A high-throughput phenotypic screen identifies clofazimine as a potential treatment for cryptosporidiosis
Love, Melissa S, Beasley, Federico C, Jumani, Rajiv S, Wright, Timothy M, Chatterjee, Arnab K, Huston, Christopher D, Schultz, Peter G, McNamara, Case W
Published in PLoS neglected tropical diseases (03.02.2017)
Published in PLoS neglected tropical diseases (03.02.2017)
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The ReFRAME library as a comprehensive drug repurposing library and its application to the treatment of cryptosporidiosis
Janes, Jeff, Young, Megan E., Chen, Emily, Rogers, Nicole H., Burgstaller-Muehlbacher, Sebastian, Hughes, Laura D., Love, Melissa S., Hull, Mitchell V., Kuhen, Kelli L., Woods, Ashley K., Joseph, Sean B., Petrassi, H. Michael, McNamara, Case W., Tremblay, Matthew S., Su, Andrew I., Schultz, Peter G., Chatterjee, Arnab K.
Published in Proceedings of the National Academy of Sciences - PNAS (16.10.2018)
Published in Proceedings of the National Academy of Sciences - PNAS (16.10.2018)
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Journal Article
Pharmacological and genetic activation of cAMP synthesis disrupts cholesterol utilization in Mycobacterium tuberculosis
Wilburn, Kaley M, Montague, Christine R, Qin, Bo, Woods, Ashley K, Love, Melissa S, McNamara, Case W, Schultz, Peter G, Southard, Teresa L, Huang, Lu, Petrassi, H Michael, VanderVen, Brian C
Published in PLoS pathogens (01.02.2022)
Published in PLoS pathogens (01.02.2022)
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Journal Article
High-Content Screening for Cryptosporidium Drug Discovery
Love, Melissa S, McNamara, Case W
Published in Methods in molecular biology (Clifton, N.J.) (01.01.2020)
Published in Methods in molecular biology (Clifton, N.J.) (01.01.2020)
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Journal Article
A suite of phenotypic assays to ensure pipeline diversity when prioritizing drug-like Cryptosporidium growth inhibitors
Jumani, Rajiv S, Hasan, Muhammad M, Stebbins, Erin E, Donnelly, Liam, Miller, Peter, Klopfer, Connor, Bessoff, Kovi, Teixeira, Jose E, Love, Melissa S, McNamara, Case W, Huston, Christopher D
Published in Nature communications (23.04.2019)
Published in Nature communications (23.04.2019)
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Journal Article
Identification of a potent benzoxaborole drug candidate for treating cryptosporidiosis
Lunde, Christopher S, Stebbins, Erin E, Jumani, Rajiv S, Hasan, Md Mahmudul, Miller, Peter, Barlow, John, Freund, Yvonne R, Berry, Pamela, Stefanakis, Rianna, Gut, Jiri, Rosenthal, Philip J, Love, Melissa S, McNamara, Case W, Easom, Eric, Plattner, Jacob J, Jacobs, Robert T, Huston, Christopher D
Published in Nature communications (27.06.2019)
Published in Nature communications (27.06.2019)
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Journal Article
Cryptosporidium life cycle small molecule probing implicates translational repression and an Apetala 2 transcription factor in macrogamont differentiation
Hasan, Muhammad M, Mattice, Ethan B, Teixeira, José E, Jumani, Rajiv S, Stebbins, Erin E, Klopfer, Connor E, Franco, Sebastian E, Love, Melissa S, McNamara, Case W, Huston, Christopher D
Published in PLoS pathogens (26.04.2024)
Published in PLoS pathogens (26.04.2024)
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Journal Article
Bicyclic azetidines kill the diarrheal pathogen Cryptosporidium in mice by inhibiting parasite phenylalanyl-tRNA synthetase
Vinayak, Sumiti, Jumani, Rajiv S, Miller, Peter, Hasan, Muhammad M, McLeod, Briana I, Tandel, Jayesh, Stebbins, Erin E, Teixeira, Jose E, Borrel, Julien, Gonse, Arthur, Zhang, Mingliang, Yu, Xianshui, Wernimont, Amy, Walpole, Chris, Eckley, Sean, Love, Melissa S, McNamara, Case W, Sharma, Manmohan, Sharma, Amit, Scherer, Christina A, Kato, Nobutaka, Schreiber, Stuart L, Melillo, Bruno, Striepen, Boris, Huston, Christopher D, Comer, Eamon
Published in Science translational medicine (30.09.2020)
Published in Science translational medicine (30.09.2020)
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Synthesis and structure-activity relationships of aryl fluorosulfate-based inhibitors as novel antitubercular agents
Yang, Baiyuan, Sukheja, Paridhi, Qin, Bo, Li, Gencheng, Bare, Grant A. L., Cascioferro, Alessandro, Love, Melissa S., Petrassi, H. Michael, Sharpless, K. Barry, Mcnamara, Case W., Chatterjee, Arnab K.
