Cardioprotective Angiotensin-(1–7) Peptide Acts as a Natural-Biased Ligand at the Angiotensin II Type 1 Receptor
Galandrin, Ségolène, Denis, Colette, Boularan, Cédric, Marie, Jacky, M’Kadmi, Céline, Pilette, Claire, Dubroca, Caroline, Nicaise, Yvan, Seguelas, Marie-Hélène, N’Guyen, Du, Banères, Jean-Louis, Pathak, Atul, Sénard, Jean-Michel, Galés, Céline
Published in Hypertension (Dallas, Tex. 1979) (01.12.2016)
Published in Hypertension (Dallas, Tex. 1979) (01.12.2016)
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Journal Article
Structure and dynamics of G protein-coupled receptor–bound ghrelin reveal the critical role of the octanoyl chain
Ferré, Guillaume, Louet, Maxime, Saurel, Oliver, Delort, Bartholomé, Czaplicki, Georges, M’Kadmi, Céline, Damian, Marjorie, Renault, Pedro, Cantel, Sonia, Gavara, Laurent, Demange, Pascal, Marie, Jacky, Fehrentz, Jean-Alain, Floquet, Nicolas, Milon, Alain, Banères, Jean-Louis
Published in Proceedings of the National Academy of Sciences - PNAS (27.08.2019)
Published in Proceedings of the National Academy of Sciences - PNAS (27.08.2019)
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Journal Article
Development of Nonpeptidic Inverse Agonists of the Ghrelin Receptor (GHSR) Based on the 1,2,4-Triazole Scaffold
Haj Salah, Khoubaib Ben, Maingot, Mathieu, Blayo, Anne-Laure, M’Kadmi, Céline, Damian, Marjorie, Mary, Sophie, Cantel, Sonia, Neasta, Jérémie, Oiry, Catherine, Péraldi-Roux, Sylvie, Fernandez, Gimena, Romero, Guadalupe García, Perello, Mario, Marie, Jacky, Banères, Jean-Louis, Fehrentz, Jean-Alain, Denoyelle, Séverine
Published in Journal of medicinal chemistry (08.10.2020)
Published in Journal of medicinal chemistry (08.10.2020)
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Journal Article
Ghrelin receptor conformational dynamics regulate the transition from a preassembled to an active receptor:Gq complex
Damian, Marjorie, Mary, Sophie, Maingot, Mathieu, M’Kadmi, Céline, Gagne, Didier, Leyris, Jean-Philippe, Denoyelle, Séverine, Gaibelet, Gérald, Gavara, Laurent, de Souza Costa, Mauricio Garcia, Perahia, David, Trinquet, Eric, Mouillac, Bernard, Galandrin, Ségolène, Galès, Céline, Fehrentz, Jean-Alain, Floquet, Nicolas, Martinez, Jean, Marie, Jacky, Banères, Jean-Louis
Published in Proceedings of the National Academy of Sciences - PNAS (03.02.2015)
Published in Proceedings of the National Academy of Sciences - PNAS (03.02.2015)
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Journal Article
Concerted conformational dynamics and water movements in the ghrelin G protein-coupled receptor
Louet, Maxime, Casiraghi, Marina, Damian, Marjorie, Costa, Mauricio GS, Renault, Pedro, Gomes, Antoniel AS, Batista, Paulo R, M'Kadmi, Céline, Mary, Sophie, Cantel, Sonia, Denoyelle, Severine, Ben Haj Salah, Khoubaib, Perahia, David, Bisch, Paulo M, Fehrentz, Jean-Alain, Catoire, Laurent J, Floquet, Nicolas, Banères, Jean-Louis
Published in eLife (03.09.2021)
Published in eLife (03.09.2021)
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Journal Article
The 1,2,4-triazole as a scaffold for the design of ghrelin receptor ligands: development of JMV 2959, a potent antagonist
Moulin, Aline, Brunel, Luc, Boeglin, Damien, Demange, Luc, Ryan, Johanne, M’Kadmi, Céline, Denoyelle, Séverine, Martinez, Jean, Fehrentz, Jean-Alain
Published in Amino acids (01.02.2013)
Published in Amino acids (01.02.2013)
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Journal Article
Evidence Supporting a Role for Constitutive Ghrelin Receptor Signaling in Fasting-Induced Hyperphagia in Male Mice
