INCB054828 (pemigatinib), a potent and selective inhibitor of fibroblast growth factor receptors 1, 2, and 3, displays activity against genetically defined tumor models
Liu, Phillip C C, Koblish, Holly, Wu, Liangxing, Bowman, Kevin, Diamond, Sharon, DiMatteo, Darlise, Zhang, Yue, Hansbury, Michael, Rupar, Mark, Wen, Xiaoming, Collier, Paul, Feldman, Patricia, Klabe, Ronald, Burke, Krista A, Soloviev, Maxim, Gardiner, Christine, He, Xin, Volgina, Alla, Covington, Maryanne, Ruggeri, Bruce, Wynn, Richard, Burn, Timothy C, Scherle, Peggy, Yeleswaram, Swamy, Yao, Wenqing, Huber, Reid, Hollis, Gregory
Published in PloS one (21.04.2020)
Published in PloS one (21.04.2020)
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Discovery of Pemigatinib: A Potent and Selective Fibroblast Growth Factor Receptor (FGFR) Inhibitor
Wu, Liangxing, Zhang, Colin, He, Chunhong, Qian, Dingquan, Lu, Liang, Sun, Yaping, Xu, Meizhong, Zhuo, Jincong, Liu, Phillip C. C, Klabe, Ronald, Wynn, Richard, Covington, Maryanne, Gallagher, Karen, Leffet, Lynn, Bowman, Kevin, Diamond, Sharon, Koblish, Holly, Zhang, Yue, Soloviev, Maxim, Hollis, Gregory, Burn, Timothy C, Scherle, Peggy, Yeleswaram, Swamy, Huber, Reid, Yao, Wenqing
Published in Journal of medicinal chemistry (12.08.2021)
Published in Journal of medicinal chemistry (12.08.2021)
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Potent Benzimidazole Sulfonamide Protein Tyrosine Phosphatase 1B Inhibitors Containing the Heterocyclic (S)-Isothiazolidinone Phosphotyrosine Mimetic
Combs, Andrew P, Zhu, Wenyu, Crawley, Matthew L, Glass, Brian, Polam, Padmaja, Sparks, Richard B, Modi, Dilip, Takvorian, Amy, McLaughlin, Erin, Yue, Eddy W, Wasserman, Zelda, Bower, Michael, Wei, Min, Rupar, Mark, Ala, Paul J, Reid, Brian M, Ellis, Dawn, Gonneville, Lucie, Emm, Thomas, Taylor, Nancy, Yeleswaram, Swamy, Li, Yanlong, Wynn, Richard, Burn, Timothy C, Hollis, Gregory, Liu, Phillip C. C, Metcalf, Brian
Published in Journal of medicinal chemistry (29.06.2006)
Published in Journal of medicinal chemistry (29.06.2006)
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Benzothiazole benzimidazole ( S)-isothiazolidinone derivatives as protein tyrosine phosphatase-1B inhibitors
Sparks, Richard B., Polam, Padmaja, Zhu, Wenyu, Crawley, Matthew L., Takvorian, Amy, McLaughlin, Erin, Wei, Min, Ala, Paul J., Gonneville, Lucie, Taylor, Nancy, Li, Yanlong, Wynn, Richard, Burn, Timothy C., Liu, Phillip C.C., Combs, Andrew P.
Published in Bioorganic & medicinal chemistry letters (01.02.2007)
Published in Bioorganic & medicinal chemistry letters (01.02.2007)
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Isothiazolidinone inhibitors of PTP1B containing imidazoles and imidazolines
Douty, Brent, Wayland, Brian, Ala, Paul J., Bower, Michael J., Pruitt, James, Bostrom, Lori, Wei, Min, Klabe, Ronald, Gonneville, Lucie, Wynn, Richard, Burn, Timothy C., Liu, Phillip C.C., Combs, Andrew P., Yue, Eddy W.
Published in Bioorganic & medicinal chemistry letters (2008)
Published in Bioorganic & medicinal chemistry letters (2008)
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Isothiazolidinone heterocycles as inhibitors of protein tyrosine phosphatases: Synthesis and structure–activity relationships of a peptide scaffold
Yue, Eddy W., Wayland, Brian, Douty, Brent, Crawley, Matthew L., McLaughlin, Erin, Takvorian, Amy, Wasserman, Zelda, Bower, Michael J., Wei, Min, Li, Yanlong, Ala, Paul J., Gonneville, Lucie, Wynn, Richard, Burn, Timothy C., Liu, Phillip C.C., Combs, Andrew P.