Published in Bioorganic & medicinal chemistry letters (15.01.2024)
Published in Bioorganic & medicinal chemistry letters (15.01.2024)
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Journal Article
Platelet Factor 4 Activity against P. falciparum and Its Translation to Nonpeptidic Mimics as Antimalarials
Love, Melissa S., Millholland, Melanie G., Mishra, Satish, Kulkarni, Swapnil, Freeman, Katie B., Pan, Wenxi, Kavash, Robert W., Costanzo, Michael J., Jo, Hyunil, Daly, Thomas M., Williams, Dewight R., Kowalska, M. Anna, Bergman, Lawrence W., Poncz, Mortimer, DeGrado, William F., Sinnis, Photini, Scott, Richard W., Greenbaum, Doron C.
Published in Cell host & microbe (13.12.2012)
Published in Cell host & microbe (13.12.2012)
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Journal Article
Structure-activity relationship of BMS906024 derivatives for Cryptosporidium parvum growth inhibition
Lee, Seungheon, Love, Melissa S., Modukuri, Ramkumar, Chatterjee, Arnab K., Huerta, Lauren, Lawson, Ann P., McNamara, Case W., Mead, Jan R., Hedstrom, Lizbeth, Cuny, Gregory D.
Published in Bioorganic & medicinal chemistry letters (15.06.2023)
Published in Bioorganic & medicinal chemistry letters (15.06.2023)
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Journal Article
Repurposing the Kinase Inhibitor Mavelertinib for Giardiasis Therapy
Michaels, Samantha A, Hulverson, Matthew A, Whitman, Grant R, Tran, Linh T, Choi, Ryan, Fan, Erkang, McNamara, Case W, Love, Melissa S, Ojo, Kayode K
Published in Antimicrobial agents and chemotherapy (19.07.2022)
Published in Antimicrobial agents and chemotherapy (19.07.2022)
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Journal Article
Pyridopyrimidinones as a new chemotype of calcium dependent protein kinase 1 (CDPK1) inhibitors for Cryptosporidium
Waldron-Young, Elise, Wijitrmektong, Wissarut, Choi, Ryan, Whitman, Grant R., Hulverson, Matthew A., Charania, Raheela, Keelaghan, Aidan, Li, Li, Srinual, Songpol, Nikhar, Sameer, McNamara, Case W., Love, Melissa S., Huerta, Lauren, Bakowski, Malina A., Hu, Ming, Van Voorhis, Wesley C., Mead, Jan R., Cuny, Gregory D.
Published in Molecular and biochemical parasitology (01.12.2024)
Published in Molecular and biochemical parasitology (01.12.2024)
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Journal Article
Pharmacokinetics and Pharmacodynamics of Clofazimine for Treatment of Cryptosporidiosis
Zhang, Cindy X, Love, Melissa S, McNamara, Case W, Chi, Victor, Woods, Ashley K, Joseph, Sean, Schaefer, Deborah A, Betzer, Dana P, Riggs, Michael W, Iroh Tam, Pui-Ying, Van Voorhis, Wesley C, Arnold, Samuel L M
Published in Antimicrobial agents and chemotherapy (18.01.2022)
Published in Antimicrobial agents and chemotherapy (18.01.2022)
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Journal Article
A Host GPCR Signaling Network Required for the Cytolysis of Infected Cells Facilitates Release of Apicomplexan Parasites
Millholland, Melanie G., Mishra, Satish, Dupont, Christopher D., Love, Melissa S., Patel, Bhumit, Shilling, Dustin, Kazanietz, Marcelo G., Foskett, J. Kevin, Hunter, Christopher A., Sinnis, Photini, Greenbaum, Doron C.
Published in Cell host & microbe (16.01.2013)
Published in Cell host & microbe (16.01.2013)
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Journal Article
Advances in bumped kinase inhibitors for human and animal therapy for cryptosporidiosis
Hulverson, Matthew A., Choi, Ryan, Arnold, Samuel L.M., Schaefer, Deborah A., Hemphill, Andrew, McCloskey, Molly C., Betzer, Dana P., Müller, Joachim, Vidadala, Rama S.R., Whitman, Grant R., Rivas, Kasey L., Barrett, Lynn K., Hackman, Robert C., Love, Melissa S., McNamara, Case W., Shaughnessy, Thomas K., Kondratiuk, Alison, Kurnick, Matthew, Banfor, Patricia N., Lynch, James J., Freiberg, Gail M., Kempf, Dale J., Maly, Dustin J., Riggs, Michael W., Ojo, Kayode K., Van Voorhis, Wesley C.
Published in International journal for parasitology (01.10.2017)
Published in International journal for parasitology (01.10.2017)
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Journal Article
Herbicidins from Streptomyces sp. CB01388 Showing Anti-Cryptosporidium Activity
Chen, Jian-Jun, Rateb, Mostafa E, Love, Melissa S, Xu, Zhengren, Yang, Dong, Zhu, Xiangcheng, Huang, Yong, Zhao, Li-Xing, Jiang, Yi, Duan, Yanwen, McNamara, Case W, Shen, Ben
Published in Journal of natural products (Washington, D.C.) (27.04.2018)
Published in Journal of natural products (Washington, D.C.) (27.04.2018)
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