Fernandez, Gimena, Cabral, Agustina, Andreoli, María F, Labarthe, Alexandra, M'Kadmi, Céline, Ramos, Jorge G, Marie, Jacky, Fehrentz, Jean-Alain, Epelbaum, Jacques, Tolle, Virginie, Perello, Mario
Published in Endocrinology (Philadelphia) (01.02.2018)
Published in Endocrinology (Philadelphia) (01.02.2018)
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Journal Article
Development of a novel fluorescent ligand of growth hormone secretagogue receptor based on the N-Terminal Leap2 region
Barrile, Franco, M'Kadmi, Céline, De Francesco, Pablo N., Cabral, Agustina, García Romero, Guadalupe, Mustafá, Emilio R., Cantel, Sonia, Damian, Marjorie, Mary, Sophie, Denoyelle, Séverine, Banères, Jean-Louis, Marie, Jacky, Raingo, Jesica, Fehrentz, Jean-Alain, Perelló, Mario
Published in Molecular and cellular endocrinology (01.12.2019)
Published in Molecular and cellular endocrinology (01.12.2019)
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Journal Article
Design and characterization of a triazole-based growth hormone secretagogue receptor modulator inhibiting the glucoregulatory and feeding actions of ghrelin
Péraldi-Roux, Sylvie, Bayle, Morgane, M'Kadmi, Céline, Damian, Marjorie, Vaillé, Justine, Fernandez, Gimena, Cornejo, Maria Paula, Marie, Jacky, Banères, Jean-Louis, Ben Haj Salah, Khoubaib, Fehrentz, Jean-Alain, Cantel, Sonia, Perello, Mario, Denoyelle, Séverine, Oiry, Catherine, Neasta, Jérémie
Published in Biochemical pharmacology (01.08.2022)
Published in Biochemical pharmacology (01.08.2022)
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Journal Article
Homogeneous time-resolved fluorescence-based assay to screen for ligands targeting the growth hormone secretagogue receptor type 1a
Leyris, Jean-Philippe, Roux, Thomas, Trinquet, Eric, Verdié, Pascal, Fehrentz, Jean-Alain, Oueslati, Nadia, Douzon, Stéphanie, Bourrier, Emmanuel, Lamarque, Laurent, Gagne, Didier, Galleyrand, Jean-Claude, M’kadmi, Céline, Martinez, Jean, Mary, Sophie, Banères, Jean-Louis, Marie, Jacky
Published in Analytical biochemistry (15.01.2011)
Published in Analytical biochemistry (15.01.2011)
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Journal Article
Quantitative MALDI-MS Binding Assays: An Alternative to Radiolabeling
Rossato, Maxime, Miralles, Guillaume, M'Kadmi, Céline, Maingot, Mathieu, Amblard, Muriel, Mouillac, Bernard, Gagne, Didier, Martinez, Jean, Subra, Gilles, Enjalbal, Christine, Cantel, Sonia
Published in ChemMedChem (06.12.2016)
Published in ChemMedChem (06.12.2016)
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Journal Article
New ligands of the ghrelin receptor based on the 1,2,4-triazole scaffold by introduction of a second chiral center
Maingot, Mathieu, Blayo, Anne-Laure, Denoyelle, Séverine, M’Kadmi, Céline, Damian, Marjorie, Mary, Sophie, Gagne, Didier, Sanchez, Pierre, Aicher, Babette, Schmidt, Peter, Müller, Gilbert, Teifel, Michael, Günther, Eckhard, Marie, Jacky, Banères, Jean-Louis, Martinez, Jean, Fehrentz, Jean-Alain
Published in Bioorganic & medicinal chemistry letters (15.05.2016)
Published in Bioorganic & medicinal chemistry letters (15.05.2016)
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Journal Article
N‑Terminal Liver-Expressed Antimicrobial Peptide 2 (LEAP2) Region Exhibits Inverse Agonist Activity toward the Ghrelin Receptor
M’Kadmi, Céline, Cabral, Agustina, Barrile, Franco, Giribaldi, Julien, Cantel, Sonia, Damian, Marjorie, Mary, Sophie, Denoyelle, Séverine, Dutertre, Sébastien, Péraldi-Roux, Sylvie, Neasta, Jérémie, Oiry, Catherine, Banères, Jean-Louis, Marie, Jacky, Perello, Mario, Fehrentz, Jean-Alain
Published in Journal of medicinal chemistry (24.01.2019)
