Search Results - "Loriga, Giovanni" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Biological Effects on μ-Receptors Affinity and Selectivity of Arylpropenyl Chain Structural Modification on Diazatricyclodecane Derivatives

Biological Effects on μ-Receptors Affinity and Selectivity of Arylpropenyl Chain Structural Modification on Diazatricyclodecane Derivatives

by Piras, Sandra, Murineddu, Gabriele, Loriga, Giovanni, Carta, Antonio, Battistello, Enrica, Merighi, Stefania, Gessi, Stefania, Corona, Paola, Asproni, Battistina, Ibba, Roberta, Temml, Veronika, Schuster, Daniela, Pinna, Gérard Aimè
Published in Molecules (Basel, Switzerland) (07.09.2021)

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Synthesis of tricyclic condensed rings incorporating the pyrazole or isoxazole moieties bonded to a 4-piperidinyl substituent

Synthesis of tricyclic condensed rings incorporating the pyrazole or isoxazole moieties bonded to a 4-piperidinyl substituent

by Pinna, Giansalvo, Loriga, Giovanni, Pinna, Gérard A, Chelucci, Giorgio
Published in Molecules (Basel, Switzerland) (10.07.2013)

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Synthesis and application in asymmetric copper(I)-catalyzed allylic oxidation of a new chiral 1,10-phenanthroline derived from pinene

Synthesis and application in asymmetric copper(I)-catalyzed allylic oxidation of a new chiral 1,10-phenanthroline derived from pinene

by Chelucci, Giorgio, Loriga, Giovanni, Murineddu, Gabriele, Pinna, Gerard A
Published in Tetrahedron letters (06.05.2002)

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Synthesis and in vitro evaluation of the anti-viral activity of N-[4-(1H(2H)-benzotriazol-1(2)-yl)phenyl]alkylcarboxamides

Synthesis and in vitro evaluation of the anti-viral activity of N-[4-(1H(2H)-benzotriazol-1(2)-yl)phenyl]alkylcarboxamides

by Carta, Antonio, Loriga, Giovanni, Piras, Sandra, Paglietti, Giuseppe, Ferrone, Marco, Fermeglia, Maurizio, Pricl, Sabrina, La Colla, Paolo, Secci, Barbara, Collu, Gabriella, Loddo, Roberta
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.11.2006)

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Synthesis and Anti-HIV-1 Activity of New Delavirdine Analogues Carrying Arylpyrrole Moieties

Synthesis and Anti-HIV-1 Activity of New Delavirdine Analogues Carrying Arylpyrrole Moieties

by PINNA, Gérard Aimè, LORIGA, Giovanni, MURINEDDU, Gabriele, GRELLA, Giuseppe, MURA, Massimo, VARGIU, Laura, MURGIONI, Chiara, COLLA, Paolo LA
Published in Chemical & pharmaceutical bulletin (01.11.2001)

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Design, synthesis and biological evaluation of 1,5-disubstituted a-amino tetrazole derivatives as non-covalent inflammasome-caspase-1 complex inhibitors with potential application against immune and inflammatory disorders

Design, synthesis and biological evaluation of 1,5-disubstituted a-amino tetrazole derivatives as non-covalent inflammasome-caspase-1 complex inhibitors with potential application against immune and inflammatory disorders

by Ulgheri, Fausta, Spanu, Pietro, Deligia, Francesco, Loriga, Giovanni, Fuggetta, Maria Pia, de Haan, Iris, Chandgudge, Ajay, Groves, Matthew, Domling, Alexander
Published in European journal of medicinal chemistry (05.02.2022)

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Design, synthesis and biological evaluation of 1,5-disubstituted α-amino tetrazole derivatives as non-covalent inflammasome-caspase-1 complex inhibitors with potential application against immune and inflammatory disorders

