Amaryllidaceae-Type Alkaloids from Pancratium maritimum: Apoptosis-Inducing Effect and Cell Cycle Arrest on Triple-Negative Breast Cancer Cells
Sancha, Shirley A. R., Gomes, Adriana V., Loureiro, Joana B., Saraiva, Lucília, Ferreira, Maria José U.
Published in Molecules (Basel, Switzerland) (06.09.2022)
Published in Molecules (Basel, Switzerland) (06.09.2022)
Get full text
Journal Article
Synthesis, Biological Evaluation, and In Silico Studies of Novel Aminated Xanthones as Potential p53-Activating Agents
Lemos, Agostinho, Gomes, Ana Sara, Loureiro, Joana B, Brandão, Pedro, Palmeira, Andreia, Pinto, Madalena M M, Saraiva, Lucília, Sousa, Maria Emília
Published in Molecules (Basel, Switzerland) (22.05.2019)
Published in Molecules (Basel, Switzerland) (22.05.2019)
Get full text
Journal Article
Structure-Activity Relationship Studies of Chalcones and Diarylpentanoids with Antitumor Activity: Potency and Selectivity Optimization
Moreira, Joana, Loureiro, Joana B, Correia, Danilo, Palmeira, Andreia, Pinto, Madalena M, Saraiva, Lucília, Cidade, Honorina
Published in Pharmaceuticals (Basel, Switzerland) (25.09.2023)
Published in Pharmaceuticals (Basel, Switzerland) (25.09.2023)
Get full text
Journal Article
Metabolism-Guided Optimization of Tryptophanol-Derived Isoindolinone p53 Activators
Barcherini, Valentina, Loureiro, Joana B, Sena, Ana, Madeira, Catarina, Leandro, Paula, Saraiva, Lucília, Antunes, Alexandra M M, Santos, Maria M M
Published in Pharmaceuticals (Basel, Switzerland) (19.01.2023)
Published in Pharmaceuticals (Basel, Switzerland) (19.01.2023)
Get full text
Journal Article
Semi-Synthesis of Small Molecules of Aminocarbazoles: Tumor Growth Inhibition and Potential Impact on p53
Long, Solida, Loureiro, Joana B, Carvalho, Carla, Gales, Luís, Saraiva, Lucília, Pinto, Madalena M M, Puthongking, Ploenthip, Sousa, Emília
Published in Molecules (Basel, Switzerland) (15.03.2021)
Published in Molecules (Basel, Switzerland) (15.03.2021)
Get full text
Journal Article
Counteracting Colon Cancer by Inhibiting Mitochondrial Respiration and Glycolysis with a Selective PKCδ Activator
Bessa, Cláudia, Loureiro, Joana B, Barros, Matilde, Isca, Vera M S, Sardão, Vilma A, Oliveira, Paulo J, Bernardino, Raquel L, Herman-de-Sousa, Carina, Costa, Maria Adelina, Correia-de-Sá, Paulo, Alves, Marco G, Rijo, Patrícia, Saraiva, Lucília
Published in International journal of molecular sciences (01.03.2023)
Published in International journal of molecular sciences (01.03.2023)
Get full text
Journal Article
3-(1,2,3-Triazol-4-yl)-β-Carbolines and 3-(1 H -Tetrazol-5-yl)-β-Carbolines: Synthesis and Evaluation as Anticancer Agents
Ribeiro, João L P, Loureiro, Joana B, Lopes, Susana M M, Saraiva, Lucília, Pinho E Melo, Teresa M V D
Published in Pharmaceuticals (Basel, Switzerland) (03.12.2022)
Published in Pharmaceuticals (Basel, Switzerland) (03.12.2022)
Get full text
Journal Article
Targeting p53 for Melanoma Treatment: Counteracting Tumour Proliferation, Dissemination and Therapeutic Resistance
Loureiro, Joana B, Raimundo, Liliana, Calheiros, Juliana, Carvalho, Carla, Barcherini, Valentina, Lima, Nuno R, Gomes, Célia, Almeida, Maria Inês, Alves, Marco G, Costa, José Luís, Santos, Maria M M, Saraiva, Lucília
Published in Cancers (01.04.2021)
Published in Cancers (01.04.2021)
Get full text
Journal Article
SLMP53-2 Restores Wild-Type-Like Function to Mutant p53 through Hsp70: Promising Activity in Hepatocellular Carcinoma
Gomes, Sara, Bosco, Bartolomeo, Loureiro, Joana B, Ramos, Helena, Raimundo, Liliana, Soares, Joana, Nazareth, Nair, Barcherini, Valentina, Domingues, Lucília, Oliveira, Carla, Bisio, Alessandra, Piazza, Silvano, Bauer, Matthias R, Brás, João P, Almeida, Maria Inês, Gomes, Célia, Reis, Flávio, Fersht, Alan R, Inga, Alberto, Santos, Maria M M, Saraiva, Lucília
Published in Cancers (10.08.2019)
Published in Cancers (10.08.2019)
Get full text
Journal Article
BRCA1/P53: Two strengths in cancer chemoprevention
Raimundo, Liliana, Ramos, Helena, Loureiro, Joana B., Calheiros, Juliana, Saraiva, Lucília
Published in Biochimica et biophysica acta. Reviews on cancer (01.01.2020)
Published in Biochimica et biophysica acta. Reviews on cancer (01.01.2020)
Get full text
Journal Article
New inhibitor of the TAp73 interaction with MDM2 and mutant p53 with promising antitumor activity against neuroblastoma
