Effective deploying of a novel DHODH inhibitor against herpes simplex type 1 and type 2 replication
Luganini, Anna, Sibille, Giulia, Mognetti, Barbara, Sainas, Stefano, Pippione, Agnese Chiara, Giorgis, Marta, Boschi, Donatella, Lolli, Marco L., Gribaudo, Giorgio
Published in Antiviral research (01.05.2021)
Published in Antiviral research (01.05.2021)
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Computational Method for Structure-Based Analysis of SAR Transfer
Bonanni, Davide, Lolli, Marco L, Bajorath, Jürgen
Published in Journal of medicinal chemistry (13.02.2020)
Published in Journal of medicinal chemistry (13.02.2020)
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Biochemical characterization of Mycobacterium tuberculosis dihydroorotate dehydrogenase and identification of a selective inhibitor
Alberti, Marta, Sainas, Stefano, Ronchi, Erika, Lolli, Marco L., Boschi, Donatella, Rizzi, Menico, Ferraris, Davide M., Miggiano, Riccardo
Published in FEBS letters (01.08.2023)
Published in FEBS letters (01.08.2023)
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Tandem mass spectrometry of homologous 3‐hydroxyfurazan and nitrile amino acids: Analysis of cooperative interactions and fragmentation processes
Grossert, J. Stuart, Crowell, Andrew M. J., Boschi, Donatella, Lolli, Marco L., White, Robert L.
Published in Journal of mass spectrometry. (01.06.2024)
Published in Journal of mass spectrometry. (01.06.2024)
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Mechanisms of antiviral activity of the new hDHODH inhibitor MEDS433 against respiratory syncytial virus replication
Luganini, Anna, Sibille, Giulia, Pavan, Marta, Mello Grand, Maurizia, Sainas, Stefano, Boschi, Donatella, Lolli, Marco L., Chiorino, Giovanna, Gribaudo, Giorgio
Published in Antiviral research (01.11.2023)
Published in Antiviral research (01.11.2023)
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Use of human Dihydroorotate Dehydrogenase (hDHODH) Inhibitors in Autoimmune Diseases and New Perspectives in Cancer Therapy
Lolli, Marco L, Sainas, Stefano, Pippione, Agnese C, Giorgis, Marta, Boschi, Donatella, Dosio, Franco
Published in Recent patents on anti-cancer drug discovery (01.01.2018)
Published in Recent patents on anti-cancer drug discovery (01.01.2018)
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A comprehensive review of synthetic strategies and SAR studies for the discovery of PfDHODH inhibitors as antimalarial agents. Part 1: triazolopyrimidine, isoxazolopyrimidine and pyrrole-based (DSM) compounds
Sharma, Manmohan, Pandey, Vinita, Poli, Giulio, Tuccinardi, Tiziano, Lolli, Marco L., Vyas, Vivek K.
Published in Bioorganic chemistry (01.05.2024)
Published in Bioorganic chemistry (01.05.2024)
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Journal Article
Targeting Myeloid Differentiation Using Potent 2‑Hydroxypyrazolo[1,5‑a]pyridine Scaffold-Based Human Dihydroorotate Dehydrogenase Inhibitors
Sainas, Stefano, Pippione, Agnese C, Lupino, Elisa, Giorgis, Marta, Circosta, Paola, Gaidano, Valentina, Goyal, Parveen, Bonanni, Davide, Rolando, Barbara, Cignetti, Alessandro, Ducime, Alex, Andersson, Mikael, Järvå, Michael, Friemann, Rosmarie, Piccinini, Marco, Ramondetti, Cristina, Buccinnà, Barbara, Al-Karadaghi, Salam, Boschi, Donatella, Saglio, Giuseppe, Lolli, Marco L
Published in Journal of medicinal chemistry (26.07.2018)
Published in Journal of medicinal chemistry (26.07.2018)
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An alternative conformation of the N-terminal loop of human dihydroorotate dehydrogenase drives binding to a potent antiproliferative agent
Alberti, Marta, Poli, Giulio, Broggini, Luca, Sainas, Stefano, Rizzi, Menico, Boschi, Donatella, Ferraris, Davide M, Martino, Elena, Ricagno, Stefano, Tuccinardi, Tiziano, Lolli, Marco L, Miggiano, Riccardo
Published in Acta crystallographica. Section D, Biological crystallography. (01.06.2024)
Published in Acta crystallographica. Section D, Biological crystallography. (01.06.2024)
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Intramolecular interactions and the neutral loss of ammonia from collisionally activated, protonated ω-aminoalkyl-3-hydroxyfurazans
Grossert, J. Stuart, Boschi, Donatella, Lolli, Marco L., White, Robert L.
