Characterization of SB‐269970‐A, a selective 5‐HT7 receptor antagonist
Hagan, Jim J, Price, Gary W, Jeffrey, Phillip, Deeks, Nigel J, Stean, Tania, Piper, David, Smith, Martin I, Upton, Neil, Medhurst, Andrew D, Middlemiss, Derek N, Riley, Graham J, Lovell, Peter J, Bromidge, Steven M, Thomas, David R
Published in British journal of pharmacology (01.06.2000)
Published in British journal of pharmacology (01.06.2000)
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The identification of potent and selective imidazole-based inhibitors of B-Raf kinase
Takle, Andrew K., Brown, Murray J.B., Davies, Susannah, Dean, David K., Francis, Gerraint, Gaiba, Alessandra, Hird, Alex W., King, Frank D., Lovell, Peter J., Naylor, Antoinette, Reith, Alastair D., Steadman, Jon G., Wilson, David M.
Published in Bioorganic & medicinal chemistry letters (15.01.2006)
Published in Bioorganic & medicinal chemistry letters (15.01.2006)
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A Novel, Potent, and Selective 5-HT7 Antagonist: (R)-3-(2-(2-(4-Methylpiperidin-1-yl)ethyl)pyrrolidine-1-sulfonyl)phenol (SB-269970)
Lovell, Peter J, Bromidge, Steven M, Dabbs, Steven, Duckworth, D. Malcolm, Forbes, Ian T, Jennings, Andrew J, King, Frank D, Middlemiss, Derek N, Rahman, Shirley K, Saunders, Damian V, Collin, Lissa L, Hagan, Jim J, Riley, Graham J, Thomas, David R
Published in Journal of medicinal chemistry (10.02.2000)
Published in Journal of medicinal chemistry (10.02.2000)
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Journal Article
Novel 5-HT1A/1B/1D receptors antagonists with potent 5-HT reuptake inhibitory activity
SERAFINOWSKA, Halina T, BLANEY, Frank E, LOVELL, Peter J, MERLO, Giancarlo G, SCOTT, Claire M, SMITH, Paul W, STARR, Kathryn R, WATSON, Jeannette M
Published in Bioorganic & medicinal chemistry letters (15.10.2008)
Published in Bioorganic & medicinal chemistry letters (15.10.2008)
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Journal Article
Discovery of Potent, Orally Bioavailable, Selective 5-HT1A/B/D Receptor Antagonists
Ward, Simon E, Eddershaw, Peter J, Scott, Claire M, Gordon, Laurie J, Lovell, Peter J, Moore, Susan H, Smith, Paul W, Starr, Kathryn R, Thewlis, Kevin M, Watson, Jeannette M
Published in Journal of medicinal chemistry (22.05.2008)
Published in Journal of medicinal chemistry (22.05.2008)
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Journal Article
Studies on a series of potent, orally bioavailable, 5-HT1 receptor ligands—Part II
Ward, Simon E., Eddershaw, Peter, Flynn, Sean T., Gordon, Laurie, Lovell, Peter J., Moore, Susan H., Scott, Claire M., Smith, Paul W., Thewlis, Kevin M., Wyman, Paul A.
Published in Bioorganic & medicinal chemistry letters (15.01.2009)
Published in Bioorganic & medicinal chemistry letters (15.01.2009)
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Journal Article
Studies on a series of potent, orally bioavailable, 5-HT(1) receptor ligands--part II
Ward, Simon E, Eddershaw, Peter, Flynn, Sean T, Gordon, Laurie, Lovell, Peter J, Moore, Susan H, Scott, Claire M, Smith, Paul W, Thewlis, Kevin M, Wyman, Paul A
Published in Bioorganic & medicinal chemistry letters (15.01.2009)
Published in Bioorganic & medicinal chemistry letters (15.01.2009)
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Journal Article
3,4 -Dihydro -2H -benzoxazinones as dual-acting 5-HT1A receptor antagonists and serotonin reuptake inhibitors
LOVELL, Peter J, BLANEY, Frank E, GOODACRE, Caroline J, SCOTT, Claire M, SMITH, Paul W, STARR, Kathryn R, THEWLIS, Kevin M, VONG, Antonio K. K, WARD, Simon E, WATSON, Jeannette M
Published in Bioorganic & medicinal chemistry letters (15.02.2007)
Published in Bioorganic & medicinal chemistry letters (15.02.2007)
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Journal Article
Studies on a series of potent, orally bioavailable, 5-HT1 receptor ligands
WARD, Simon E, JOHNSON, Christopher N, LOVELL, Peter J, SCOTT, Claire M, SMITH, Paul W, STEMP, Geoffrey, THEWLIS, Kevin M, VONG, Antonio K, WATSON, Jeannette M
Published in Bioorganic & medicinal chemistry letters (15.09.2007)
Published in Bioorganic & medicinal chemistry letters (15.09.2007)
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Journal Article
Highly stereoselective addition of organozinc reagents to pentopyranose derived glycals: effect of protecting group and assignment of C-glycoside stereochemistry
Cook, Matthew J, Fletcher, Matthew J.E, Gray, Diane, Lovell, Peter J, Gallagher, Timothy
Published in Tetrahedron (31.05.2004)
Published in Tetrahedron (31.05.2004)
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Journal Article
A series of bisaryl imidazolidin-2-ones has shown to be selective and orally active 5-HT2C receptor antagonists
