Discovery of GLPG3667, a Selective ATP Competitive Tyrosine Kinase 2 Inhibitor for the Treatment of Autoimmune Diseases
Mammoliti, Oscar, Martina, Sébastien, Claes, Pieter, Coti, Ghjuvanni, Blanque, Roland, Jagerschmidt, Catherine, Shoji, Kenji, Borgonovi, Monica, De Vos, Steve, Marsais, Florence, Oste, Line, Quinton, Evelyne, López-Ramos, Miriam, Amantini, David, Brys, Reginald, Jimenez, Juan-Miguel, Galien, René, van der Plas, Steven
Published in Journal of medicinal chemistry (28.05.2024)
Published in Journal of medicinal chemistry (28.05.2024)
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Journal Article
Optimization of Selectivity and Pharmacokinetic Properties of Salt‑Inducible Kinase Inhibitors that Led to the Discovery of Pan-SIK Inhibitor GLPG3312
Temal-Laib, Taouès, Peixoto, Christophe, Desroy, Nicolas, De Lemos, Elsa, Bonnaterre, Florence, Bienvenu, Natacha, Picolet, Olivier, Sartori, Eric, Bucher, Denis, López-Ramos, Miriam, Roca Magadán, Carlos, Laenen, Wendy, Flower, Thomas, Mollat, Patrick, Bugaud, Olivier, Touitou, Robert, Pereira Fernandes, Anna, Lavazais, Stephanie, Monjardet, Alain, Borgonovi, Monica, Gosmini, Romain, Brys, Reginald, Amantini, David, De Vos, Steve, Andrews, Martin
Published in Journal of medicinal chemistry (11.01.2024)
Published in Journal of medicinal chemistry (11.01.2024)
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Journal Article
Discovery of Clinical Candidate GLPG3970: A Potent and Selective Dual SIK2/SIK3 Inhibitor for the Treatment of Autoimmune and Inflammatory Diseases
Peixoto, Christophe, Joncour, Agnes, Temal-Laib, Taouès, Tirera, Amynata, Dos Santos, Aurélie, Jary, Hélène, Bucher, Denis, Laenen, Wendy, Pereira Fernandes, Anna, Lavazais, Stephanie, Delachaume, Carole, Merciris, Didier, Saccomani, Corinne, Drennan, Michael, López-Ramos, Miriam, Wakselman, Emanuelle, Dupont, Sonia, Borgonovi, Monica, Roca Magadan, Carlos, Monjardet, Alain, Brys, Reginald, De Vos, Steve, Andrews, Martin, Jimenez, Juan-Miguel, Amantini, David, Desroy, Nicolas
Published in Journal of medicinal chemistry (11.04.2024)
Published in Journal of medicinal chemistry (11.04.2024)
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Journal Article
HPPD: Ligand- and Target-Based Virtual Screening on a Herbicide Target
López-Ramos, Miriam, Perruccio, Francesca
Published in Journal of chemical information and modeling (24.05.2010)
Published in Journal of chemical information and modeling (24.05.2010)
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Journal Article
New potent dual inhibitors of CK2 and Pim kinases: discovery and structural insights
López-Ramos, Miriam, Prudent, Renaud, Moucadel, Virginie, Sautel, Céline F, Barette, Caroline, Lafanechère, Laurence, Mouawad, Liliane, Grierson, David, Schmidt, Frédéric, Florent, Jean-Claude, Filippakopoulos, Panagis, Bullock, Alex N, Knapp, Stefan, Reiser, Jean-Baptiste, Cochet, Claude
Published in The FASEB journal (01.09.2010)
Published in The FASEB journal (01.09.2010)
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Journal Article
Robust sample size for weibull demonstration test plan
Alvarado Iniesta, Alejandro, Piña Monarrez, Manuel R, Ramos López, Miriam L, Molina Arredondo, Rey D
Published in Dyna (Medellín, Colombia) (01.06.2016)
Published in Dyna (Medellín, Colombia) (01.06.2016)
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Journal Article
Expanding the chemical diversity of CK2 inhibitors
Prudent, Renaud, Moucadel, Virginie, López-Ramos, Miriam, Aci, Samia, Laudet, Beatrice, Mouawad, Liliane, Barette, Caroline, Einhorn, Jacques, Einhorn, Cathy, Denis, Jean-Noel, Bisson, Gilles, Schmidt, Frédéric, Roy, Sylvaine, Lafanechere, Laurence, Florent, Jean-Claude, Cochet, Claude
Published in Molecular and cellular biochemistry (01.09.2008)
Published in Molecular and cellular biochemistry (01.09.2008)
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Journal Article
Progress toward JAK1-selective inhibitors
Menet, Christel J, Mammoliti, Oscar, López-Ramos, Miriam
Published in Future medicinal chemistry (01.01.2015)
Published in Future medicinal chemistry (01.01.2015)
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Journal Article
Salicylaldehyde derivatives as new protein kinase CK2 inhibitors
Prudent, Renaud, López-Ramos, Miriam, Moucadel, Virginie, Barette, Caroline, Grierson, David, Mouawad, Liliane, Florent, Jean-Claude, Lafanechère, Laurence, Schmidt, Frédéric, Cochet, Claude
Published in Biochimica et biophysica acta (01.12.2008)
Published in Biochimica et biophysica acta (01.12.2008)
