015)
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Journal Article
Dual control of caveolar membrane traffic by microtubules and the actin cytoskeleton
Mundy, Dorothy I, Machleidt, Thomas, Ying, Yun-shu, Anderson, Richard G W, Bloom, George S
Published in Journal of cell science (15.11.2002)
Published in Journal of cell science (15.11.2002)
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Journal Article
Real-time analysis of the binding of fluorescent VEGF 165 a to VEGFR2 in living cells: Effect of receptor tyrosine kinase inhibitors and fate of internalized agonist-receptor complexes
Kilpatrick, Laura E, Friedman-Ohana, Rachel, Alcobia, Diana C, Riching, Kristin, Peach, Chloe J, Wheal, Amanda J, Briddon, Stephen J, Robers, Matthew B, Zimmerman, Kris, Machleidt, Thomas, Wood, Keith V, Woolard, Jeanette, Hill, Stephen J
Published in Biochemical pharmacology (01.07.2017)
Published in Biochemical pharmacology (01.07.2017)
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