GOODACRE, Caroline J, BROMIDGE, Steven M, TRAIL, Brenda K, WOOD, Martyn D, CLAPHAM, David, KING, Frank D, LOVELL, Peter J, ALLEN, Mike, CAMPBELL, Lorraine P, HOLLAND, Vicky, RILEY, Graham J, STARR, Kathryn R
Published in Bioorganic & medicinal chemistry letters (15.11.2005)
Published in Bioorganic & medicinal chemistry letters (15.11.2005)
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Journal Article
[3H]‐SB‐269970 – A selective antagonist radioligand for 5‐HT7 receptors
Thomas, David R, Atkinson, Peter J, Ho, Michael, Bromidge, Steven M, Lovell, Peter J, Villani, Anthony J, Hagan, Jim J, Middlemiss, Derek N, Price, Gary W
Published in British journal of pharmacology (01.05.2000)
Published in British journal of pharmacology (01.05.2000)
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Journal Article
(R)-3,N-Dimethyl-N-[1-methyl-3-(4-methylpiperidin-1-yl)propyl]benzenesulfonamide: The First Selective 5-HT7 Receptor Antagonist
Forbes, Ian T, Dabbs, Steven, Duckworth, D. Malcolm, Jennings, Andrew J, King, Frank D, Lovell, Peter J, Brown, Anthony M, Collin, Lissa, Hagan, Jim J, Middlemiss, Derek N, Riley, Graham J, Thomas, David R, Upton, Neil
Published in Journal of medicinal chemistry (26.02.1998)
Published in Journal of medicinal chemistry (26.02.1998)
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Journal Article
Phenyl benzenesulfonamides are novel and selective 5-HT6 antagonists : Identification of N-(2,5-dibromo-3-fluorophenyl)-4-methoxy-3-piperazin-1-ylbenzenesulfonamide (SB-357134)
BROMIDGE, Steven M, CLARKE, Stephen E, NEWMAN, Helen, RILEY, Graham, ROGERS, Derek, ROUTLEDGE, Carol, SERAFINOWSKA, Halina, SMITH, Douglas R, GAGER, Tracey, GRIFFITH, Kerry, JEFFREY, Phillip, JENNINGS, Andrew J, JOINER, Graham F, KING, Frank D, LOVELL, Peter J, MOSS, Stephen F
Published in Bioorganic & medicinal chemistry letters (08.01.2001)
Published in Bioorganic & medicinal chemistry letters (08.01.2001)
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Journal Article
Cover Picture: The Synthesis of Azadirachtin: A Potent Insect Antifeedant (Chem. Eur. J. 34/2008)
Ley, Steven V., Abad-Somovilla, Antonio, Anderson, James C., Ayats, Carles, Bänteli, Rolf, Beckmann, Edith, Boyer, Alistair, Brasca, Maria G., Brice, Abigail, Broughton, Howard B., Burke, Brenda J., Cleator, Ed, Craig, Donald, Denholm, Alastair A., Denton, Ross M., Durand-Reville, Thomas, Gobbi, Luca B., Göbel, Michael, Gray, Brian Lawrence, Grossmann, Robert B., Gutteridge, Claire E., Hahn, Norbert, Harding, Sarah L., Jennens, David C., Jennens, Lynn, Lovell, Peter J., Lovell, Helen J., de la Puente, Mary L., Kolb, Hartmuth C., Koot, Win-Jan, Maslen, Sarah L., McCusker, Catherine F., Mattes, Amos, Pape, Andrew R., Pinto, Andrea, Santafianos, Dinos, Scott, James S., Smith, Stephen C., Somers, Andrew Q., Spilling, Christopher D., Stelzer, Frank, Toogood, Peter L., Turner, Richard M., Veitch, Gemma E., Wood, Anthony, Zumbrunn, Cornelia
Published in Chemistry : a European journal (26.11.2008)
Published in Chemistry : a European journal (26.11.2008)
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Journal Article
Bicyclic piperazinylbenzenesulphonamides are potent and selective 5-HT6 receptor antagonists
BROMIDGE, Steven M, CLARKE, Stephen E, KING, Frank D, LOVELL, Peter J, NEWMAN, Helen, RILEY, Graham, ROUTLEDGE, Carol, SERAFINOWSKA, Halina T, SMITH, Douglas R, THOMAS, David R
Published in Bioorganic & medicinal chemistry letters (20.05.2002)
Published in Bioorganic & medicinal chemistry letters (20.05.2002)
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Journal Article
The Synthesis of Azadirachtin: A Potent Insect Antifeedant
Ley, Steven V., Abad-Somovilla, Antonio, Anderson, James C., Ayats, Carles, Bänteli, Rolf, Beckmann, Edith, Boyer, Alistair, Brasca, Maria G., Brice, Abigail, Broughton, Howard B., Burke, Brenda J., Cleator, Ed, Craig, Donald, Denholm, Alastair A., Denton, Ross M., Durand-Reville, Thomas, Gobbi, Luca B., Göbel, Michael, Gray, Brian Lawrence, Grossmann, Robert B., Gutteridge, Claire E., Hahn, Norbert, Harding, Sarah L., Jennens, David C., Jennens, Lynn, Lovell, Peter J., Lovell, Helen J., de la Puente, Mary L., Kolb, Hartmuth C., Koot, Win-Jan, Maslen, Sarah L., McCusker, Catherine F., Mattes, Amos, Pape, Andrew R., Pinto, Andrea, Santafianos, Dinos, Scott, James S., Smith, Stephen C., Somers, Andrew Q., Spilling, Christopher D., Stelzer, Frank, Toogood, Peter L., Turner, Richard M., Veitch, Gemma E., Wood, Anthony, Zumbrunn, Cornelia
Published in Chemistry : a European journal (26.11.2008)
Published in Chemistry : a European journal (26.11.2008)
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