N‑Acylethanolamine Acid Amidase (NAAA): Structure, Function, and Inhibition
Piomelli, Daniele, Scalvini, Laura, Fotio, Yannick, Lodola, Alessio, Spadoni, Gilberto, Tarzia, Giorgio, Mor, Marco
Published in Journal of medicinal chemistry (23.07.2020)
Published in Journal of medicinal chemistry (23.07.2020)
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Theoretical Model of EphA2-Ephrin A1 Inhibition
Jedwabny, Wiktoria, Lodola, Alessio, Dyguda-Kazimierowicz, Edyta
Published in Molecules (Basel, Switzerland) (11.07.2018)
Published in Molecules (Basel, Switzerland) (11.07.2018)
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Selective N-acylethanolamine-hydrolyzing acid amidase inhibition reveals a key role for endogenous palmitoylethanolamide in inflammation
Solorzano, Carlos, Zhu, Chenggang, Battista, Natalia, Astarita, Giuseppe, Lodola, Alessio, Rivara, Silvia, Mor, Marco, Russo, Roberto, Maccarrone, Mauro, Antonietti, Francesca, Duranti, Andrea, Tontini, Andrea, Cuzzocrea, Salvatore, Tarzia, Giorgio, Piomelli, Daniele
Published in Proceedings of the National Academy of Sciences - PNAS (08.12.2009)
Published in Proceedings of the National Academy of Sciences - PNAS (08.12.2009)
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Targeting glucosylceramide synthase induces antiproliferative and proapoptotic effects in osimertinib-resistant NSCLC cell models
La Monica, Silvia, Vacondio, Federica, Eltayeb, Kamal, Lodola, Alessio, Volta, Francesco, Viglioli, Martina, Ferlenghi, Francesca, Galvani, Francesca, Galetti, Maricla, Bonelli, Mara, Fumarola, Claudia, Cavazzoni, Andrea, Flammini, Lisa, Verzè, Michela, Minari, Roberta, Petronini, Pier Giorgio, Tiseo, Marcello, Mor, Marco, Alfieri, Roberta
Published in Scientific reports (18.03.2024)
Published in Scientific reports (18.03.2024)
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Different roles for the acyl chain and the amine leaving group in the substrate selectivity of N-Acylethanolamine acid amidase
Ghidini, Andrea, Scalvini, Laura, Palese, Francesca, Lodola, Alessio, Mor, Marco, Piomelli, Daniele
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2021)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2021)
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Analysis of ADAM12-Mediated Ephrin-A1 Cleavage and Its Biological Functions
Ieguchi, Katsuaki, Tomita, Takeshi, Takao, Toshifumi, Omori, Tsutomu, Mishima, Taishi, Shimizu, Isao, Tognolini, Massimiliano, Lodola, Alessio, Tsunoda, Takuya, Kobayashi, Shinichi, Wada, Satoshi, Maru, Yoshiro
Published in International journal of molecular sciences (01.03.2021)
Published in International journal of molecular sciences (01.03.2021)
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Homology models of melatonin receptors: challenges and recent advances
Pala, Daniele, Lodola, Alessio, Bedini, Annalida, Spadoni, Gilberto, Rivara, Silvia
Published in International Journal of Molecular Sciences (12.04.2013)
Published in International Journal of Molecular Sciences (12.04.2013)
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Book Review
A Pharmacological Investigation of Eph-Ephrin Antagonism in Prostate Cancer: UniPR1331 Efficacy Evidence
Festuccia, Claudio, Corrado, Miriam, Rossetti, Alessandra, Castelli, Riccardo, Lodola, Alessio, Gravina, Giovanni Luca, Tognolini, Massimiliano, Giorgio, Carmine
Published in Pharmaceuticals (Basel, Switzerland) (01.10.2023)
Published in Pharmaceuticals (Basel, Switzerland) (01.10.2023)
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Protein-Protein Interaction Inhibitors Targeting the Eph-Ephrin System with a Focus on Amino Acid Conjugates of Bile Acids
Guidetti, Lorenzo, Castelli, Riccardo, Scalvini, Laura, Ferlenghi, Francesca, Corrado, Miriam, Giorgio, Carmine, Tognolini, Massimiliano, Lodola, Alessio
Published in Pharmaceuticals (Basel, Switzerland) (24.01.2022)
Published in Pharmaceuticals (Basel, Switzerland) (24.01.2022)
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Pushing the Boundaries of Vinylogous Reactivity: Catalytic Enantioselective Mukaiyama Aldol Reactions of Highly Unsaturated 2-Silyloxyindoles
