Inhibitors of the chymotrypsin-like activity of proteasome based on di- and tri-peptidyl α-keto aldehydes (glyoxals)
Lynas, John F., Harriott, Patrick, Healy, Adrienne, McKervey, M.Anthony, Walker, Brian
Published in Bioorganic & medicinal chemistry letters (17.02.1998)
Published in Bioorganic & medicinal chemistry letters (17.02.1998)
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Journal Article
Irreversible inhibition of the bacterial cysteine protease-transpeptidase sortase (SrtA) by substrate-derived affinity labels
Scott, Christopher J, McDowell, Andrew, Martin, S Lorraine, Lynas, John F, Vandenbroeck, Koen, Walker, Brian
Published in Biochemical journal (15.09.2002)
Published in Biochemical journal (15.09.2002)
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Journal Article
Solid-phase synthesis and biological screening of N-alpha-mercaptoamide template-based matrix metalloprotease inhibitors
Lynas, J F, Martin, S L, Walker, B, Baxter, A D, Bird, J, Bhogal, R, Montana, J G, Owen, D A
Published in Combinatorial chemistry & high throughput screening (01.02.2000)
Published in Combinatorial chemistry & high throughput screening (01.02.2000)
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Journal Article
Evaluation of Dipeptide α-Keto-β-aldehydes as New Inhibitors of Cathepsin S
Walker, Brian, Lynas, John F., Meighan, Mark A., Brömme, Dieter
Published in Biochemical and biophysical research communications (28.08.2000)
Published in Biochemical and biophysical research communications (28.08.2000)
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Journal Article
Potent new leucine aminopeptidase inhibitor of novel structure synthesised by a modified Wadsworth–Emmons (Horner) Wittig procedure
Walker, Brian, Darkins, Paul A., McKervey, M.Anthony, Moncrieff, Hazel M., Lynas, John F.
Published in Bioorganic & medicinal chemistry letters (03.07.2000)
Published in Bioorganic & medicinal chemistry letters (03.07.2000)
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Journal Article
Psychological impact of genetic testing for familial hypercholesterolemia within a previously aware population: A randomized controlled trial
Marteau, Theresa, Senior, Victoria, Humphries, Steve E., Bobrow, Martin, Cranston, Treena, Crook, Martin A., Day, Lorna, Fernandez, Maryam, Horne, Rob, Iversen, Andrew, Jackson, Zoe, Lynas, Jacqui, Middleton-Price, Helen, Savine, Richard, Sikorski, Jim, Watson, Melanie, Weinman, John, Wierzbicki, Anthony S., Wray, Richard
Published in American journal of medical genetics. Part A (30.07.2004)
Published in American journal of medical genetics. Part A (30.07.2004)
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Journal Article
Dipeptide proline diphenyl phosphonates are potent, irreversible inhibitors of seprase (FAPα)
Gilmore, Brendan F., Lynas, John F., Scott, Christopher J., McGoohan, Caroline, Martin, Lorraine, Walker, Brian
Published in Biochemical and biophysical research communications (28.07.2006)
Published in Biochemical and biophysical research communications (28.07.2006)
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Journal Article
Proteasome proteolytic activity in hematopoietic cells from patients with chronic myeloid leukemia and multiple myeloma
Magill, L, Lynas, J, Morris, TC, Walker, B, Irvine, AE
Published in Haematologica (Roma) (01.12.2004)
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Published in Haematologica (Roma) (01.12.2004)
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