Corrector VX-809 stabilizes the first transmembrane domain of CFTR
Loo, Tip W., Bartlett, M. Claire, Clarke, David M.
Published in Biochemical pharmacology (01.09.2013)
Published in Biochemical pharmacology (01.09.2013)
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Journal Article
Predicting P-glycoprotein-mediated drug transport based on support vector machine and three-dimensional crystal structure of P-glycoprotein
Bikadi, Zsolt, Hazai, Istvan, Malik, David, Jemnitz, Katalin, Veres, Zsuzsa, Hari, Peter, Ni, Zhanglin, Loo, Tip W, Clarke, David M, Hazai, Eszter, Mao, Qingcheng
Published in PloS one (04.10.2011)
Published in PloS one (04.10.2011)
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Journal Article
Human P-glycoprotein Contains a Greasy Ball-and-Socket Joint at the Second Transmission Interface
Loo, Tip W., Bartlett, M. Claire, Clarke, David M.
Published in The Journal of biological chemistry (12.07.2013)
Published in The Journal of biological chemistry (12.07.2013)
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Journal Article
Processing Mutations Disrupt Interactions between the Nucleotide Binding and Transmembrane Domains of P-glycoprotein and the Cystic Fibrosis Transmembrane Conductance Regulator (CFTR)
Loo, Tip W., Bartlett, M. Claire, Clarke, David M.
Published in The Journal of biological chemistry (17.10.2008)
Published in The Journal of biological chemistry (17.10.2008)
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Journal Article
Additive effect of multiple pharmacological chaperones on maturation of CFTR processing mutants
Wang, Ying, Loo, Tip W, Bartlett, M Claire, Clarke, David M
Published in Biochemical journal (01.09.2007)
Published in Biochemical journal (01.09.2007)
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Journal Article
Rhodamine Inhibitors of P-Glycoprotein: An Amide/Thioamide “Switch” for ATPase Activity
Gannon, Michael K, Holt, Jason J, Bennett, Stephanie M, Wetzel, Bryan R, Loo, Tip W, Bartlett, M. Claire, Clarke, David M, Sawada, Geri A, Higgins, J. William, Tombline, Gregory, Raub, Thomas J, Detty, Michael R
Published in Journal of medicinal chemistry (28.05.2009)
Published in Journal of medicinal chemistry (28.05.2009)
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Journal Article
Arginines in the First Transmembrane Segment Promote Maturation of a P-glycoprotein Processing Mutant by Hydrogen Bond Interactions with Tyrosines in Transmembrane Segment 11
Loo, Tip W., Bartlett, M. Claire, Clarke, David M.
Published in The Journal of biological chemistry (05.09.2008)
Published in The Journal of biological chemistry (05.09.2008)
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Journal Article