Synthetic Approaches to the New Drugs Approved During 2015
Flick, Andrew C, Ding, Hong X, Leverett, Carolyn A, Kyne, Robert E, Liu, Kevin K. -C, Fink, Sarah J, O’Donnell, Christopher J
Published in Journal of medicinal chemistry (10.08.2017)
Published in Journal of medicinal chemistry (10.08.2017)
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Discovery of 1‑{(3R,4R)‑3-[({5-Chloro-2-[(1-methyl‑1H‑pyrazol-4-yl)amino]‑7H‑pyrrolo[2,3‑d]pyrimidin-4-yl}oxy)methyl]-4-methoxypyrrolidin-1-yl}prop-2-en-1-one (PF-06459988), a Potent, WT Sparing, Irreversible Inhibitor of T790M-Containing EGFR Mutants
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Published in Journal of medicinal chemistry (10.03.2016)
Published in Journal of medicinal chemistry (10.03.2016)
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Synthetic approaches to the 2011 new drugs
Ding, Hong X., Liu, Kevin K.-C., Sakya, Subas M., Flick, Andrew C., O’Donnell, Christopher J.
Published in Bioorganic & medicinal chemistry (01.06.2013)
Published in Bioorganic & medicinal chemistry (01.06.2013)
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Esophageal tuberculosis induced dysphagia: a case report
Olson, Dylan, Liu, Kevin C, Merza, Anthony P, Tilahun, Ermias, Aziz Aadam, A
Published in BMC gastroenterology (22.03.2022)
Published in BMC gastroenterology (22.03.2022)
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Identification of Cys255 in HIF‐1α as a novel site for development of covalent inhibitors of HIF‐1α/ARNT PasB domain protein–protein interaction
Cardoso, Rosa, Love, Robert, Nilsson, Carol L., Bergqvist, Simon, Nowlin, Dawn, Yan, Jiangli, Liu, Kevin K.‐C., Zhu, Jing, Chen, Ping, Deng, Ya‐Li, Dyson, H. Jane, Greig, Michael J., Brooun, Alexei
Published in Protein science (01.12.2012)
Published in Protein science (01.12.2012)
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Medicare Advantage in Soft Tissue Sarcoma May Be Associated with Worse Patient Outcomes
Wang, Jennifer C, Liu, Kevin C, Gettleman, Brandon S, Piple, Amit S, Chen, Matthew S, Menendez, Lawrence R, Heckmann, Nathanael D, Christ, Alexander B
Published in Journal of clinical medicine (01.08.2023)
Published in Journal of clinical medicine (01.08.2023)
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Risk Factors for Peripheral Nerve Injury Following Revision Total Hip Arthroplasty in 112,310 Patients
Chen, Xiao T, Korber, Shane S, Liu, Kevin C, Gettleman, Brandon S, Shahrestani, Shane, Heckmann, Nathanael D, Christ, Alexander B
Published in Journal of clinical medicine (01.03.2024)
Published in Journal of clinical medicine (01.03.2024)
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Synthetic approaches to the 2010 new drugs
Liu, Kevin K.-C., Sakya, Subas M., O’Donnell, Christopher J., Flick, Andrew C., Ding, Hong X.
Published in Bioorganic & medicinal chemistry (01.02.2012)
Published in Bioorganic & medicinal chemistry (01.02.2012)
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Synthetic approaches to the 2009 new drugs
Liu, Kevin K.-C., Sakya, Subas M., O’Donnell, Christopher J., Flick, Andrew C., Li, Jin
Published in Bioorganic & medicinal chemistry (01.02.2011)
Published in Bioorganic & medicinal chemistry (01.02.2011)
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Conformationally-restricted cyclic sulfones as potent and selective mTOR kinase inhibitors
Liu, Kevin K.-C., Bailey, Simon, Dinh, Dac M., Lam, Hieu, Li, Chunze, Wells, Peter A., Yin, Min-Jean, Zou, Aihua
Published in Bioorganic & medicinal chemistry letters (01.08.2012)
Published in Bioorganic & medicinal chemistry letters (01.08.2012)
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Characteristics of Very Young Patients Undergoing Total Hip Arthroplasty: A Contemporary Assessment
Wang, Jennifer C., Liu, Kevin C., Gettleman, Brandon S., Chen, Matthew, Piple, Amit S., Yang, Jaewon, Heckmann, Nathanael D., Christ, Alexander B.
