(1-(4-(Naphthalen-2-yl)pyrimidin-2-yl)piperidin-4-yl)methanamine: A Wingless β-Catenin Agonist That Increases Bone Formation Rate
Pelletier, Jeffrey C, Lundquist, Joseph T, Gilbert, Adam M, Alon, Nipa, Bex, Frederick J, Bhat, Bheem M, Bursavich, Mattew G, Coleburn, Valerie E, Felix, Luciana A, Green, Daniel M, Green, Paula, Hauze, Diane B, Kharode, Yogendra P, Lam, Ho-Sun, Lockhead, Susan R, Magolda, Ronald L, Matteo, Jeanne J, Mehlmann, John F, Milligan, Colleen, Murrills, Richard J, Pirrello, Jennifer, Selim, Sally, Sharp, Michael C, Unwalla, Ray J, Vera, Matthew D, Wrobel, Jay E, Yaworsky, Paul, Bodine, Peter V. N
Published in Journal of medicinal chemistry (26.11.2009)
Published in Journal of medicinal chemistry (26.11.2009)
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Improvement of Physiochemical Properties of the Tetrahydroazepinoindole Series of Farnesoid X Receptor (FXR) Agonists: Beneficial Modulation of Lipids in Primates
Lundquist, Joseph T, Harnish, Douglas C, Kim, Callain Y, Mehlmann, John F, Unwalla, Rayomand J, Phipps, Kristin M, Crawley, Matthew L, Commons, Thomas, Green, Daniel M, Xu, Weixin, Hum, Wah-Tung, Eta, Julius E, Feingold, Irene, Patel, Vikram, Evans, Mark J, Lai, KehDih, Borges-Marcucci, Lisa, Mahaney, Paige E, Wrobel, Jay E
Published in Journal of medicinal chemistry (25.02.2010)
Published in Journal of medicinal chemistry (25.02.2010)
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2-Phenyl-4-piperazinylbenzimidazoles: Orally active inhibitors of the gonadotropin releasing hormone (GnRH) receptor
Pelletier, Jeffrey C., Chengalvala, Murty, Cottom, Josh, Feingold, Irene, Garrick, Lloyd, Green, Daniel, Hauze, Diane, Huselton, Christine, Jetter, James, Kao, Wenling, Kopf, Gregory S., Lundquist, Joseph T., Mann, Charles, Mehlmann, John, Rogers, John, Shanno, Linda, Wrobel, Jay
Published in Bioorganic & medicinal chemistry (01.07.2008)
Published in Bioorganic & medicinal chemistry (01.07.2008)
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Efficient, Regioselective Palladium-Catalyzed Tandem Heck-Isomerization Reaction of Aryl Bromides and Non-Allylic Benzyl Alcohols
Crawley, Matthew L, Phipps, Kristin M, Goljer, Igor, Mehlmann, John F, Lundquist, Joseph T, Ullrich, John W, Yang, Cuijian, Mahaney, Paige E
Published in Organic letters (05.03.2009)
Published in Organic letters (05.03.2009)
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Synthesis and biological evaluation of piperazinyl heterocyclic antagonists of the gonadotropin releasing hormone (GnRH) receptor
Vera, Matthew D., Lundquist, Joseph T., Chengalvala, Murty V., Cottom, Joshua E., Feingold, Irene B., Garrick, Lloyd M., Green, Daniel M., Hauze, Diane B., Mann, Charles W., Mehlmann, John F., Rogers, John F., Shanno, Linda, Wrobel, Jay E., Pelletier, Jeffrey C.
Published in Bioorganic & medicinal chemistry letters (15.04.2010)
Published in Bioorganic & medicinal chemistry letters (15.04.2010)
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Small molecule antagonists of the gonadotropin-releasing hormone (GnRH) receptor : Structure-activity relationships of small heterocyclic groups appended to the 2-phenyl-4-piperazinyl-benzimidazole template
HAUZE, Diane B, CHENGALVALA, Murty V, MANN, Charles W, MEHLMANN, John F, ROGERS, John F, SHANNO, Linda, WROBEL, Jay, PELLETIER, Jeffrey C, COTTOM, Joshua E, FEINGOLD, Irene B, GARRICK, Lloyd, GREEN, Daniel M, HUSELTON, Christine, WENLING KAO, KEES, Kenneth, LUNDQUIST, Joseph T
Published in Bioorganic & medicinal chemistry letters (01.04.2009)
Published in Bioorganic & medicinal chemistry letters (01.04.2009)
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Discovery of 6-({4-[2-(4-tert-Butylphenyl)-1H-benzimidazol-4-yl]piperazin-1-yl}methyl)quinoxaline (WAY-207024): An Orally Active Antagonist of the Gonadotropin Releasing Hormone Receptor (GnRH-R)
Pelletier, Jeffrey C, Chengalvala, Murty V, Cottom, Joshua E, Feingold, Irene B, Green, Daniel M, Hauze, Diane B, Huselton, Christine A, Jetter, James W, Kopf, Gregory S, Lundquist, Joseph T, Magolda, Ronald L, Mann, Charles W, Mehlmann, John F, Rogers, John F, Shanno, Linda K, Adams, William R, Tio, Cesario O, Wrobel, Jay E
Published in Journal of medicinal chemistry (09.04.2009)
Published in Journal of medicinal chemistry (09.04.2009)
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Pyrrole[2,3- d]azepino compounds as agonists of the farnesoid X receptor (FXR)
Mehlmann, John F., Crawley, Matthew L., Lundquist, Joseph T., Unwalla, Ray J., Harnish, Douglas C., Evans, Mark J., Kim, Callain Y., Wrobel, Jay E., Mahaney, Paige E.
Published in Bioorganic & medicinal chemistry letters (15.09.2009)
Published in Bioorganic & medicinal chemistry letters (15.09.2009)
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Journal Article
골수퍼옥시다제 저해제의 전구약물
STROBEL ERIC, ZHANG YAN, PELLETIER JEFFREY C, REITZ ALLEN B, LUNDQUIST JOSEPH THEODORE IV, MCWHERTER MELODY A, DUBOWCHIK GENE M
Year of Publication 14.06.2022
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Year of Publication 14.06.2022
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