Published in Bioorganic & medicinal chemistry (01.09.2006)
Published in Bioorganic & medicinal chemistry (01.09.2006)
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Characterization of INCB086550: A Potent and Novel Small-Molecule PD-L1 Inhibitor
Koblish, Holly K, Wu, Liangxing, Wang, Liang-Chuan S, Liu, Phillip C C, Wynn, Richard, Rios-Doria, Jonathan, Spitz, Susan, Liu, Hao, Volgina, Alla, Zolotarjova, Nina, Kapilashrami, Kanishk, Behshad, Elham, Covington, Maryanne, Yang, Yan-Ou, Li, Jingwei, Diamond, Sharon, Soloviev, Maxim, O'Hayer, Kevin, Rubin, Stephen, Kanellopoulou, Chrysi, Yang, Gengjie, Rupar, Mark, DiMatteo, Darlise, Lin, Luping, Stevens, Christina, Zhang, Yue, Thekkat, Pramod, Geschwindt, Ryan, Marando, Cindy, Yeleswaram, Swamy, Jackson, Jeff, Scherle, Peggy, Huber, Reid, Yao, Wenqing, Hollis, Gregory
Published in Cancer discovery (02.06.2022)
Published in Cancer discovery (02.06.2022)
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Targeting MYCN-expressing triple-negative breast cancer with BET and MEK inhibitors
Schafer, Johanna M, Lehmann, Brian D, Gonzalez-Ericsson, Paula I, Marshall, Clayton B, Beeler, J Scott, Redman, Lindsay N, Jin, Hailing, Sanchez, Violeta, Stubbs, Matthew C, Scherle, Peggy, Johnson, Kimberly N, Sheng, Quanhu, Roland, Joseph T, Bauer, Joshua A, Shyr, Yu, Chakravarthy, Bapsi, Mobley, Bret C, Hiebert, Scott W, Balko, Justin M, Sanders, Melinda E, Liu, Phillip C C, Pietenpol, Jennifer A
Published in Science translational medicine (11.03.2020)
Published in Science translational medicine (11.03.2020)
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Parsaclisib Is a Next-Generation Phosphoinositide 3-Kinase δ Inhibitor with Reduced Hepatotoxicity and Potent Antitumor and Immunomodulatory Activities in Models of B-Cell Malignancy
Shin, Niu, Stubbs, Matthew, Koblish, Holly, Yue, Eddy W., Soloviev, Maxim, Douty, Brent, Wang, Kathy He, Wang, Qian, Gao, Mingming, Feldman, Patricia, Yang, Gengjie, Hall, Leslie, Hansbury, Michael, O’Connor, Sybil, Leffet, Lynn, Collins, Robert, Katiyar, Kamna, He, Xin, Waeltz, Paul, Collier, Paul, Lu, Jin, Li, Yun-Long, Li, Yanlong, Liu, Phillip C.C., Burn, Timothy, Covington, Maryanne, Diamond, Sharon, Shuey, Dana, Roberts, Alan, Yeleswaram, Swamy, Hollis, Greg, Metcalf, Brian, Yao, Wenqing, Huber, Reid, Combs, Andrew, Newton, Robert, Scherle, Peggy
Published in The Journal of pharmacology and experimental therapeutics (01.07.2020)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2020)
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The Novel Bromodomain and Extraterminal Domain Inhibitor INCB054329 Induces Vulnerabilities in Myeloma Cells That Inform Rational Combination Strategies
Stubbs, Matthew C, Burn, Timothy C, Sparks, Richard, Maduskuie, Thomas, Diamond, Sharon, Rupar, Mark, Wen, Xiaoming, Volgina, Alla, Zolotarjova, Nina, Waeltz, Paul, Favata, Margaret, Jalluri, Ravi, Liu, Huiqing, Liu, Xuesong Mike, Li, Jun, Collins, Robert, Falahatpisheh, Nikoo, Polam, Padmaja, DiMatteo, Darlise, Feldman, Patricia, Dostalik, Valerie, Thekkat, Pramod, Gardiner, Christine, He, Xin, Li, Yanlong, Covington, Maryanne, Wynn, Richard, Ruggeri, Bruce, Yeleswaram, Swamy, Xue, Chu-Biao, Yao, Wenqing, Combs, Andrew P, Huber, Reid, Hollis, Gregory, Scherle, Peggy, Liu, Phillip C C
Published in Clinical cancer research (01.01.2019)
Published in Clinical cancer research (01.01.2019)
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Validation of standards for quantitative assessment of JAK2 c.1849G>T (p.V617F) allele burden analysis in clinical samples
Collier, Paul, Patel, Keyur, Waeltz, Paul, Rupar, Mark, Luthra, Rajyalakshmi, Liu, Phillip C C, Hollis, Gregory, Huber, Reid, Verstovsek, Srdan, Burn, Timothy C
Published in Genetic testing and molecular biomarkers (01.05.2013)
Published in Genetic testing and molecular biomarkers (01.05.2013)
