Screening for amino acid substitutions in the Candida albicans Erg11 protein of azole-susceptible and azole-resistant clinical isolates: new substitutions and a review of the literature
Morio, Florent, Loge, Cedric, Besse, Bernard, Hennequin, Christophe, Le Pape, Patrice
Published in Diagnostic microbiology and infectious disease (01.04.2010)
Published in Diagnostic microbiology and infectious disease (01.04.2010)
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Exosomes as New Biomarkers and Drug Delivery Tools for the Prevention and Treatment of Various Diseases: Current Perspectives
Liu, Qi, Li, Shiying, Dupuy, Amandine, Mai, Hoa le, Sailliet, Nicolas, Logé, Cédric, Robert, J.-Michel H., Brouard, Sophie
Published in International journal of molecular sciences (01.08.2021)
Published in International journal of molecular sciences (01.08.2021)
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New Quinoxaline Derivatives as Dual Pim-1/2 Kinase Inhibitors: Design, Synthesis and Biological Evaluation
Oyallon, Bruno, Brachet-Botineau, Marie, Logé, Cédric, Robert, Thomas, Bach, Stéphane, Ibrahim, Sajida, Raoul, William, Croix, Cécile, Berthelot, Pascal, Guillon, Jean, Pinaud, Noël, Gouilleux, Fabrice, Viaud-Massuard, Marie-Claude, Denevault-Sabourin, Caroline
Published in Molecules (Basel, Switzerland) (06.02.2021)
Published in Molecules (Basel, Switzerland) (06.02.2021)
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New azole antifungals with a fused triazinone scaffold
Montoir, David, Guillon, Rémi, Gazzola, Sophie, Ourliac-Garnier, Isabelle, Soklou, Kossi Efouako, Tonnerre, Alain, Picot, Carine, Planchat, Aurélien, Pagniez, Fabrice, Le Pape, Patrice, Logé, Cédric
Published in European journal of medicinal chemistry (01.03.2020)
Published in European journal of medicinal chemistry (01.03.2020)
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Journal Article
Structure-based design of novel quinoxaline-2-carboxylic acids and analogues as Pim-1 inhibitors
Oyallon, Bruno, Brachet-Botineau, Marie, Logé, Cédric, Bonnet, Pascal, Souab, Mohamed, Robert, Thomas, Ruchaud, Sandrine, Bach, Stéphane, Berthelot, Pascal, Gouilleux, Fabrice, Viaud-Massuard, Marie-Claude, Denevault-Sabourin, Caroline
Published in European journal of medicinal chemistry (25.06.2018)
Published in European journal of medicinal chemistry (25.06.2018)
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Journal Article
Dibenzofuran Derivatives Inspired from Cercosporamide as Dual Inhibitors of Pim and CLK1 Kinases
Dao, Viet Hung, Ourliac-Garnier, Isabelle, Logé, Cédric, McCarthy, Florence O, Bach, Stéphane, da Silva, Teresinha Gonçalves, Denevault-Sabourin, Caroline, Thiéfaine, Jérôme, Baratte, Blandine, Robert, Thomas, Gouilleux, Fabrice, Brachet-Botineau, Marie, Bazin, Marc-Antoine, Marchand, Pascal
Published in Molecules (Basel, Switzerland) (30.10.2021)
Published in Molecules (Basel, Switzerland) (30.10.2021)
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4-cholesten-3-one decreases breast cancer cell viability and alters membrane raft-localized EGFR expression by reducing lipogenesis and enhancing LXR-dependent cholesterol transporters
Elia, Josiane, Carbonnelle, Delphine, Logé, Cédric, Ory, Lucie, Huvelin, Jean-Michel, Tannoury, Mona, Diab-Assaf, Mona, Petit, Karina, Nazih, Hassan
Published in Lipids in health and disease (02.09.2019)
Published in Lipids in health and disease (02.09.2019)
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Synthesis and molecular modelling studies of 8-arylpyrido[3′,2′:4,5]thieno[3,2-d]pyrimidin-4-amines as multitarget Ser/Thr kinases inhibitors
Loidreau, Yvonnick, Deau, Emmanuel, Marchand, Pascal, Nourrisson, Marie-Renée, Logé, Cédric, Coadou, Gaël, Loaëc, Nadège, Meijer, Laurent, Besson, Thierry
Published in European journal of medicinal chemistry (06.03.2015)
Published in European journal of medicinal chemistry (06.03.2015)
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Journal Article
Discovery of a Novel Broad-Spectrum Antifungal Agent Derived from Albaconazole
Guillon, Rémi, Pagniez, Fabrice, Picot, Carine, Hédou, Damien, Tonnerre, Alain, Chosson, Elizabeth, Duflos, Muriel, Besson, Thierry, Logé, Cédric, Le Pape, Patrice
Published in ACS medicinal chemistry letters (14.02.2013)
Published in ACS medicinal chemistry letters (14.02.2013)
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Journal Article
Potassium 6-Oxo-7,13,16,22-tetraazatetracyclo[12.6.2.18,12.017,21]tricosa-1(20),8(23),9,11,14,16,18,21-octaen-2-yne-15-carboxylate
