Identification of a novel effector domain of BIN1 for cancer suppression
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Published in Journal of cellular biochemistry (01.10.2011)
Published in Journal of cellular biochemistry (01.10.2011)
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Substituted Indazoles as Nav1.7 Blockers for the Treatment of Pain
Frost, Jennifer M, DeGoey, David A, Shi, Lei, Gum, Rebecca J, Fricano, Meagan M, Lundgaard, Greta L, El-Kouhen, Odile F, Hsieh, Gin C, Neelands, Torben, Matulenko, Mark A, Daanen, Jerome F, Pai, Madhavi, Ghoreishi-Haack, Nayereh, Zhan, Cenchen, Zhang, Xu-Feng, Kort, Michael E
Published in Journal of medicinal chemistry (14.04.2016)
Published in Journal of medicinal chemistry (14.04.2016)
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Journal Article
Protein kinase C-related kinase targets nuclear localization signals in a subset of class IIa histone deacetylases
Harrison, Brooke C., Huynh, Khai, Lundgaard, Greta L., Helmke, Steven M., Perryman, M. Benjamin, McKinsey, Timothy A.
Published in FEBS letters (19.03.2010)
Published in FEBS letters (19.03.2010)
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Discovery of (R)-(3-fluoropyrrolidin-1-yl)(6-((5-(trifluoromethyl) pyridin-2-yl)oxy)quinolin-2-yl)methanone (ABBV-318) and analogs as small molecule Na(v)1.7/Nav1.8 blockers for the treatment of pain
Patel, Meena, Peltier, Hillary M., Matulenko, Mark A., Koenig, John R., Scanio, Marc J. C., Gum, Rebecca J., El-Kouhen, Odile F., Fricano, Meagan M., Lundgaard, Greta L., Neelands, Torben, Zhang, Xu-Feng, Zhan, Cenchen, Pai, Madhavi, Ghoreishi-Haack, Nayereh, Hudzik, Thomas, Gintant, Gary, Martin, Ruth, McGaraughty, Steve, Xu, Jun, Bow, Daniel, Kalvass, John C., Kym, Philip R., DeGoey, David A., Kort, Michael E.
Published in Bioorganic & medicinal chemistry (01.06.2022)
Published in Bioorganic & medicinal chemistry (01.06.2022)
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Journal Article
Substituted Indazoles as Na(v)1.7 Blockers for the Treatment of Pain
Frost, Jennifer M., DeGoey, David A., Shi, Lei, Gum, Rebecca J., Fricano, Meagan M., Lundgaard, Greta L., El-Kouhen, Odile F., Hsieh, Gin C., Neelands, Torben, Matulenko, Mark A., Daanen, Jerome F., Pai, Madhavi, Ghoreishi-Haack, Nayereh, Zhan, Cenchen, Zhang, Xu-Feng, Kort, Michael E.
Published in Journal of medicinal chemistry (14.04.2016)
Published in Journal of medicinal chemistry (14.04.2016)
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Journal Article
Discovery of (R)-(3-fluoropyrrolidin-1-yl)(6-((5-(trifluoromethyl)pyridin-2-yl)oxy)quinolin-2-yl)methanone (ABBV-318) and analogs as small molecule Na v 1.7/ Nav1.8 blockers for the treatment of pain
Patel, Meena V, Peltier, Hillary M, Matulenko, Mark A, Koenig, John R, C Scanio, Marc J, Gum, Rebecca J, El-Kouhen, Odile F, Fricano, Meagan M, Lundgaard, Greta L, Neelands, Torben, Zhang, Xu-Feng, Zhan, Cenchen, Pai, Madhavi, Ghoreishi-Haack, Nayereh, Hudzik, Thomas, Gintant, Gary, Martin, Ruth, McGaraughty, Steve, Xu, Jun, Bow, Daniel, Kalvass, John C, Kym, Philip R, DeGoey, David A, Kort, Michael E
Published in Bioorganic & medicinal chemistry (01.06.2022)
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Published in Bioorganic & medicinal chemistry (01.06.2022)
Journal Article
Substituted Indazoles as Na v 1.7 Blockers for the Treatment of Pain
Frost, Jennifer M., DeGoey, David A., Shi, Lei, Gum, Rebecca J., Fricano, Meagan M., Lundgaard, Greta L., El-Kouhen, Odile F., Hsieh, Gin C., Neelands, Torben, Matulenko, Mark A., Daanen, Jerome F., Pai, Madhavi, Ghoreishi-Haack, Nayereh, Zhan, Cenchen, Zhang, Xu-Feng, Kort, Michael E.
Published in Journal of medicinal chemistry (14.04.2016)
Published in Journal of medicinal chemistry (14.04.2016)
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TERTIARY AMIDES AND METHOD OF USE
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Year of Publication 25.04.2019
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Year of Publication 25.04.2019
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TERTIARY AMIDES AND METHOD OF USE
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Year of Publication 30.11.2017
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Year of Publication 30.11.2017
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TERTIARY AMIDES AND METHOD OF USE
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Year of Publication 12.10.2017
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Year of Publication 25.07.2018
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Year of Publication 25.07.2018
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Tertiary amides and method of use
ZHANG, QINGWEI, ZHU, WEI, BUNNELLE, WILLIAM H, DENG, XIANG-JUN, TAO, RUI-HONG, DEGOEY, DAVID A, LI, MING-FENG, ZHANG, LIN, FU, LI-QIANG, CLAPHAM, BRUCE, BLACK, LAWRENCE A, LUNDGAARD, GRETA L, CHEN, DA, HAZELWOOD, LISA A, PATEL, MEENA V, ZHENG, QIAN-GANG, LANG, QING-YU, KONG, LING-LONG, LEE, CHIH-HUNG
Year of Publication 01.11.2017
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Year of Publication 01.11.2017
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