Gomes, Sara, Raimundo, Liliana, Soares, Joana, Loureiro, Joana B., Leão, Mariana, Ramos, Helena, Monteiro, Madalena N., Lemos, Agostinho, Moreira, Joana, Pinto, Madalena, Chlapek, Petr, Veselska, Renata, Sousa, Emília, Saraiva, Lucília
Published in Cancer letters (01.04.2019)
Published in Cancer letters (01.04.2019)
Get full text
Journal Article
A Diarylpentanoid with Potential Activation of the p53 Pathway: Combination of in silico Screening Studies, Synthesis, and Biological Activity Evaluation
Moreira, Joana, Almeida, Joana, Loureiro, Joana B., Ramos, Helena, Palmeira, Andreia, Pinto, Madalena M., Saraiva, Lucília, Cidade, Honorina
Published in ChemMedChem (06.10.2021)
Published in ChemMedChem (06.10.2021)
Get full text
Journal Article
Targeting the MDM2-p53 protein-protein interaction with prenylchalcones: Synthesis of a small library and evaluation of potential antitumor activity
Brandão, Pedro, Loureiro, Joana B., Carvalho, Sylvie, Hamadou, Meriem Hadjer, Cravo, Sara, Moreira, Joana, Pereira, Daniela, Palmeira, Andreia, Pinto, Madalena, Saraiva, Lucília, Cidade, Honorina
Published in European journal of medicinal chemistry (05.08.2018)
Published in European journal of medicinal chemistry (05.08.2018)
Get full text
Journal Article
Improving anticancer activity towards colon cancer cells with a new p53‐activating agent
Raimundo, Liliana, Espadinha, Margarida, Soares, Joana, Loureiro, Joana B, Alves, Marco G, Santos, Maria M M, Saraiva, Lucília
Published in British journal of pharmacology (01.10.2018)
Published in British journal of pharmacology (01.10.2018)
Get full text
Journal Article
Mutant p53 reactivator SLMP53-2 hinders ultraviolet B radiation-induced skin carcinogenesis
Loureiro, Joana B., Ribeiro, Rita, Nazareth, Nair, Ferreira, Tiago, Lopes, Elizabeth A., Gama, Adelina, Machuqueiro, Miguel, Alves, Marco G., Marabini, Laura, Oliveira, Paula A., Santos, Maria M.M., Saraiva, Lucília
Published in Pharmacological research (01.01.2022)
Published in Pharmacological research (01.01.2022)
Get full text
Journal Article
SLMP53-1 interacts with wild-type and mutant p53 DNA-binding domain and reactivates multiple hotspot mutations
Gomes, Ana Sara, Ramos, Helena, Gomes, Sara, Loureiro, Joana B., Soares, Joana, Barcherini, Valentina, Monti, Paola, Fronza, Gilberto, Oliveira, Carla, Domingues, Lucília, Bastos, Margarida, Dourado, Daniel F.A.R., Carvalho, Ana Luísa, Romão, Maria João, Pinheiro, Benedita, Marcelo, Filipa, Carvalho, Alexandra, Santos, Maria M.M., Saraiva, Lucília
Published in Biochimica et biophysica acta. General subjects (01.01.2020)
Published in Biochimica et biophysica acta. General subjects (01.01.2020)
Get full text
Journal Article
DIMP53‐1: a novel small‐molecule dual inhibitor of p53–MDM2/X interactions with multifunctional p53‐dependent anticancer properties
Soares, Joana, Espadinha, Margarida, Raimundo, Liliana, Ramos, Helena, Gomes, Ana Sara, Gomes, Sara, Loureiro, Joana B., Inga, Alberto, Reis, Flávio, Gomes, Célia, Santos, Maria M. M., Saraiva, Lucília
Published in Molecular oncology (01.06.2017)
Published in Molecular oncology (01.06.2017)
Get full text
Journal Article
Discovery of a small-molecule protein kinase Cδ-selective activator with promising application in colon cancer therapy
Bessa, Cláudia, Soares, Joana, Raimundo, Liliana, Loureiro, Joana B, Gomes, Célia, Reis, Flávio, Soares, Miguel L, Santos, Daniel, Dureja, Chetna, Chaudhuri, Saumya R, Lopez-Haber, Cynthia, Kazanietz, Marcelo G, Gonçalves, Jorge, Simões, Maria F, Rijo, Patrícia, Saraiva, Lucília
Published in Cell death & disease (18.01.2018)
Published in Cell death & disease (18.01.2018)
Get full text
Journal Article
Amaryllidaceae-Type Alkaloids from IPancratium maritimum/I: Apoptosis-Inducing Effect and Cell Cycle Arrest on Triple-Negative Breast Cancer Cells
Sancha, Shirley A. R, Gomes, Adriana V, Loureiro, Joana B, Saraiva, Lucília, Ferreira, Maria José U
Published in Molecules (Basel, Switzerland) (01.09.2022)
Published in Molecules (Basel, Switzerland) (01.09.2022)
Get full text
Journal Article
Development of lipid nanoparticles containing the xanthone LEM2 for topical treatment of melanoma
Malta, Rafaela, Loureiro, Joana B., Costa, Paulo, Sousa, Emília, Pinto, Madalena, Saraiva, Lucília, Amaral, M. Helena
Published in Journal of drug delivery science and technology (01.02.2021)
Published in Journal of drug delivery science and technology (01.02.2021)
Get full text
Journal Article