Structure-activity relationships of actively FhuE transported rifabutin derivatives with potent activity against Acinetobacter baumannii
Maingot, M., Bourotte, M., Vetter, A.C., Schellhorn, B., Antraygues, K., Scherer, H., Gitzinger, M., Kemmer, C., Dale, G.E., Defert, O., Lociuro, S., Brönstrup, M., Willand, N., Trebosc, V.
Published in European journal of medicinal chemistry (05.04.2023)
Published in European journal of medicinal chemistry (05.04.2023)
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In vitro activity of the novel diaminopyrimidine, iclaprim, in combination with folate inhibitors and other antimicrobials with different mechanisms of action
Laue, H., Weiss, L., Bernardi, A., Hawser, S., Lociuro, S., Islam, K.
Published in Journal of antimicrobial chemotherapy (01.12.2007)
Published in Journal of antimicrobial chemotherapy (01.12.2007)
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A microdose study of 14C-AR-709 in healthy men: pharmacokinetics, absolute bioavailability and concentrations in key compartments of the lung
Lappin, G., Boyce, M. J., Matzow, T., Lociuro, S., Seymour, M., Warrington, S. J.
Published in European journal of clinical pharmacology (01.09.2013)
Published in European journal of clinical pharmacology (01.09.2013)
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4″- O-(ω-Quinolylamino-alkylamino)propionyl derivatives of selected macrolides with the activity against the key erythromycin resistant respiratory pathogens
Fajdetić, A., Čipčić Paljetak, H., Lazarevski, G., Hutinec, A., Alihodžić, S., Đerek, M., Štimac, V., Andreotti, D., Šunjić, V., Berge, J.M., Mutak, S., Dumić, M., Lociuro, S., Holmes, D.J., Maršić, N., Eraković Haber, V., Spaventi, R.
Published in Bioorganic & medicinal chemistry (01.09.2010)
Published in Bioorganic & medicinal chemistry (01.09.2010)
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Effect of human plasma on the antimicrobial activity of iclaprim in vitro
Laue, H., Valensise, T., Seguin, A., Hawser, S., Lociuro, S., Islam, K.
Published in Journal of antimicrobial chemotherapy (01.12.2007)
Published in Journal of antimicrobial chemotherapy (01.12.2007)
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Increased hydrophobic interactions of iclaprim with Staphylococcus aureus dihydrofolate reductase are responsible for the increase in affinity and antibacterial activity
Oefner, Christian, Bandera, Monica, Haldimann, Andreas, Laue, Heike, Schulz, Henk, Mukhija, Seema, Parisi, Sandro, Weiss, Laurent, Lociuro, Sergio, Dale, Glenn E.
Published in Journal of antimicrobial chemotherapy (01.04.2009)
Published in Journal of antimicrobial chemotherapy (01.04.2009)
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Synthesis of novel pentacyclic beta-lactam antibacterial agents
Andreotti, D, Biondi, S, Donati, D, Lociuro, S, Pain, G
Published in Canadian journal of chemistry (01.06.2000)
Published in Canadian journal of chemistry (01.06.2000)
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A microdose study of ^sup 14^C-AR-709 in healthy men: pharmacokinetics, absolute bioavailability and concentrations in key compartments of the lung
Lappin, G, Boyce, M J, Matzow, T, Lociuro, S, Seymour, M, Warrington, S J
Published in European journal of clinical pharmacology (01.09.2013)
Published in European journal of clinical pharmacology (01.09.2013)
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A Nutrient-limited Screen Unmasks Rifabutin Hyperactivity for XDR Acinetobacter baumannii
Luna, B., Trebosc, V., Lee, B., Bakowski, M., Ulhaq, A., Yan, J., Lu, P., Cheng, J., Nielsen, T., Lim, J., Ketphan, W., Eoh, H., McNamara, C., Skandalis, N., She, R., Kemmer, C., Lociuro, S., Dale, G. E., Spellberg, B.
Published in Nature microbiology (08.06.2020)
Published in Nature microbiology (08.06.2020)
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Degradation studies of antibiotic MDL 62,879 (GE2270A) and revision of the structure
Tavecchia, Paolo, Gentili, Patrizia, Kurz, Michael, Sottani, Cristina, Bonfichi, Riccardo, Selva, Enrico, Lociuro, Sergio, Restelli, Ermenegildo, Ciabatti, Romeo
Published in Tetrahedron (17.04.1995)
Published in Tetrahedron (17.04.1995)
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Allylic functionalization of 2,5- and 2,4-cyclohexadiene-1,3-dicarboxylates
Seneci, P, Caspani, M, Monti, F, Carrano, L, Lociuro, S
Published in Synthetic communications (01.01.1998)
Published in Synthetic communications (01.01.1998)
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Chemical modification of the GE 2270A macrocycle (MDL 62,879)
Tavecchia, Paolo, Kurz, Michael, Colombo, Luigi, Bonfichi, Riccardo, Selva, Enrico, Lociuro, Sergio, Marzorati, Ettore, Ciabatti, Romeo
Published in Tetrahedron (01.06.1996)
Published in Tetrahedron (01.06.1996)
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REVISED STRUCTURE OF THE ANTIBIOTIC GE 2270A
TAVECCHIA, PAOLO, GENTILI, PATRIZIA, KURZ, MICHAEL, SOTTANI, CRISTINA, BONFICHI, RICCARDO, LOCIURO, SERGIO, SELVA, ENRICO
Published in Journal of antibiotics (1994)
Published in Journal of antibiotics (1994)
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Synthesis and activity studies on 3-(carboxyalkylthio)rifamycin S derivatives
Cellai, L, Martuccio, C, Marzano, M, Onori, BM, Mannina, L, Benedetto, A, DiCaro, A, Lociuro, S, Ripamonti, F
Published in GAZZETTA CHIMICA ITALIANA (01.06.1997)
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Published in GAZZETTA CHIMICA ITALIANA (01.06.1997)
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