Structural basis for PPAR partial or full activation revealed by a novel ligand binding mode
Capelli, Davide, Cerchia, Carmen, Montanari, Roberta, Loiodice, Fulvio, Tortorella, Paolo, Laghezza, Antonio, Cervoni, Laura, Pochetti, Giorgio, Lavecchia, Antonio
Published in Scientific reports (06.10.2016)
Published in Scientific reports (06.10.2016)
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Journal Article
Beyond the Canonical Endocannabinoid System. A Screening of PPAR Ligands as FAAH Inhibitors
Brunetti, Leonardo, Carrieri, Antonio, Piemontese, Luca, Tortorella, Paolo, Loiodice, Fulvio, Laghezza, Antonio
Published in International journal of molecular sciences (01.10.2020)
Published in International journal of molecular sciences (01.10.2020)
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Journal Article
Food Industry Byproducts as Starting Material for Innovative, Green Feed Formulation: A Sustainable Alternative for Poultry Feeding
Brunetti, Leonardo, Leuci, Rosalba, Colonna, Maria Antonietta, Carrieri, Rossana, Celentano, Francesco Emanuele, Bozzo, Giancarlo, Loiodice, Fulvio, Selvaggi, Maria, Tufarelli, Vincenzo, Piemontese, Luca
Published in Molecules (Basel, Switzerland) (25.07.2022)
Published in Molecules (Basel, Switzerland) (25.07.2022)
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A New Series of Aryloxyacetic Acids Endowed with Multi-Target Activity towards Peroxisome Proliferator-Activated Receptors (PPARs), Fatty Acid Amide Hydrolase (FAAH), and Acetylcholinesterase (AChE)
Leuci, Rosalba, Brunetti, Leonardo, Laghezza, Antonio, Piemontese, Luca, Carrieri, Antonio, Pisani, Leonardo, Tortorella, Paolo, Catto, Marco, Loiodice, Fulvio
Published in Molecules (Basel, Switzerland) (31.01.2022)
Published in Molecules (Basel, Switzerland) (31.01.2022)
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Journal Article
Natural Scaffolds with Multi-Target Activity for the Potential Treatment of Alzheimer's Disease
Piemontese, Luca, Vitucci, Gabriele, Catto, Marco, Laghezza, Antonio, Perna, Filippo Maria, Rullo, Mariagrazia, Loiodice, Fulvio, Capriati, Vito, Solfrizzo, Michele
Published in Molecules (Basel, Switzerland) (29.08.2018)
Published in Molecules (Basel, Switzerland) (29.08.2018)
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Journal Article
Chiral phenoxyacetic acid analogues inhibit colon cancer cell proliferation acting as PPARγ partial agonists
Sabatino, Lina, Ziccardi, Pamela, Cerchia, Carmen, Muccillo, Livio, Piemontese, Luca, Loiodice, Fulvio, Colantuoni, Vittorio, Lupo, Angelo, Lavecchia, Antonio
Published in Scientific reports (01.04.2019)
Published in Scientific reports (01.04.2019)
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Journal Article
Combining fatty acid amide hydrolase (FAAH) inhibition with peroxisome proliferator-activated receptor (PPAR) activation: a new potential multi-target therapeutic strategy for the treatment of Alzheimer's disease
Brunetti, Leonardo, Laghezza, Antonio, Loiodice, Fulvio, Tortorella, Paolo, Piemontese, Luca
Published in Neural regeneration research (01.01.2020)
Published in Neural regeneration research (01.01.2020)
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Journal Article
Resveratrol and Its Metabolites Bind to PPARs
Calleri, Enrica, Pochetti, Giorgio, Dossou, Katina S. S., Laghezza, Antonio, Montanari, Roberta, Capelli, Davide, Prada, Ellen, Loiodice, Fulvio, Massolini, Gabriella, Bernier, Michel, Moaddel, Ruin
Published in Chembiochem : a European journal of chemical biology (26.05.2014)
Published in Chembiochem : a European journal of chemical biology (26.05.2014)
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Journal Article
(2-Aminobenzothiazole)-Methyl-1,1-Bisphosphonic Acids: Targeting Matrix Metalloproteinase 13 Inhibition to the Bone
Laghezza, Antonio, Piemontese, Luca, Brunetti, Leonardo, Caradonna, Alessia, Agamennone, Mariangela, Loiodice, Fulvio, Tortorella, Paolo
Published in Pharmaceuticals (Basel, Switzerland) (24.01.2021)
Published in Pharmaceuticals (Basel, Switzerland) (24.01.2021)
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Journal Article