Design, synthesis and biological evaluation of 1,5-disubstituted α-amino tetrazole derivatives as non-covalent inflammasome-caspase-1 complex inhibitors with potential application against immune and inflammatory disorders

by Ulgheri, Fausta, Spanu, Pietro, Deligia, Francesco, Loriga, Giovanni, Fuggetta, Maria Pia, de Haan, Iris, Chandgudge, Ajay, Groves, Matthew, Domling, Alexander
Published in European journal of medicinal chemistry (05.02.2022)

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Novel thienocycloalkylpyridazinones as useful scaffolds for acetylcholinesterase inhibition and serotonin 5-HT6 receptor interaction

Novel thienocycloalkylpyridazinones as useful scaffolds for acetylcholinesterase inhibition and serotonin 5-HT6 receptor interaction

by Asproni, Battistina, Catto, Marco, Loriga, Giovanni, Murineddu, Gabriele, Corona, Paola, Purgatorio, Rosa, Cichero, Elena, Fossa, Paola, Scarano, Naomi, Martínez, Antón L., Brea, José, Pinna, Gérard A.
Published in Bioorganic & medicinal chemistry (15.04.2023)

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Synthesis and Cytotoxic Activities of Pyrrole[2,3-d]pyridazin-4-one Derivatives

Synthesis and Cytotoxic Activities of Pyrrole[2,3-d]pyridazin-4-one Derivatives

by Murineddu, Gabriele, Cignarella, Giorgio, Chelucci, Giorgio, Loriga, Giovanni, Pinna, Gérard Aimè
Published in Chemical & pharmaceutical bulletin (01.06.2002)

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Tricyclic pyrazoles. Part 1: synthesis and biological evaluation of novel 1,4-dihydroindeno[1,2-c]pyrazol-based ligands for CB1and CB2 cannabinoid receptors

Tricyclic pyrazoles. Part 1: synthesis and biological evaluation of novel 1,4-dihydroindeno[1,2-c]pyrazol-based ligands for CB1and CB2 cannabinoid receptors

by Mussinu, Jean Mario, Ruiu, Stefania, Mulè, Antonio C, Pau, Amedeo, Carai, Mauro A M, Loriga, Giovanni, Murineddu, Gabriele, Pinna, Gérard A
Published in Bioorganic & medicinal chemistry (17.01.2003)

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Pyridinyl- and pyridazinyl-3,6-diazabicyclo[3.1.1]heptane-anilines: Novel selective ligands with subnanomolar affinity for alpha(4)beta(2) nACh receptors

Pyridinyl- and pyridazinyl-3,6-diazabicyclo[3.1.1]heptane-anilines: Novel selective ligands with subnanomolar affinity for alpha(4)beta(2) nACh receptors

by Deligia, Francesco, Murineddu, Gabriele, Gotti, Cecilia, Ragusa, Giulio, Fasoli, Francesca, Sciaccaluga, Miriam, Plutino, Simona, Fucile, Sergio, Loriga, Giovanni, Asproni, Battistina, Pinna, Gerard A.
Published in European journal of medicinal chemistry (25.05.2018)

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Pyridinyl- and pyridazinyl-3,6-diazabicyclo[3.1.1]heptane-anilines: Novel selective ligands with subnanomolar affinity for α4β2 nACh receptors

Pyridinyl- and pyridazinyl-3,6-diazabicyclo[3.1.1]heptane-anilines: Novel selective ligands with subnanomolar affinity for α4β2 nACh receptors

by Deligia, Francesco, Murineddu, Gabriele, Gotti, Cecilia, Ragusa, Giulio, Fasoli, Francesca, Sciaccaluga, Miriam, Plutino, Simona, Fucile, Sergio, Loriga, Giovanni, Asproni, Battistina, Pinna, Gerard A.
Published in European journal of medicinal chemistry (25.05.2018)

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Chromophore-modified bis-benzo[ g]indole carboxamides: synthesis and antiproliferative activity of bis-benzo[ g]indazole-3-carboxamides and related dimers

