The tumor suppressor folliculin inhibits lactate dehydrogenase A and regulates the Warburg effect
Woodford, Mark R, Baker-Williams, Alexander J, Sager, Rebecca A, Backe, Sarah J, Blanden, Adam R, Hashmi, Fiza, Kancherla, Priyanka, Gori, Alessandro, Loiselle, David R, Castelli, Matteo, Serapian, Stefano A, Colombo, Giorgio, Haystead, Timothy A, Jensen, Sandra M, Stetler-Stevenson, William G, Loh, Stewart N, Schmidt, Laura S, Linehan, W Marston, Bah, Alaji, Bourboulia, Dimitra, Bratslavsky, Gennady, Mollapour, Mehdi
Published in Nature structural & molecular biology (01.08.2021)
Published in Nature structural & molecular biology (01.08.2021)
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Post-translational Regulation of FNIP1 Creates a Rheostat for the Molecular Chaperone Hsp90
Sager, Rebecca A., Woodford, Mark R., Backe, Sarah J., Makedon, Alan M., Baker-Williams, Alexander J., DiGregorio, Bryanna T., Loiselle, David R., Haystead, Timothy A., Zachara, Natasha E., Prodromou, Chrisostomos, Bourboulia, Dimitra, Schmidt, Laura S., Linehan, W. Marston, Bratslavsky, Gennady, Mollapour, Mehdi
Published in Cell reports (Cambridge) (29.01.2019)
Published in Cell reports (Cambridge) (29.01.2019)
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Journal Article
An inducible heat shock protein 70 small molecule inhibitor demonstrates anti-dengue virus activity, validating Hsp70 as a host antiviral target
Howe, Matthew K, Speer, Brittany L, Hughes, Philip F, Loiselle, David R, Vasudevan, Subhash, Haystead, Timothy A J
Published in Antiviral research (01.06.2016)
Published in Antiviral research (01.06.2016)
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Journal Article
Expression of membrane Hsp90 is a molecular signature of T cell activation
Scarneo, Scott A, Smith, Aaron P, Favret, Jacob, O'Connell, Robert, Pickeral, Joy, Yang, Kelly W, Ferrari, Guido, Loiselle, David R, Hughes, Philip F, Kulkarni, Manjusha M, Gargesha, Madhusudhana, Scott, Bryan, Roy, Debashish, Haynes, Barton F, Kwiek, Jesse J, Haystead, Timothy A J
Published in Scientific reports (27.10.2022)
Published in Scientific reports (27.10.2022)
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Journal Article
Phosphorylation and Ubiquitination Regulate Protein Phosphatase 5 Activity and Its Prosurvival Role in Kidney Cancer
Dushukyan, Natela, Dunn, Diana M., Sager, Rebecca A., Woodford, Mark R., Loiselle, David R., Daneshvar, Michael, Baker-Williams, Alexander J., Chisholm, John D., Truman, Andrew W., Vaughan, Cara K., Haystead, Timothy A., Bratslavsky, Gennady, Bourboulia, Dimitra, Mollapour, Mehdi
Published in Cell reports (Cambridge) (14.11.2017)
Published in Cell reports (Cambridge) (14.11.2017)
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Copine A Interacts with Actin Filaments and Plays a Role in Chemotaxis and Adhesion
Buccilli, Matthew J, Ilacqua, April N, Han, Mingxi, Banas, Andrew A, Wight, Elise M, Mao, Hanqian, Perry, Samantha P, Salter, Tasha S, Loiselle, David R, Haystead, Timothy A J, Damer, Cynthia K
Published in Cells (Basel, Switzerland) (21.07.2019)
Published in Cells (Basel, Switzerland) (21.07.2019)
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Journal Article
Takinib, a Selective TAK1 Inhibitor, Broadens the Therapeutic Efficacy of TNF-α Inhibition for Cancer and Autoimmune Disease
Totzke, Juliane, Gurbani, Deepak, Raphemot, Rene, Hughes, Philip F., Bodoor, Khaldon, Carlson, David A., Loiselle, David R., Bera, Asim K., Eibschutz, Liesl S., Perkins, Marisha M., Eubanks, Amber L., Campbell, Phillip L., Fox, David A., Westover, Kenneth D., Haystead, Timothy A.J., Derbyshire, Emily R.
Published in Cell chemical biology (17.08.2017)
Published in Cell chemical biology (17.08.2017)
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Journal Article
Targeting therapy-resistant prostate cancer via a direct inhibitor of the human heat shock transcription factor 1
Dong, Bushu, Jaeger, Alex M, Hughes, Philip F, Loiselle, David R, Hauck, J Spencer, Fu, Yao, Haystead, Timothy A, Huang, Jiaoti, Thiele, Dennis J
Published in Science translational medicine (16.12.2020)
Published in Science translational medicine (16.12.2020)
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Transcription factor–driven alternative localization of Cryptococcus neoformans superoxide dismutase
Smith, Aaron D., Garcia-Santamarina, Sarela, Ralle, Martina, Loiselle, David R., Haystead, Timothy A., Thiele, Dennis J.