Blouet, Camille, Letast, Stéphanie, Robert, Thomas, Bach, Stéphane, Pinaud, Noël, Joubert, Nicolas, Viaud-Massuard, Marie-Claude, Guillon, Jean, Logé, Cédric, Denevault-Sabourin, Caroline
Published in MolBank (01.12.2023)
Published in MolBank (01.12.2023)
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Journal Article
Novel synthesis of angular thiazolo[5,4-f] and [4,5-h]quinazolines, preparation of their linear thiazolo[4,5-g] and [5,4-g]quinazoline analogs
Hédou, Damien, Guillon, Rémi, Lecointe, Charlotte, Logé, Cédric, Chosson, Elizabeth, Besson, Thierry
Published in Tetrahedron (15.04.2013)
Published in Tetrahedron (15.04.2013)
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Journal Article
Activation of EGFR by small compounds through coupling the generation of hydrogen peroxide to stable dimerization of Cu/Zn SOD1
Sakanyan, Vehary, Hulin, Philippe, Alves de Sousa, Rodolphe, Silva, Viviane A. O., Hambardzumyan, Artur, Nedellec, Steven, Tomasoni, Christophe, Logé, Cédric, Pineau, Charles, Roussakis, Christos, Fleury, Fabrice, Artaud, Isabelle
Published in Scientific reports (17.02.2016)
Published in Scientific reports (17.02.2016)
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Journal Article
The amino acid substitution N136Y in Candida albicans sterol 14alpha-demethylase is involved in fluconazole resistance
Alvarez-Rueda, Nidia, Fleury, Audrey, Logé, Cédric, Pagniez, Fabrice, Robert, Estelle, Morio, Florent, Le Pape, Patrice
Published in Medical mycology (Oxford) (01.10.2016)
Published in Medical mycology (Oxford) (01.10.2016)
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Synthesis of 3,5-bis(2-indolyl)pyridine and 3-[(2-indolyl)-5-phenyl]pyridine derivatives as CDK inhibitors and cytotoxic agents
Jacquemard, Ulrich, Dias, Nathalie, Lansiaux, Amélie, Bailly, Christian, Logé, Cédric, Robert, Jean-Michel, Lozach, Olivier, Meijer, Laurent, Mérour, Jean-Yves, Routier, Sylvain
Published in Bioorganic & medicinal chemistry (01.05.2008)
Published in Bioorganic & medicinal chemistry (01.05.2008)
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Journal Article
Synthesis of new pyridazino[4,5-b]indol-4-ones and pyridazin-3(2H)-one analogs as DYRK1A inhibitors
Bruel, Amélie, Bénéteau, Romain, Chabanne, Mylène, Lozach, Olivier, Le Guevel, Rémy, Ravache, Myriam, Bénédetti, Hélène, Meijer, Laurent, Logé, Cédric, Robert, Jean-Michel
Published in Bioorganic & medicinal chemistry letters (01.11.2014)
Published in Bioorganic & medicinal chemistry letters (01.11.2014)
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Journal Article
Development of new highly potent imidazo[1,2-b]pyridazines targeting Toxoplasma gondii calcium-dependent protein kinase 1
Moine, Espérance, Dimier-Poisson, Isabelle, Enguehard-Gueiffier, Cécile, Logé, Cédric, Pénichon, Mélanie, Moiré, Nathalie, Delehouzé, Claire, Foll-Josselin, Béatrice, Ruchaud, Sandrine, Bach, Stéphane, Gueiffier, Alain, Debierre-Grockiego, Françoise, Denevault-Sabourin, Caroline
Published in European journal of medicinal chemistry (13.11.2015)
Published in European journal of medicinal chemistry (13.11.2015)
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Novel 9-oxo-thiazolo[5,4- f]quinazoline-2-carbonitrile derivatives as dual cyclin-dependent kinase 1 (CDK1)/glycogen synthase kinase-3 (GSK-3) inhibitors: Synthesis, biological evaluation and molecular modeling studies
Logé, Cédric, Testard, Alexandra, Thiéry, Valérie, Lozach, Olivier, Blairvacq, Mélina, Robert, Jean-Michel, Meijer, Laurent, Besson, Thierry
Published in European journal of medicinal chemistry (01.07.2008)
Published in European journal of medicinal chemistry (01.07.2008)
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Study of N1-alkylation of indoles from the reaction of 2(or 3)-aminoindole-3-(or 2) carbonitriles with DMF-dialkylacetals
Loidreau, Yvonnick, Melissen, Sigismund, Levacher, Vincent, Loge, Cedric, Graton, Jerome, Le Questel, Jean-Yves, Besson, Thierry
Published in Organic & biomolecular chemistry (07.07.2012)
Published in Organic & biomolecular chemistry (07.07.2012)
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Discovery of (7-aryl-1,5-naphthyridin-2-yl)ureas as dual inhibitors of ERK2 and Aurora B kinases with antiproliferative activity against cancer cells
Defaux, Julien, Antoine, Maud, Logé, Cédric, Le Borgne, Marc, Schuster, Tilmann, Seipelt, Irene, Aicher, Babette, Teifel, Michael, Günther, Eckhard, Gerlach, Matthias, Marchand, Pascal
Published in Bioorganic & medicinal chemistry letters (15.08.2014)
Published in Bioorganic & medicinal chemistry letters (15.08.2014)
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