Substituted piperidines - highly potent renin inhibitors due to induced fit adaptation of the active site
Vieira, Eric, Binggeli, Alfred, Breu, Volker, Bur, Daniel, Fischli, Walter, Güller, Rolf, Hirth, Georges, Märki, Hans Peter, Müller, Marcel, Oefner, Christian, Scalone, Michelangelo, Stadler, Heinz, Wihelm, Maurice, Wostl, Wolfgang
Published in Bioorganic & medicinal chemistry letters (17.05.1999)
Published in Bioorganic & medicinal chemistry letters (17.05.1999)
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Piperidine-renin inhibitors compounds with improved physicochemical properties
Güller, Rolf, Binggeli, Alfred, Breu, Volker, Bur, Daniel, Fischli, Walter, Hirth, Georges, Jenny, Christian, Kansy, Manfred, Montavon, François, Müller, Marcel, Oefner, Christian, Stadler, Heinz, Vieira, Eric, Wilhelm, Maurice, Wostl, Wolfgang, Märki, Hans Peter
Published in Bioorganic & medicinal chemistry letters (17.05.1999)
Published in Bioorganic & medicinal chemistry letters (17.05.1999)
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Piperidine renin inhibitors: from leads to drug candidates
Märki, H.P., Binggeli, A., Bittner, B., Bohner-Lang, V., Breu, V., Bur, D., Coassolo, Ph, Clozel, J.P., D'Arcy, A., Doebeli, H., Fischli 1, W., Funk, Ch, Foricher, J., Giller, T., Grüninger, F., Guenzi, A., Güller, R., Hartung, T., Hirth, G., Jenny, Ch, Kansy, M., Klinkhammer, U., Lave, T., Lohri, B., Luft, F.C., Mervaala, E.M., Müller, D.N., Müller, M., Montavon, F., Oefner, Ch, Qiu, C., Reichel, A., Sanwald-Ducray, P., Scalone, M., Schleimer, M., Schmid, R., Stadler, H., Treiber 1, A., Valdenaire 2, O., Vieira, E., Waldmeier, P., Wiegand-Chou, R., Wilhelm, M., Wostl, W., Zell, M., Zell, R.
Published in Farmaco (Società chimica italiana : 1989) (01.01.2001)
Published in Farmaco (Società chimica italiana : 1989) (01.01.2001)
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Conference Proceeding
Renin inhibition by substituted piperidines: A novel paradigm for the inhibition of monomeric aspartic proteinases?
Oefner, C, Binggeli, A, Breu, V, Bur, D, Clozel, J-P, D'Arcy, A, Dorn, A, Fischli, W, Grüninger, F, Güller, R, Hirth, G, Märki, HP, Mathews, S, Müller, M, Ridley, RG, Stadier, H, Vieira, E, Wilhelm, M, Winkler, FK, Wostl, W
Published in Chemistry & biology (01.03.1999)
Published in Chemistry & biology (01.03.1999)
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effect of the carbohydrate pattern of three isocaloric mixed breakfasts on the postprandial concentrations of plasma glucose, -insulin, -growth hormone and free fatty acids in normal man
Ziegler, E, Chiumello, G, Marki, H.H
Published in International journal for vitamin and nutrition research (1973)
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Published in International journal for vitamin and nutrition research (1973)
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Androgen binding in human plasma and its physiological significance (author's transl)
Lutz, R A, Märki, H H, Weder, H G
Published in Journal of clinical chemistry and clinical biochemistry (01.02.1977)
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Published in Journal of clinical chemistry and clinical biochemistry (01.02.1977)
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A Novel Partial Agonist of Peroxisome Proliferator-Activated Receptor-γ (PPARγ) Recruits PPARγ-Coactivator-1α, Prevents Triglyceride Accumulation, and Potentiates Insulin Signaling in Vitro
Burgermeister, Elke, Schnoebelen, Astride, Flament, Angele, Benz, Jörg, Stihle, Martine, Gsell, Bernard, Rufer, Arne, Ruf, Armin, Kuhn, Bernd, Märki, Hans Peter, Mizrahi, Jacques, Sebokova, Elena, Niesor, Eric, Meyer, Markus
Published in Molecular endocrinology (Baltimore, Md.) (01.04.2006)
Published in Molecular endocrinology (Baltimore, Md.) (01.04.2006)
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In vitro pharmacological properties of a series of isoprenaline derivatives
Eigenmann, R, Burkard, W P, Holck, M, Märki, H P, Osterrieder, W, Goodman, M, Melmon, K L
Published in Arzneimittel-Forschung (01.08.1989)
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Published in Arzneimittel-Forschung (01.08.1989)
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Classification and clinical significance of dysproteinemias and paraproteinemias
WUHRMANN, F, MARKI, H H
Published in Jornal da Sociedade das Ciencias Medicas de Lisboa (01.01.1962)
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Published in Jornal da Sociedade das Ciencias Medicas de Lisboa (01.01.1962)
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Study of Brazilian agricultural workers. A medico-socio-psychological study
Wiesmann, E, Mosimann, J, Drolshammer, I, Eckert, J, Märki, H, Munzinger, J, Schurter, V, Schweizer, H
Published in Acta tropica (1975)
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Published in Acta tropica (1975)
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