Inhibition of MYC by the SMARCB1 tumor suppressor
Weissmiller, April M., Wang, Jing, Lorey, Shelly L., Howard, Gregory C., Martinez, Ernest, Liu, Qi, Tansey, William P.
Published in Nature communications (01.05.2019)
Published in Nature communications (01.05.2019)
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Interaction of the oncoprotein transcription factor MYC with its chromatin cofactor WDR5 is essential for tumor maintenance
Thomas, Lance R., Adams, Clare M., Wang, Jing, Weissmiller, April M., Creighton, Joy, Lorey, Shelly L., Liu, Qi, Fesik, Stephen W., Eischen, Christine M., Tansey, William P.
Published in Proceedings of the National Academy of Sciences - PNAS (10.12.2019)
Published in Proceedings of the National Academy of Sciences - PNAS (10.12.2019)
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MYC regulates ribosome biogenesis and mitochondrial gene expression programs through its interaction with host cell factor-1
Popay, Tessa M, Wang, Jing, Adams, Clare M, Howard, Gregory Caleb, Codreanu, Simona G, Sherrod, Stacy D, McLean, John A, Thomas, Lance R, Lorey, Shelly L, Machida, Yuichi J, Weissmiller, April M, Eischen, Christine M, Liu, Qi, Tansey, William P
Published in eLife (08.01.2021)
Published in eLife (08.01.2021)
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WDR5 is a conserved regulator of protein synthesis gene expression
Bryan, Audra F, Wang, Jing, Howard, Gregory C, Guarnaccia, Alissa D, Woodley, Chase M, Aho, Erin R, Rellinger, Eric J, Matlock, Brittany K, Flaherty, David K, Lorey, Shelly L, Chung, Dai H, Fesik, Stephen W, Liu, Qi, Weissmiller, April M, Tansey, William P
Published in Nucleic acids research (06.04.2020)
Published in Nucleic acids research (06.04.2020)
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Displacement of WDR5 from Chromatin by a WIN Site Inhibitor with Picomolar Affinity
Aho, Erin R., Wang, Jing, Gogliotti, Rocco D., Howard, Gregory C., Phan, Jason, Acharya, Pankaj, Macdonald, Jonathan D., Cheng, Ken, Lorey, Shelly L., Lu, Bin, Wenzel, Sabine, Foshage, Audra M., Alvarado, Joseph, Wang, Feng, Shaw, J. Grace, Zhao, Bin, Weissmiller, April M., Thomas, Lance R., Vakoc, Christopher R., Hall, Matthew D., Hiebert, Scott W., Liu, Qi, Stauffer, Shaun R., Fesik, Stephen W., Tansey, William P.
Published in Cell reports (Cambridge) (12.03.2019)
Published in Cell reports (Cambridge) (12.03.2019)
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WIN site inhibition disrupts a subset of WDR5 function
Siladi, Andrew J., Wang, Jing, Florian, Andrea C., Thomas, Lance R., Creighton, Joy H., Matlock, Brittany K., Flaherty, David K., Lorey, Shelly L., Howard, Gregory C., Fesik, Stephen W., Weissmiller, April M., Liu, Qi, Tansey, William P.
Published in Scientific reports (03.02.2022)
Published in Scientific reports (03.02.2022)
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Multiple interactions of the oncoprotein transcription factor MYC with the SWI/SNF chromatin remodeler
Woodley, Chase M., Romer, Alexander S., Wang, Jing, Guarnaccia, Alissa D., Elion, David L., Maxwell, Jack N., Guerrazzi, Kiana, McCann, Tyler S., Popay, Tessa M., Matlock, Brittany K., Flaherty, David K., Lorey, Shelly L., Liu, Qi, Tansey, William P., Weissmiller, April M.
Published in Oncogene (20.05.2021)
Published in Oncogene (20.05.2021)
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B cell responses to HIV antigen are a potent correlate of viremia in HIV-1 infection and improve with PD-1 blockade
Nicholas, Katherine J, Zern, Emily K, Barnett, Louise, Smith, Rita M, Lorey, Shelly L, Copeland, Courtney A, Sadagopal, Shanmugalakshmi, Kalams, Spyros A
Published in PloS one (16.12.2013)
Published in PloS one (16.12.2013)
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Structure-based discovery of potent WD repeat domain 5 inhibitors that demonstrate efficacy and safety in preclinical animal models
Teuscher, Kevin B, Chowdhury, Somenath, Meyers, Kenneth M, Tian, Jianhua, Sai, Jiqing, Van Meveren, Mayme, South, Taylor M, Sensintaffar, John L, Rietz, Tyson A, Goswami, Soumita, Wang, Jing, Grieb, Brian C, Lorey, Shelly L, Howard, Gregory C, Liu, Qi, Moore, William J, Stott, Gordon M, Tansey, William P, Lee, Taekyu, Fesik, Stephen W
Published in Proceedings of the National Academy of Sciences - PNAS (03.01.2023)
Published in Proceedings of the National Academy of Sciences - PNAS (03.01.2023)
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Ribosome subunit attrition and activation of the p53-MDM4 axis dominate the response of MLL-rearranged cancer cells to WDR5 WIN site inhibition
Howard, Gregory Caleb, Wang, Jing, Rose, Kristie L, Jones, Camden, Patel, Purvi, Tsui, Tina, Florian, Andrea C, Vlach, Logan, Lorey, Shelly L, Grieb, Brian C, Smith, Brianna N, Slota, Macey J, Reynolds, Elizabeth M, Goswami, Soumita, Savona, Michael R, Mason, Frank M, Lee, Taekyu, Fesik, Stephen, Liu, Qi, Tansey, William P
Published in eLife (29.04.2024)
Published in eLife (29.04.2024)
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Impact of WIN site inhibitor on the WDR5 interactome
Guarnaccia, Alissa D., Rose, Kristie L., Wang, Jing, Zhao, Bin, Popay, Tessa M., Wang, Christina E., Guerrazzi, Kiana, Hill, Salisha, Woodley, Chase M., Hansen, Tyler J., Lorey, Shelly L., Shaw, J. Grace, Payne, William G., Weissmiller, April M., Olejniczak, Edward T., Fesik, Stephen W., Liu, Qi, Tansey, William P.