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BET Inhibition Enhances the Antileukemic Activity of Low-dose Venetoclax in Acute Myeloid Leukemia
Ramsey, Haley E, Greenwood, Dalton, Zhang, Susu, Childress, Merrida, Arrate, Maria P, Gorska, Agnieszka E, Fuller, Londa, Zhao, Yue, Stengel, Kristy, Fischer, Melissa A, Stubbs, Matthew C, Liu, Phillip C C, Boyd, Kelli, Rathmell, Jeffrey C, Hiebert, Scott W, Savona, Michael R
Published in Clinical cancer research (15.01.2021)
Published in Clinical cancer research (15.01.2021)
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High-throughput determination of mode of inhibition in lead identification and optimization
Wei, Min, Wynn, Richard, Hollis, Gregory, Liao, Boshan, Margulis, Alexander, Reid, Brian G, Klabe, Ronald, Liu, Phillip C C, Becker-Pasha, Mary, Rupar, Mark, Burn, Timothy C, McCall, Dale E, Li, Yanlong
Published in Journal of biomolecular screening (01.03.2007)
Published in Journal of biomolecular screening (01.03.2007)
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Efficacy of Novel Bromodomain and Extraterminal Inhibitors in Combination with Chemotherapy for Castration-Resistant Prostate Cancer
Vázquez, Ramiro, Civenni, Gianluca, Kokanovic, Aleksandra, Shinde, Dheeraj, Cantergiani, Jasmine, Marchetti, Martina, Zoppi, Giada, Ruggeri, Bruce, Liu, Phillip C.C., Carbone, Giuseppina M., Catapano, Carlo V.
Published in European urology oncology (01.06.2021)
Published in European urology oncology (01.06.2021)
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Identification of ADAM10 as a major source of HER2 ectodomain sheddase activity in HER2 overexpressing breast cancer cells
Liu, Phillip C.C., Liu, Xiangdong, Li, Yanlong, Covington, Maryanne, Wynn, Richard, Huber, Reid, Hillman, Milton, Yang, Gengjie, Ellis, Dawn, Marando, Cindy, Katiyar, Kamna, Bradley, Jodi, Abremski, Kenneth, Stow, Mark, Rupar, Mark, Zhuo, Jincong, Li, Yun-Long, Lin, Qiyan, Burns, David, Xu, Meizhong, Zhang, Colin, Qian, Ding-Quan, He, Chunhong, Sharief, Vaqar, Weng, Lingkai, Agrios, Costas, Shi, Eric, Metcalf, Brian, Newton, Robert, Friedman, Steven, Yao, Wenqing, Scherle, Peggy A., Hollis, Gregory, Burn, Timothy C.
Published in Cancer biology & therapy (01.06.2006)
Published in Cancer biology & therapy (01.06.2006)
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Combined Inhibition of Janus Kinase 1/2 for the Treatment of JAK2V617F-Driven Neoplasms: Selective Effects on Mutant Cells and Improvements in Measures of Disease Severity
Liu, Phillip C C, Caulder, Eian, Li, Jun, Waeltz, Paul, Margulis, Alex, Wynn, Richard, Becker-Pasha, Mary, Li, Yanlong, Crowgey, Erin, Hollis, Gregory, Haley, Patrick, Sparks, Richard B, Combs, Andrew P, Rodgers, James D, Burn, Timothy C, Vaddi, Kris, Fridman, Jordan S
Published in Clinical cancer research (15.11.2009)
Published in Clinical cancer research (15.11.2009)
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Abstract 3780: Activity of the BET inhibitor INCB054329 in models of lymphoma
Stubbs, Matthew, Collins, Robert, Volgina, Alla, Liu, Mike, Favata, Margaret, Rupar, Mark, Wen, Xiaomng, Sparks, Richard, Maduskuie, Thomas, Covington, Maryanne, Burn, Timothy, Ruggeri, Bruce, Combs, Andrew P., Yao, Wenqing, Huber, Reid, Hollis, Gregory, Scherle, Peggy, Liu, Phillip CC
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Induction of endogenous genes by peroxisome proliferator activated receptor alpha ligands in a human kidney cell line and in vivo
Liu, Phillip C.C., Huber, Reid, Stow, Mark D., Schlingmann, Karen L., Collier, Paul, Liao, Boshan, Link, John, Burn, Tim C., Hollis, Greg, Young, Peter R., Mukherjee, Ranjan
Published in The Journal of steroid biochemistry and molecular biology (01.05.2003)
Published in The Journal of steroid biochemistry and molecular biology (01.05.2003)
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