Mutational profiling of SARS-CoV-2 papain-like protease reveals requirements for function, structure, and drug escape
Wu, Xinyu, Go, Margareta, Nguyen, Julie V., Kuchel, Nathan W., Lu, Bernadine G. C., Zeglinski, Kathleen, Lowes, Kym N., Calleja, Dale J., Mitchell, Jeffrey P., Lessene, Guillaume, Komander, David, Call, Matthew E., Call, Melissa J.
Published in Nature communications (23.07.2024)
Published in Nature communications (23.07.2024)
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Mechanism and inhibition of the papain‐like protease, PLpro, of SARS‐CoV‐2
Klemm, Theresa, Ebert, Gregor, Calleja, Dale J, Allison, Cody C, Richardson, Lachlan W, Bernardini, Jonathan P, Lu, Bernadine GC, Kuchel, Nathan W, Grohmann, Christoph, Shibata, Yuri, Gan, Zhong Yan, Cooney, James P, Doerflinger, Marcel, Au, Amanda E, Blackmore, Timothy R, Heden van Noort, Gerbrand J, Geurink, Paul P, Ovaa, Huib, Newman, Janet, Riboldi‐Tunnicliffe, Alan, Czabotar, Peter E, Mitchell, Jeffrey P, Feltham, Rebecca, Lechtenberg, Bernhard C, Lowes, Kym N, Dewson, Grant, Pellegrini, Marc, Lessene, Guillaume, Komander, David
Published in The EMBO journal (15.09.2020)
Published in The EMBO journal (15.09.2020)
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Insights Into Drug Repurposing, as Well as Specificity and Compound Properties of Piperidine-Based SARS-CoV-2 PLpro Inhibitors
Calleja, Dale J, Kuchel, Nathan, Lu, Bernadine G C, Birkinshaw, Richard W, Klemm, Theresa, Doerflinger, Marcel, Cooney, James P, Mackiewicz, Liana, Au, Amanda E, Yap, Yu Q, Blackmore, Timothy R, Katneni, Kasiram, Crighton, Elly, Newman, Janet, Jarman, Kate E, Call, Melissa J, Lechtenberg, Bernhard C, Czabotar, Peter E, Pellegrini, Marc, Charman, Susan A, Lowes, Kym N, Mitchell, Jeffrey P, Nachbur, Ueli, Lessene, Guillaume, Komander, David
Published in Frontiers in chemistry (12.04.2022)
Published in Frontiers in chemistry (12.04.2022)
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i-bodies, Human Single Domain Antibodies That Antagonize Chemokine Receptor CXCR4
Griffiths, Katherine, Dolezal, Olan, Cao, Benjamin, Nilsson, Susan K., See, Heng B., Pfleger, Kevin D.G., Roche, Michael, Gorry, Paul R., Pow, Andrew, Viduka, Katerina, Lim, Kevin, Lu, Bernadine G.C., Chang, Denison H.C., Murray-Rust, Thomas, Kvansakul, Marc, Perugini, Matthew A., Dogovski, Con, Doerflinger, Marcel, Zhang, Yuan, Parisi, Kathy, Casey, Joanne L., Nuttall, Stewart D., Foley, Michael
Published in The Journal of biological chemistry (10.06.2016)
Published in The Journal of biological chemistry (10.06.2016)
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The X-ray Crystal Structure of Full-Length Human Plasminogen
Law, Ruby H.P., Caradoc-Davies, Tom, Cowieson, Nathan, Horvath, Anita J., Quek, Adam J., Encarnacao, Joanna Amarante, Steer, David, Cowan, Angus, Zhang, Qingwei, Lu, Bernadine G.C., Pike, Robert N., Smith, A. Ian, Coughlin, Paul B., Whisstock, James C.
Published in Cell reports (Cambridge) (29.03.2012)
Published in Cell reports (Cambridge) (29.03.2012)
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Methods to measure the kinetics of protease inhibition by serpins
Horvath, Anita J, Lu, Bernadine G C, Pike, Robert N, Bottomley, Stephen P
Published in Methods in enzymology (2011)
Published in Methods in enzymology (2011)
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Mechanism and inhibition of SARS-CoV-2 PLpro
Klemm, Theresa, Ebert, Gregor, Calleja, Dale J, Allison, Cody C, Richardson, Lachlan W, Bernardini, Jonathan P, Lu, Bernadine G C, Kuchel, Nathan W, Grohmann, Christoph, Shibata, Yuri, Zhong Yan Gan, Cooney, James P, Doerflinger, Marcel, Au, Amanda E, Blackmore, Timothy R, Geurink, Paul P, Ovaa, Huib, Newman, Janet, Riboldi-Tunnicliffe, Alan, Czabotar, Peter E, Mitchell, Jeffrey P, Feltham, Rebecca, Lechtenberg, Bernhard C, Lowes, Kym N, Dewson, Grant, Pellegrini, Marc, Lessene, Guillaume, Komander, David
Published in bioRxiv (19.06.2020)
Published in bioRxiv (19.06.2020)
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