An orally available, brain penetrant, small molecule lowers huntingtin levels by enhancing pseudoexon inclusion
Keller, Caroline Gubser, Shin, Youngah, Monteys, Alex Mas, Renaud, Nicole, Beibel, Martin, Teider, Natalia, Peters, Thomas, Faller, Thomas, St-Cyr, Sophie, Knehr, Judith, Roma, Guglielmo, Reyes, Alejandro, Hild, Marc, Lukashev, Dmitriy, Theil, Diethilde, Dales, Natalie, Cha, Jang-Ho, Borowsky, Beth, Dolmetsch, Ricardo, Davidson, Beverly L, Sivasankaran, Rajeev
Published in Nature communications (03.03.2022)
Published in Nature communications (03.03.2022)
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Immunological mechanisms of the antitumor effects of supplemental oxygenation
Hatfield, Stephen M, Kjaergaard, Jorgen, Lukashev, Dmitriy, Schreiber, Taylor H, Belikoff, Bryan, Abbott, Robert, Sethumadhavan, Shalini, Philbrook, Phaethon, Ko, Kami, Cannici, Ryan, Thayer, Molly, Rodig, Scott, Kutok, Jeffrey L, Jackson, Edwin K, Karger, Barry, Podack, Eckhard R, Ohta, Akio, Sitkovsky, Michail V
Published in Science translational medicine (04.03.2015)
Published in Science translational medicine (04.03.2015)
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Journal Article
A2A Adenosine Receptor Protects Tumors from Antitumor T Cells
Ohta, Akio, Gorelik, Elieser, Prasad, Simon J., Ronchese, Franca, Lukashev, Dmitriy, Wong, Michael K. K., Huang, Xiaojun, Caldwell, Sheila, Liu, Kebin, Smith, Patrick, Chen, Jiang-Fan, Jackson, Edwin K., Apasov, Sergey, Abrams, Scott, Sitkovsky, Michail
Published in Proceedings of the National Academy of Sciences - PNAS (29.08.2006)
Published in Proceedings of the National Academy of Sciences - PNAS (29.08.2006)
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Journal Article
Toll-like Receptor 3 Regulates Angiogenesis and Apoptosis in Prostate Cancer Cell Lines through Hypoxia-Inducible Factor 1α
Paone, Alessio, Galli, Roberta, Gabellini, Chiara, Lukashev, Dmitriy, Starace, Donatella, Gorlach, Agnes, De Cesaris, Paola, Ziparo, Elio, Del Bufalo, Donatella, Sitkovsky, Michail V., Filippini, Antonio, Riccioli, Anna
Published in Neoplasia (New York, N.Y.) (01.07.2010)
Published in Neoplasia (New York, N.Y.) (01.07.2010)
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1,3,7-Trimethylxanthine (Caffeine) May Exacerbate Acute Inflammatory Liver Injury by Weakening the Physiological Immunosuppressive Mechanism
Ohta, Akio, Lukashev, Dmitriy, Jackson, Edwin K, Fredholm, Bertil B, Sitkovsky, Michail
Published in The Journal of immunology (1950) (01.12.2007)
Published in The Journal of immunology (1950) (01.12.2007)
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Sphingosine-1-Phosphate Reduces CD4+ T-Cell Activation in Type 1 Diabetes Through Regulation of Hypoxia-Inducible Factor Short Isoform I.1 and CD69
SRINIVASAN, Suseela, BOLICK, David T, LUKASHEV, Dmitriy, LAPPAS, Courtney, SITKOVSKY, Michail, LYNCH, Kevin R, HEDRICK, Catherine C
Published in Diabetes (New York, N.Y.) (01.02.2008)
Published in Diabetes (New York, N.Y.) (01.02.2008)
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Analysis of A2a receptor-deficient mice reveals no significant compensatory increases in the expression of A2b, A1, and A3 adenosine receptors in lymphoid organs
Lukashev, Dmitriy E, Smith, Patrick T, Caldwell, Charles C, Ohta, Akio, Apasov, Sergey G, Sitkovsky, Michail V
Published in Biochemical pharmacology (15.06.2003)
Published in Biochemical pharmacology (15.06.2003)
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Journal Article
Regulated control of gene therapies by drug-induced splicing
Monteys, Alex Mas, Hundley, Amiel A, Ranum, Paul T, Tecedor, Luis, Muehlmatt, Amy, Lim, Euyn, Lukashev, Dmitriy, Sivasankaran, Rajeev, Davidson, Beverly L
Published in Nature (London) (12.08.2021)
Published in Nature (London) (12.08.2021)
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Journal Article
Physiological regulation of acute inflammation by A2A adenosine receptor
Lukashev, Dmitriy E., Ohta, Akio, Sitkovsky, Michail V.
Published in Drug development research (01.03.2005)
Published in Drug development research (01.03.2005)
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Journal Article
Systemic oxygenation weakens the hypoxia and hypoxia inducible factor 1α-dependent and extracellular adenosine-mediated tumor protection
Hatfield, Stephen M., Kjaergaard, Jorgen, Lukashev, Dmitriy, Belikoff, Bryan, Schreiber, Taylor H., Sethumadhavan, Shalini, Abbott, Robert, Philbrook, Phaethon, Thayer, Molly, Shujia, Dai, Rodig, Scott, Kutok, Jeffrey L., Ren, Jin, Ohta, Akio, Podack, Eckhard R., Karger, Barry, Jackson, Edwin K., Sitkovsky, Michail
Published in Journal of molecular medicine (Berlin, Germany) (01.12.2014)
Published in Journal of molecular medicine (Berlin, Germany) (01.12.2014)
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Physiological control of immune response and inflammatory tissue damage by hypoxia-inducible factors and adenosine A2A receptors
Sitkovsky, Michail V, Lukashev, Dmitriy, Apasov, Sergey, Kojima, Hidefumi, Koshiba, Masahiro, Caldwell, Charles, Ohta, Akio, Thiel, Manfred
Published in Annual review of immunology (2004)
Published in Annual review of immunology (2004)
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Cutting Edge: Hypoxia-Inducible Factor 1α and Its Activation-Inducible Short Isoform I.1 Negatively Regulate Functions of CD4+ and CD8+ T Lymphocytes
Lukashev, Dmitriy, Klebanov, Boris, Kojima, Hidefumi, Grinberg, Alex, Ohta, Akiko, Berenfeld, Ludmilla, Wenger, Roland H., Ohta, Akio, Sitkovsky, Michail
Published in The Journal of immunology (1950) (15.10.2006)
Published in The Journal of immunology (1950) (15.10.2006)
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Author Correction: Regulated control of gene therapies by drug-induced splicing
Monteys, Alex Mas, Hundley, Amiel A, Ranum, Paul T, Tecedor, Luis, Muehlmatt, Amy, Lim, Euyn, Lukashev, Dmitriy, Sivasankaran, Rajeev, Davidson, Beverly L
Published in Nature (London) (17.02.2022)
Published in Nature (London) (17.02.2022)
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Journal Article
A2B adenosine receptor blockade enhances macrophage-mediated bacterial phagocytosis and improves polymicrobial sepsis survival in mice
Belikoff, Bryan G, Hatfield, Stephen, Georgiev, Peter, Ohta, Akio, Lukashev, Dmitriy, Buras, Jon A, Remick, Daniel G, Sitkovsky, Michail
Published in The Journal of immunology (1950) (15.02.2011)
Published in The Journal of immunology (1950) (15.02.2011)
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