Curti, Claudio, Sartori, Andrea, Battistini, Lucia, Brindani, Nicoletta, Rassu, Gloria, Pelosi, Giorgio, Lodola, Alessio, Mor, Marco, Casiraghi, Giovanni, Zanardi, Franca
Published in Chemistry : a European journal (20.04.2015)
Published in Chemistry : a European journal (20.04.2015)
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Amino Acid Conjugates of Lithocholic Acid As Antagonists of the EphA2 Receptor
Incerti, Matteo, Tognolini, Massimiliano, Russo, Simonetta, Pala, Daniele, Giorgio, Carmine, Hassan-Mohamed, Iftiin, Noberini, Roberta, Pasquale, Elena B, Vicini, Paola, Piersanti, Silvia, Rivara, Silvia, Barocelli, Elisabetta, Mor, Marco, Lodola, Alessio
Published in Journal of medicinal chemistry (11.04.2013)
Published in Journal of medicinal chemistry (11.04.2013)
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Metabolic Soft Spot and Pharmacokinetics: Functionalization of C-3 Position of an Eph-Ephrin Antagonist Featuring a Bile Acid Core as an Effective Strategy to Obtain Oral Bioavailability in Mice
Ferlenghi, Francesca, Giorgio, Carmine, Incerti, Matteo, Guidetti, Lorenzo, Chiodelli, Paola, Rusnati, Marco, Tognolini, Massimiliano, Vacondio, Federica, Mor, Marco, Lodola, Alessio
Published in Pharmaceuticals (Basel, Switzerland) (28.12.2021)
Published in Pharmaceuticals (Basel, Switzerland) (28.12.2021)
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Irreversible Inhibition of Epidermal Growth Factor Receptor Activity by 3-Aminopropanamides
Carmi, Caterina, Galvani, Elena, Vacondio, Federica, Rivara, Silvia, Lodola, Alessio, Russo, Simonetta, Aiello, Stefania, Bordi, Fabrizio, Costantino, Gabriele, Cavazzoni, Andrea, Alfieri, Roberta R, Ardizzoni, Andrea, Petronini, Pier Giorgio, Mor, Marco
Published in Journal of medicinal chemistry (08.03.2012)
Published in Journal of medicinal chemistry (08.03.2012)
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Expanding the Arsenal of FGFR Inhibitors: A Novel Chloroacetamide Derivative as a New Irreversible Agent With Anti-proliferative Activity Against FGFR1-Amplified Lung Cancer Cell Lines
Fumarola, Claudia, Bozza, Nicole, Castelli, Riccardo, Ferlenghi, Francesca, Marseglia, Giuseppe, Lodola, Alessio, Bonelli, Mara, La Monica, Silvia, Cretella, Daniele, Alfieri, Roberta, Minari, Roberta, Galetti, Maricla, Tiseo, Marcello, Ardizzoni, Andrea, Mor, Marco, Petronini, Pier Giorgio
Published in Frontiers in oncology (2019)
Published in Frontiers in oncology (2019)
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Cyclohexylcarbamic Acid 3‘- or 4‘-Substituted Biphenyl-3-yl Esters as Fatty Acid Amide Hydrolase Inhibitors: Synthesis, Quantitative Structure−Activity Relationships, and Molecular Modeling Studies
Mor, Marco, Rivara, Silvia, Lodola, Alessio, Plazzi, Pier Vincenzo, Tarzia, Giorgio, Duranti, Andrea, Tontini, Andrea, Piersanti, Giovanni, Kathuria, Satish, Piomelli, Daniele
Published in Journal of medicinal chemistry (07.10.2004)
Published in Journal of medicinal chemistry (07.10.2004)
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Exploiting Free-Energy Minima to Design Novel EphA2 Protein-Protein Antagonists: From Simulation to Experiment and Return
Russo, Simonetta, Callegari, Donatella, Incerti, Matteo, Pala, Daniele, Giorgio, Carmine, Brunetti, Jlenia, Bracci, Luisa, Vicini, Paola, Barocelli, Elisabetta, Capoferri, Luigi, Rivara, Silvia, Tognolini, Massimiliano, Mor, Marco, Lodola, Alessio
Published in Chemistry : a European journal (06.06.2016)
Published in Chemistry : a European journal (06.06.2016)
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New classes of potent heparanase inhibitors from ligand-based virtual screening
Pala, Daniele, Scalvini, Laura, Elisi, Gian Marco, Lodola, Alessio, Mor, Marco, Spadoni, Gilberto, Ferrara, Fabiana F., Pavoni, Emiliano, Roscilli, Giuseppe, Milazzo, Ferdinando M., Battistuzzi, Gianfranco, Rivara, Silvia, Giannini, Giuseppe
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
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