Published in Journal of medicinal chemistry (24.01.2019)
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Journal Article
Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling
M'Kadmi, Céline, Leyris, Jean-Philippe, Onfroy, Lauriane, Galés, Céline, Saulière, Aude, Gagne, Didier, Damian, Marjorie, Mary, Sophie, Maingot, Mathieu, Denoyelle, Séverine, Verdié, Pascal, Fehrentz, Jean-Alain, Martinez, Jean, Banères, Jean-Louis, Marie, Jacky
Published in The Journal of biological chemistry (06.11.2015)
Published in The Journal of biological chemistry (06.11.2015)
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Journal Article
The novel nonapeptide acein targets angiotensin converting enzyme in the brain and induces dopamine release
Neasta, Jérémie, Valmalle, Charlène, Coyne, Anne‐Claire, Carnazzi, Eric, Subra, Gilles, Galleyrand, Jean‐Claude, Gagne, Didier, M'Kadmi, Céline, Bernad, Nicole, Bergé, Gilbert, Cantel, Sonia, Marin, Philippe, Marie, Jacky, Banères, Jean‐Louis, Kemel, Marie‐Lou, Daugé, Valérie, Puget, Karine, Martinez, Jean
Published in British journal of pharmacology (01.04.2016)
Published in British journal of pharmacology (01.04.2016)
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Journal Article
α-Tocopherol and α-tocopheryl phosphate interact with the cannabinoid system in the rodent hippocampus
Crouzin, Nadine, de Jesus Ferreira, Marie-Céleste, Cohen-Solal, Catherine, M'Kadmi, Céline, Bernad, Nicole, Martinez, Jean, Barbanel, Gérard, Vignes, Michel, Guiramand, Janique
Published in Free radical biology & medicine (01.11.2011)
Published in Free radical biology & medicine (01.11.2011)
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Journal Article
Allosteric modulation of ghrelin receptor signaling by lipids
Damian, Marjorie, Louet, Maxime, Gomes, Antoniel Augusto Severo, M'Kadmi, Céline, Denoyelle, Séverine, Cantel, Sonia, Mary, Sophie, Bisch, Paulo M, Fehrentz, Jean-Alain, Catoire, Laurent J, Floquet, Nicolas, Banères, Jean-Louis
Published in Nature communications (24.06.2021)
Published in Nature communications (24.06.2021)
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Journal Article
Detergent-free Isolation of Functional G Protein-Coupled Receptors into Nanometric Lipid Particles
Logez, Christel, Damian, Marjorie, Legros, Céline, Dupré, Clémence, Guéry, Mélody, Mary, Sophie, Wagner, Renaud, M’Kadmi, Céline, Nosjean, Olivier, Fould, Benjamin, Marie, Jacky, Fehrentz, Jean-Alain, Martinez, Jean, Ferry, Gilles, Boutin, Jean A, Banères, Jean-Louis
Published in Biochemistry (Easton) (12.01.2016)
Published in Biochemistry (Easton) (12.01.2016)
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Journal Article
Trisubstituted 1,2,4-triazoles as ligands for the ghrelin receptor: On the significance of the orientation and substitution at position 3
Moulin, Aline, Demange, Luc, Ryan, Joanne, M’Kadmi, Céline, Galleyrand, Jean-Claude, Martinez, Jean, Fehrentz, Jean-Alain
Published in Bioorganic & medicinal chemistry letters (2008)
Published in Bioorganic & medicinal chemistry letters (2008)
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Journal Article
Involvement of tryptophan W276 and of two surrounding amino acid residues in the high constitutive activity of the ghrelin receptor GHS-R1a
Gozé, Catherine, Bergé, Gilbert, M'Kadmi, Céline, Floquet, Nicolas, Gagne, Didier, Galleyrand, Jean-Claude, Fehrentz, Jean-Alain, Martinez, Jean
Published in European journal of pharmacology (25.09.2010)
Published in European journal of pharmacology (25.09.2010)
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