Published in The Journal of biological chemistry (01.01.2021)
Published in The Journal of biological chemistry (01.01.2021)
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Journal Article
A bioorthogonal chemical reporter for fatty acid synthase–dependent protein acylation
Karthigeyan, Krithika P., Zhang, Lizhi, Loiselle, David R., Haystead, Timothy A.J., Bhat, Menakshi, Yount, Jacob S., Kwiek, Jesse J.
Published in The Journal of biological chemistry (01.11.2021)
Published in The Journal of biological chemistry (01.11.2021)
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Journal Article
Targeting Borrelia burgdorferi HtpG with a berserker molecule, a strategy for anti-microbial development
Carlson, Dave L., Kowalewski, Mark, Bodoor, Khaldon, Lietzan, Adam D., Hughes, Philip F., Gooden, David, Loiselle, David R., Alcorta, David, Dingman, Zoey, Mueller, Elizabeth A., Irnov, Irnov, Modla, Shannon, Chaya, Tim, Caplan, Jeffrey, Embers, Monica, Miller, Jennifer C., Jacobs-Wagner, Christine, Redinbo, Matthew R., Spector, Neil, Haystead, Timothy A.J.
Published in Cell chemical biology (21.03.2024)
Published in Cell chemical biology (21.03.2024)
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Progressive Rod–Cone Degeneration (PRCD) Protein Requires N‑Terminal S‑Acylation and Rhodopsin Binding for Photoreceptor Outer Segment Localization and Maintaining Intracellular Stability
Spencer, William J, Pearring, Jillian N, Salinas, Raquel Y, Loiselle, David R, Skiba, Nikolai P, Arshavsky, Vadim Y
Published in Biochemistry (Easton) (13.09.2016)
Published in Biochemistry (Easton) (13.09.2016)
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Journal Article
A Fluorescent Hsp90 Probe Demonstrates the Unique Association between Extracellular Hsp90 and Malignancy in Vivo
Crowe, Lauren B, Hughes, Philip F, Alcorta, David A, Osada, Takuya, Smith, Aaron P, Totzke, Juliane, Loiselle, David R, Lutz, Isaac D, Gargesha, Madhusudhana, Roy, Debasish, Roques, Jose, Darr, David, Lyerly, H. Kim, Spector, Neil L, Haystead, Timothy A.J
Published in ACS chemical biology (21.04.2017)
Published in ACS chemical biology (21.04.2017)
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Journal Article
A highly selective Hsp90 affinity chromatography resin with a cleavable linker
Hughes, Philip F., Barrott, Jared J., Carlson, David A., Loiselle, David R., Speer, Brittany L., Bodoor, Khaldon, Rund, Lauretta A., Haystead, Timothy A.J.
Published in Bioorganic & medicinal chemistry (15.05.2012)
Published in Bioorganic & medicinal chemistry (15.05.2012)
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Journal Article
Identification of an Allosteric Small-Molecule Inhibitor Selective for the Inducible Form of Heat Shock Protein 70
Howe, Matthew K., Bodoor, Khaldon, Carlson, David A., Hughes, Philip F., Alwarawrah, Yazan, Loiselle, David R., Jaeger, Alex M., Darr, David B., Jordan, Jamie L., Hunter, Lucas M., Molzberger, Eileen T., Gobillot, Theodore A., Thiele, Dennis J., Brodsky, Jeffrey L., Spector, Neil L., Haystead, Timothy A.J.
Published in Chemistry & biology (18.12.2014)
Published in Chemistry & biology (18.12.2014)
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Journal Article
Optical and Radioiodinated Tethered Hsp90 Inhibitors Reveal Selective Internalization of Ectopic Hsp90 in Malignant Breast Tumor Cells
Barrott, Jared J., Hughes, Philip F., Osada, Takuya, Yang, Xiao-Yi, Hartman, Zachary C., Loiselle, David R., Spector, Neil L., Neckers, Len, Rajaram, Narasimhan, Hu, Fangyao, Ramanujam, Nimmi, Vaidyanathan, Ganesan, Zalutsky, Michael R., Lyerly, H. Kim, Haystead, Timothy A.
Published in Chemistry & biology (19.09.2013)
Published in Chemistry & biology (19.09.2013)
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Journal Article
Chemical Modification of Cysteine Residues Is a Misleading Indicator of Their Status as Active Site Residues in the Vitamin K-dependent γ-Glutamyl Carboxylation Reaction
Tie, Jian-Ke, Jin, Da-Yun, Loiselle, David R., Pope, R. Marshall, Straight, David L., Stafford, Darrel W.
Published in The Journal of biological chemistry (24.12.2004)
Published in The Journal of biological chemistry (24.12.2004)
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Journal Article
Improved Protein Identification through the Use of Unstained Gels
Loiselle, David R, Thelin, William R, Parker, Carol E, Dicheva, Nedyalka N, Kesner, Barry A, Mocanu, Viorel, Wang, Frank, Milgram, Sharon L, Warren, Maria R. Esteban, Borchers, Christoph H
Published in Journal of proteome research (01.05.2005)
Published in Journal of proteome research (01.05.2005)
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