Published in Cell reports (Cambridge) (19.01.2021)
Published in Cell reports (Cambridge) (19.01.2021)
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Synergistic action of WDR5 and HDM2 inhibitors in SMARCB1-deficient cancer cells
Florian, Andrea C, Woodley, Chase M, Wang, Jing, Grieb, Brian C, Slota, Macey J, Guerrazzi, Kiana, Hsu, Chih-Yuan, Matlock, Brittany K, Flaherty, David K, Lorey, Shelly L, Fesik, Stephen W, Howard, Gregory C, Liu, Qi, Weissmiller, April M, Tansey, William P
Published in NAR cancer (01.03.2022)
Published in NAR cancer (01.03.2022)
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Antiretroviral Therapy Reduces the Magnitude and T Cell Receptor Repertoire Diversity of HIV-Specific T Cell Responses without Changing T Cell Clonotype Dominance
CONRAD, Joseph A, RAMALINGAM, Ramesh K, DUNCAN, Coley B, SMITH, Rita M, JIE WEI, BARNETT, Louise, SIMONS, Brenna C, LOREY, Shelly L, KALAMS, Spyros A
Published in Journal of Virology (01.04.2012)
Published in Journal of Virology (01.04.2012)
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Enhancement of Human Immunodeficiency Virus (HIV)-Specific CD8+ T Cells in Cerebrospinal Fluid Compared to Those in Blood among Antiretroviral Therapy-Naïve HIV-Positive Subjects
SADAGOPAL, Shanmugalakshmi, LOREY, Shelly L, KALAMS, Spyros A, BARNETT, Louise, BASHAM, Rebecca, LEBO, Laurie, ERDEM, Husamettin, HAMAN, Kirsten, AVISON, Malcolm, WADDELL, Kevin, HAAS, David W
Published in Journal of Virology (01.11.2008)
Published in Journal of Virology (01.11.2008)
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Clonal expansion and TCR-independent differentiation shape the HIV-specific CD8+ effector-memory T-cell repertoire in vivo
Meyer-Olson, Dirk, Simons, Brenna C., Conrad, Joseph A., Smith, Rita M., Barnett, Louise, Lorey, Shelly L., Duncan, Coley B., Ramalingam, Ramesh, Kalams, Spyros A.
Published in Blood (22.07.2010)
Published in Blood (22.07.2010)
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Despite Biased TRBV Gene Usage against a Dominant HLA B57-Restricted Epitope, TCR Diversity Can Provide Recognition of Circulating Epitope Variants
Simons, Brenna C, VanCompernolle, Scott E, Smith, Rita M, Wei, Jie, Barnett, Louise, Lorey, Shelly L, Meyer-Olson, Dirk, Kalams, Spyros A
Published in The Journal of immunology (1950) (01.10.2008)
Published in The Journal of immunology (1950) (01.10.2008)
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Enhanced PD-1 Expression by T Cells in Cerebrospinal Fluid Does Not Reflect Functional Exhaustion during Chronic Human Immunodeficiency Virus Type 1 Infection
SADAGOPAL, Shanmugalakshmi, LOREY, Shelly L, BARNETT, Louise, SUTHERLAND, Deborah, BASHAM, Rebecca, ERDEM, Husamettin, KALAMS, Spyros A, HASA, David W
Published in Journal of Virology (01.01.2010)
Published in Journal of Virology (01.01.2010)
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Dominant clonotypes within HIV-specific T cell responses are programmed death-1high and CD127low and display reduced variant cross-reactivity
Conrad, Joseph A, Ramalingam, Ramesh K, Smith, Rita M, Barnett, Louise, Lorey, Shelly L, Wei, Jie, Simons, Brenna C, Sadagopal, Shanmugalakshmi, Meyer-Olson, Dirk, Kalams, Spyros A
Published in The Journal of immunology (1950) (15.06.2011)
Published in The Journal of immunology (1950) (15.06.2011)
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Journal Article
Ribosome subunit attrition and activation of the p53-MDM4 axis dominate the response of MLL-rearranged cancer cells to WDR5 WIN site inhibition
Howard, Gregory C, Wang, Jing, Rose, Kristie Lindsey, Jones, Camden, Patel, Purvi, Tsui, Tina, Florian, Andrea C, Vlach, Logan, Lorey, Shelly L, Grieb, Brian C, Smith, Brianna N, Slota, Macey J, Reynolds, Elizabeth M, Goswami, Soumita, Savona, Michael R, Mason, Frank M, Lee, Taekyu, Fesik, Stephen W, Liu, Qi, Tansey, William P
Published in bioRxiv (10.01.2024)
Published in bioRxiv (10.01.2024)
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