Understanding the role of Leu22 variants in methotrexate resistance: comparison of wild-type and Leu22Arg variant mouse and human dihydrofolate reductase ternary crystal complexes with methotrexate and NADPH
Cody, Vivian, Luft, Joe R., Pangborn, Walt
Published in Acta crystallographica. Section D, Biological crystallography. (01.02.2005)
Published in Acta crystallographica. Section D, Biological crystallography. (01.02.2005)
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Structure-Based Design and Synthesis of Lipophilic 2,4-Diamino-6-Substituted Quinazolines and Their Evaluation as Inhibitors of Dihydrofolate Reductases and Potential Antitumor Agents
Gangjee, Aleem, Vidwans, Anup P, Vasudevan, Anil, Queener, Sherry F, Kisliuk, Roy L, Cody, Vivian, Li, Ruming, Galitsky, Nikolai, Luft, Joe R, Pangborn, Walter
Published in Journal of medicinal chemistry (27.08.1998)
Published in Journal of medicinal chemistry (27.08.1998)
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Structure determination of tetrahydroquinazoline antifolates in complex with human and Pneumocystis carinii dihydrofolate reductase: correlations between enzyme selectivity and stereochemistry
Cody, Vivian, Luft, Joe R., Pangborn, Walt, Gangjee, Aleem, Queener, Sherry F.
Published in Acta crystallographica. Section D, Biological crystallography. (01.04.2004)
Published in Acta crystallographica. Section D, Biological crystallography. (01.04.2004)
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Automatic classification of sub-microlitre protein-crystallization trials in 1536-well plates
Cumbaa, Christian A., Lauricella, Angela, Fehrman, Nancy, Veatch, Christina, Collins, Robert, Luft, Joe, DeTitta, George, Jurisica, Igor
Published in Acta crystallographica. Section D, Biological crystallography. (01.09.2003)
Published in Acta crystallographica. Section D, Biological crystallography. (01.09.2003)
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Selective Pneumocystis carinii Dihydrofolate Reductase Inhibitors: Design, Synthesis, and Biological Evaluation of New 2,4-Diamino-5-substituted-furo[2,3-d]pyrimidines
Gangjee, Aleem, Guo, Xin, Queener, Sherry F., Cody, Vivian, Galitsky, Nikolai, Luft, Joe R., Pangborn, Walter
Published in Journal of medicinal chemistry (09.04.1998)
Published in Journal of medicinal chemistry (09.04.1998)
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