Published in European journal of mass spectrometry (Chichester, England) (01.02.2024)
Published in European journal of mass spectrometry (Chichester, England) (01.02.2024)
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Journal Article
Identification of Human Dihydroorotate Dehydrogenase Inhibitor by a Pharmacophore-Based Virtual Screening Study
Galati, Salvatore, Sainas, Stefano, Giorgis, Marta, Boschi, Donatella, Lolli, Marco L., Ortore, Gabriella, Poli, Giulio, Tuccinardi, Tiziano
Published in Molecules (Basel, Switzerland) (07.06.2022)
Published in Molecules (Basel, Switzerland) (07.06.2022)
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Targeting Acute Myelogenous Leukemia Using Potent Human Dihydroorotate Dehydrogenase Inhibitors Based on the 2‑Hydroxypyrazolo[1,5‑a]pyridine Scaffold: SAR of the Biphenyl Moiety
Sainas, Stefano, Giorgis, Marta, Circosta, Paola, Gaidano, Valentina, Bonanni, Davide, Pippione, Agnese C, Bagnati, Renzo, Passoni, Alice, Qiu, Yaqi, Cojocaru, Carina Florina, Canepa, Barbara, Bona, Alessandro, Rolando, Barbara, Mishina, Mariia, Ramondetti, Cristina, Buccinnà, Barbara, Piccinini, Marco, Houshmand, Mohammad, Cignetti, Alessandro, Giraudo, Enrico, Al-Karadaghi, Salam, Boschi, Donatella, Saglio, Giuseppe, Lolli, Marco L
Published in Journal of medicinal chemistry (13.05.2021)
Published in Journal of medicinal chemistry (13.05.2021)
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Journal Article
Targeting Acute Myelogenous Leukemia Using Potent Human Dihydroorotate Dehydrogenase Inhibitors Based on the 2‑Hydroxypyrazolo[1,5‑a]pyridine Scaffold: SAR of the Aryloxyaryl Moiety
Sainas, Stefano, Giorgis, Marta, Circosta, Paola, Poli, Giulio, Alberti, Marta, Passoni, Alice, Gaidano, Valentina, Pippione, Agnese C., Vitale, Nicoletta, Bonanni, Davide, Rolando, Barbara, Cignetti, Alessandro, Ramondetti, Cristina, Lanno, Alessia, Ferraris, Davide M., Canepa, Barbara, Buccinnà, Barbara, Piccinini, Marco, Rizzi, Menico, Saglio, Giuseppe, Al-Karadaghi, Salam, Boschi, Donatella, Miggiano, Riccardo, Tuccinardi, Tiziano, Lolli, Marco L.
Published in Journal of medicinal chemistry (13.10.2022)
Published in Journal of medicinal chemistry (13.10.2022)
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Dihydroorotate dehydrogenase inhibitors in anti-infective drug research
Boschi, Donatella, Pippione, Agnese Chiara, Sainas, Stefano, Lolli, Marco L.
Published in European journal of medicinal chemistry (01.12.2019)
Published in European journal of medicinal chemistry (01.12.2019)
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Journal Article
Hydroxytriazole derivatives as potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitors discovered by bioisosteric scaffold hopping approach
Pippione, Agnese C., Giraudo, Alessandro, Bonanni, Davide, Carnovale, Irene M., Marini, Elisabetta, Cena, Clara, Costale, Annalisa, Zonari, Daniele, Pors, Klaus, Sadiq, Maria, Boschi, Donatella, Oliaro-Bosso, Simonetta, Lolli, Marco L.
Published in European journal of medicinal chemistry (20.10.2017)
Published in European journal of medicinal chemistry (20.10.2017)
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Journal Article
Insight in Quinazoline-based HDAC Inhibitors as Anti-cancer Agents
Martino, Elena, Thakur, Shruti, Kumar, Arun, Yadav, Ashok Kumar, Boschi, Donatella, Kumar, Deepak, Lolli, Marco
Published in Mini reviews in medicinal chemistry (07.06.2024)
Published in Mini reviews in medicinal chemistry (07.06.2024)
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4-Hydroxy-1,2,3-triazole moiety as bioisostere of the carboxylic acid function: a novel scaffold to probe the orthosteric γ-aminobutyric acid receptor binding site
Giraudo, Alessandro, Krall, Jacob, Nielsen, Birgitte, Sørensen, Troels E., Kongstad, Kenneth T., Rolando, Barbara, Boschi, Donatella, Frølund, Bente, Lolli, Marco L.
Published in European journal of medicinal chemistry (05.10.2018)
Published in European journal of medicinal chemistry (05.10.2018)
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Journal Article
Design, synthesis, biological evaluation and X-ray structural studies of potent human dihydroorotate dehydrogenase inhibitors based on hydroxylated azole scaffolds
Sainas, Stefano, Pippione, Agnese C., Giorgis, Marta, Lupino, Elisa, Goyal, Parveen, Ramondetti, Cristina, Buccinnà, Barbara, Piccinini, Marco, Braga, Rodolpho C., Andrade, Carolina H., Andersson, Mikael, Moritzer, Ann-Christin, Friemann, Rosmarie, Mensa, Stefano, Al-Karadaghi, Salam, Boschi, Donatella, Lolli, Marco L.
Published in European journal of medicinal chemistry (31.03.2017)
Published in European journal of medicinal chemistry (31.03.2017)
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Hydroxyazole scaffold-based Plasmodium falciparum dihydroorotate dehydrogenase inhibitors: Synthesis, biological evaluation and X-ray structural studies
Pippione, Agnese C., Sainas, Stefano, Goyal, Parveen, Fritzson, Ingela, Cassiano, Gustavo C., Giraudo, Alessandro, Giorgis, Marta, Tavella, Tatyana A., Bagnati, Renzo, Rolando, Barbara, Caing-Carlsson, Rhawnie, Costa, Fabio T.M., Andrade, Carolina Horta, Al-Karadaghi, Salam, Boschi, Donatella, Friemann, Rosmarie, Lolli, Marco L.
Published in European journal of medicinal chemistry (01.02.2019)
Published in European journal of medicinal chemistry (01.02.2019)
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