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Journal Article
IMIDAZO[4,5-B]PYRIDINE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF INFLAMMATORY DISORDERS
COTI, Ghjuvanni, CLAES, Pieter, MARTINA, Sébastien, MAMMOLITI, Oscar, AMANTINI, David, LÓPEZ RAMOS, Miriam, ANNOOT, Denis, GALIEN, René, VAN DER PLAS, Steven, BRYS, Reginald
Year of Publication 12.01.2024
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Year of Publication 12.01.2024
Patent
IMIDAZO[4,5-B]PYRIDINE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF INFLAMMATORY DISORDERS
COTI, Ghjuvanni, CLAES, Pieter, MARTINA, Sébastien, MAMMOLITI, Oscar, AMANTINI, David, LÓPEZ RAMOS, Miriam, ANNOOT, Denis, GALIEN, René, VAN DER PLAS, Steven, BRYS, Reginald
Year of Publication 31.10.2023
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Year of Publication 31.10.2023
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IMIDAZO[4,5-B]PYRIDINE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF INFLAMMATORY DISORDERS
COTI, Ghjuvanni, CLAES, Pieter, MARTINA, Sébastien, MAMMOLITI, Oscar, AMANTINI, David, LÓPEZ RAMOS, Miriam, ANNOOT, Denis, GALIEN, René, VAN DER PLAS, Steven, BRYS, Reginald
Year of Publication 25.10.2023
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Year of Publication 25.10.2023
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IMIDAZO[4,5-B]PYRIDINE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF INFLAMMATORY DISORDERS
BRYS, Reginald, Christophe, Xavier, VAN DER PLAS, Steven, Emiel, MAMMOLITI, Oscar, AMANTINI, David, MARTINA, Sébastien, Laurent, Xavier, LÓPEZ RAMOS, Miriam, COTI, Ghjuvanni, Petru, Diunisu, ANNOOT, Denis, Maurice, GALIEN, René, Alexandre, CLAES, Pieter, Isabelle, Roger
Year of Publication 13.03.2024
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Year of Publication 13.03.2024
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IMIDAZO[4,5-B]PYRIDINE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF INFLAMMATORY DISORDERS
BRYS, REGINALD CHRISTOPHE XAVIER, MAMMOLITI, OSCAR, LÓPEZ RAMOS, MIRIAM, AMANTINI, DAVID, MARTINA, SÉBASTIEN LAURENT XAVIER, VAN DER PLAS, STEVEN EMIEL, COTI, GHJUVANNI PETRU DIUNISU, GALIEN, RENÉ ALEXANDRE, CLAES, PIETER ISABELLE ROGER, ANNOOT, DENIS MAURICE
Year of Publication 11.03.2024
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Year of Publication 11.03.2024
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IMIDAZO[4,5-B]PYRIDINE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF INFLAMMATORY DISORDERS
Martina, Sébastien Laurent Xavier, Mammoliti, Oscar, Amantini, David, Coti, Ghjuvanni Petru Diunisu, Van Der Plas, Steven Emiel, Claes, Pieter Isabelle Roger, Annoot, Denis Maurice, Brys, Reginald Christophe Xavier, López Ramos, Miriam, Galien, René Alexandre
Year of Publication 16.02.2024
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Year of Publication 16.02.2024
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IMIDAZO[4,5-B]PYRIDINFORBINDELSER OG FARMACEUTISKE SAMMENSÆTNINGER DERAF TIL BEHANDLING AF INFLAMMATORISKE FORSTYRRELSER
BRYS, Reginald, Christophe, Xavier, VAN DER PLAS, Steven, Emiel, MAMMOLITI, Oscar, AMANTINI, David, MARTINA, Sébastien, Laurent, Xavier, LÓPEZ RAMOS, Miriam, COTI, Ghjuvanni, Petru, Diunisu, ANNOOT, Denis, Maurice, GALIEN, René, Alexandre, CLAES, Pieter, Isabelle, Roger
Year of Publication 15.01.2024
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Year of Publication 15.01.2024
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IMIDAZO[4,5-B]PYRIDINE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF INFLAMMATORY DISORDERS
BRYS, Reginald, Christophe, Xavier, VAN DER PLAS, Steven, Emiel, MAMMOLITI, Oscar, AMANTINI, David, MARTINA, Sébastien, Laurent, Xavier, LÓPEZ RAMOS, Miriam, COTI, Ghjuvanni, Petru, Diunisu, ANNOOT, Denis, Maurice, GALIEN, René, Alexandre, CLAES, Pieter, Isabelle, Roger
Year of Publication 27.12.2023
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Year of Publication 27.12.2023
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IMIDAZO[4,5-B]PYRIDINE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF INFLAMMATORY DISORDERS
ANNOOT, DENIS, MAURICE, COTI, GHJUVANNI, PETRU, DIUNISU, MAMMOLITI, OSCAR, AMANTINI, DAVID, LÓPEZ, RAMOS, MIRIAM, BRYS, REGINALD, CHRISTOPHE, XAVIER, MARTINA, SÉBASTIEN, LAURENT, XAVIER, CLAES, PIETER, ISABELLE, ROGER, VAN DER PLAS, STEVEN, EMIEL, GALIEN, RENÉ, ALEXANDRE
Year of Publication 30.11.2023
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Year of Publication 30.11.2023
Patent