Derivatives of Tenuazonic Acid as Potential New Multi-Target Anti-Alzheimer's Disease Agents
Poliseno, Viviana, Chaves, Sílvia, Brunetti, Leonardo, Loiodice, Fulvio, Carrieri, Antonio, Laghezza, Antonio, Tortorella, Paolo, Magalhães, João D, Cardoso, Sandra M, Santos, M Amélia, Piemontese, Luca
Published in Biomolecules (Basel, Switzerland) (15.01.2021)
Published in Biomolecules (Basel, Switzerland) (15.01.2021)
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Journal Article
Biological Screening and Crystallographic Studies of Hydroxy γ-Lactone Derivatives to Investigate PPARγ Phosphorylation Inhibition
Capelli, Davide, Cazzaniga, Giulia, Mori, Matteo, Laghezza, Antonio, Loiodice, Fulvio, Quaglia, Martina, Negro, Elisa, Meneghetti, Fiorella, Villa, Stefania, Montanari, Roberta
Published in Biomolecules (Basel, Switzerland) (01.04.2023)
Published in Biomolecules (Basel, Switzerland) (01.04.2023)
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Journal Article
Novel Phenothiazine/Donepezil-like Hybrids Endowed with Antioxidant Activity for a Multi-Target Approach to the Therapy of Alzheimer’s Disease
Carocci, Alessia, Barbarossa, Alexia, Leuci, Rosalba, Carrieri, Antonio, Brunetti, Leonardo, Laghezza, Antonio, Catto, Marco, Limongelli, Francesco, Chaves, Sílvia, Tortorella, Paolo, Altomare, Cosimo Damiano, Santos, Maria Amélia, Loiodice, Fulvio, Piemontese, Luca
Published in Antioxidants (23.08.2022)
Published in Antioxidants (23.08.2022)
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Journal Article
An Effective Virtual Screening Protocol To Identify Promising p53–MDM2 Inhibitors
Tortorella, Paolo, Laghezza, Antonio, Durante, Milena, Gomez-Monterrey, Isabel, Bertamino, Alessia, Campiglia, Pietro, Loiodice, Fulvio, Daniele, Simona, Martini, Claudia, Agamennone, Mariangela
Published in Journal of chemical information and modeling (27.06.2016)
Published in Journal of chemical information and modeling (27.06.2016)
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Journal Article
Bone-Seeking Matrix Metalloproteinase Inhibitors for the Treatment of Skeletal Malignancy
Laghezza, Antonio, Piemontese, Luca, Brunetti, Leonardo, Caradonna, Alessia, Agamennone, Mariangela, Di Pizio, Antonella, Pochetti, Giorgio, Montanari, Roberta, Capelli, Davide, Tauro, Marilena, Loiodice, Fulvio, Tortorella, Paolo
Published in Pharmaceuticals (Basel, Switzerland) (01.06.2020)
Published in Pharmaceuticals (Basel, Switzerland) (01.06.2020)
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Journal Article
Betulinic acid is a PPARγ antagonist that improves glucose uptake, promotes osteogenesis and inhibits adipogenesis
Brusotti, Gloria, Montanari, Roberta, Capelli, Davide, Cattaneo, Giulia, Laghezza, Antonio, Tortorella, Paolo, Loiodice, Fulvio, Peiretti, Franck, Bonardo, Bernadette, Paiardini, Alessandro, Calleri, Enrica, Pochetti, Giorgio
Published in Scientific reports (18.07.2017)
Published in Scientific reports (18.07.2017)
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Journal Article
Dual targeting of cancer-related human matrix metalloproteinases and carbonic anhydrases by chiral N-(biarylsulfonyl)-phosphonic acids
Luisi, Grazia, Angelini, Guido, Gasbarri, Carla, Laghezza, Antonio, Agamennone, Mariangela, Loiodice, Fulvio, Supuran, Claudiu T., Campestre, Cristina, Tortorella, Paolo
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2017)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2017)
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Journal Article
Molecular switch for CLC-K Cl⁻ channel block/activation: Optimal pharmacophoric requirements towards high-affinity ligands
Liantonio, Antonella, Picollo, Alessandra, Carbonara, Giuseppe, Fracchiolla, Giuseppe, Tortorella, Paolo, Loiodice, Fulvio, Laghezza, Antonio, Babini, Elena, Zifarelli, Giovanni, Pusch, Michael, Camerino, Diana Conte
Published in Proceedings of the National Academy of Sciences - PNAS (29.01.2008)
Published in Proceedings of the National Academy of Sciences - PNAS (29.01.2008)
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