Chromophore-modified bis-benzo[ g]indole carboxamides: synthesis and antiproliferative activity of bis-benzo[ g]indazole-3-carboxamides and related dimers

by Pinna, Gérard A, Pirisi, Maria A, Mussinu, Jean-Mario, Murineddu, Gabriele, Loriga, Giovanni, Pau, Amedeo, Grella, Giuseppe E
Published in Farmaco (Società chimica italiana : 1989) (01.09.2003)

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Novel thienocycloalkylpyridazinones as useful scaffolds for acetylcholinesterase inhibition and serotonin 5-HT 6 receptor interaction

Novel thienocycloalkylpyridazinones as useful scaffolds for acetylcholinesterase inhibition and serotonin 5-HT 6 receptor interaction

by Asproni, Battistina, Catto, Marco, Loriga, Giovanni, Murineddu, Gabriele, Corona, Paola, Purgatorio, Rosa, Cichero, Elena, Fossa, Paola, Scarano, Naomi, Martínez, Antón L, Brea, José, Pinna, Gérard A
Published in Bioorganic & medicinal chemistry (15.04.2023)

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Novel pyrrolocycloalkylpyrazole analogues as CB1 ligands

Novel pyrrolocycloalkylpyrazole analogues as CB1 ligands

by Asproni, Battistina, Manca, Ilaria, Pinna, Giansalvo, Cichero, Elena, Fossa, Paola, Murineddu, Gabriele, Lazzari, Paolo, Loriga, Giovanni, Pinna, Gérard A.
Published in Chemical biology & drug design (01.01.2018)

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Novel pyrrolocycloalkylpyrazole analogues as CB 1 ligands

Novel pyrrolocycloalkylpyrazole analogues as CB 1 ligands

by Asproni, Battistina, Manca, Ilaria, Pinna, Giansalvo, Cichero, Elena, Fossa, Paola, Murineddu, Gabriele, Lazzari, Paolo, Loriga, Giovanni, Pinna, Gérard A
Published in Chemical biology & drug design (01.01.2018)

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Synthesis, Pharmacological Evaluation, and Docking Studies of Novel Pyridazinone-Based Cannabinoid Receptor Type2 Ligands

Synthesis, Pharmacological Evaluation, and Docking Studies of Novel Pyridazinone-Based Cannabinoid Receptor Type2 Ligands

by Ragusa, Giulio, Bencivenni, Serena, Morales, Paula, Callaway, Tyra, Hurst, Dow P., Asproni, Battistina, Merighi, Stefania, Loriga, Giovanni, Pinna, Gerard A., Reggio, Patricia H., Gessi, Stefania, Murineddu, Gabriele
Published in ChemMedChem (06.06.2018)

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Tricyclic pyrazoles. Part 6. Benzofuro[3,2-c]pyrazole: A versatile architecture for CB2 selective ligands

Tricyclic pyrazoles. Part 6. Benzofuro[3,2-c]pyrazole: A versatile architecture for CB2 selective ligands

by Pinna, Giovanni, Loriga, Giovanni, Lazzari, Paolo, Ruiu, Stefania, Falzoi, Matteo, Frau, Simona, Pau, Amedeo, Murineddu, Gabriele, Asproni, Battistina, Pinna, Gerard A.
Published in European journal of medicinal chemistry (23.07.2014)

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Differential modulation of GABA(A) receptor function by aryl pyrazoles

Differential modulation of GABA(A) receptor function by aryl pyrazoles

by Mascia, Maria Paola, Ledda, Giovanni, Orrù, Alessandro, Marongiu, Alessandro, Loriga, Giovanni, Maciocco, Elisabetta, Biggio, Giovanni, Ruiu, Stefania
Published in European journal of pharmacology (15.06.2014)

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Differential modulation of GABAA receptor function by aryl pyrazoles

Differential modulation of GABAA receptor function by aryl pyrazoles

by Mascia, Maria Paola, Ledda, Giovanni, Orrù, Alessandro, Marongiu, Alessandro, Loriga, Giovanni, Maciocco, Elisabetta, Biggio, Giovanni, Ruiu, Stefania
Published in European journal of pharmacology (15.06.2014)

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