Published in Arthroplasty today (01.02.2024)
Published in Arthroplasty today (01.02.2024)
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An Updated Estimate of Total Hip and Total Knee Arthroplasty Inpatient Case Volume During the 2020 COVID-19 Pandemic in the United States
Heckmann, Nathanael D., Mayfield, Cory K., Richardson, Mary K., Liu, Kevin C., Wang, Jennifer C., Piple, Amit S., Stambough, Jeffrey B., Oakes, Daniel A., Christ, Alexander B., Lieberman, Jay R.
Published in Arthroplasty today (01.04.2024)
Published in Arthroplasty today (01.04.2024)
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Discovery of the Highly Potent PI3K/mTOR Dual Inhibitor PF-04979064 through Structure-Based Drug Design
Cheng, Hengmiao, Li, Chunze, Bailey, Simon, Baxi, Sangita M, Goulet, Lance, Guo, Lisa, Hoffman, Jacqui, Jiang, Ying, Johnson, Theodore Otto, Johnson, Ted W, Knighton, Daniel R, Li, John, Liu, Kevin K.-C, Liu, Zhengyu, Marx, Matthew A, Walls, Marlena, Wells, Peter A, Yin, Min-Jean, Zhu, Jinjiang, Zientek, Michael
Published in ACS medicinal chemistry letters (10.01.2013)
Published in ACS medicinal chemistry letters (10.01.2013)
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Synthetic approaches to the 2014 new drugs
Flick, Andrew C., Ding, Hong X., Leverett, Carolyn A., Kyne, Robert E., Liu, Kevin K.-C., Fink, Sarah J., O’Donnell, Christopher J.
Published in Bioorganic & medicinal chemistry (01.05.2016)
Published in Bioorganic & medicinal chemistry (01.05.2016)
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Synthetic approaches to the 2008 new drugs
Liu, Kevin K-C, Sakya, Subas M, O'Donnell, Christopher J, Li, Jin
Published in Mini reviews in medicinal chemistry (01.12.2009)
Published in Mini reviews in medicinal chemistry (01.12.2009)
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Quinazolines with intra-molecular hydrogen bonding scaffold (iMHBS) as PI3K/mTOR dual inhibitors
Liu, Kevin K.C., Huang, Xiaojun, Bagrodia, Shubha, Chen, Jeffrey H., Greasley, Samantha, Cheng, Hengmiao, Sun, Shaoxian, Knighton, Dan, Rodgers, Caroline, Rafidi, Kristina, Zou, Aihua, Xiao, Jiezhan, Yan, Shengyong
Published in Bioorganic & medicinal chemistry letters (15.02.2011)
Published in Bioorganic & medicinal chemistry letters (15.02.2011)
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Journal Article
Synthetic approaches to the 2013 new drugs
Ding, Hong X., Leverett, Carolyn A., Kyne, Robert E., Liu, Kevin K.-C., Fink, Sarah J., Flick, Andrew C., O’Donnell, Christopher J.
Published in Bioorganic & medicinal chemistry (01.05.2015)
Published in Bioorganic & medicinal chemistry (01.05.2015)
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4-Methylpteridinones as orally active and selective PI3K/mTOR dual inhibitors
Liu, Kevin K.-C., Bagrodia, Shubha, Bailey, Simon, Cheng, Hengmiao, Chen, Hui, Gao, Lisa, Greasley, Samantha, Hoffman, Jacqui E., Hu, Qiyue, Johnson, Ted O., Knighton, Dan, Liu, Zhengyu, Marx, Matthew A., Nambu, Mitchell D., Ninkovic, Sacha, Pascual, Bernadette, Rafidi, Kristina, Rodgers, Caroline M.-L., Smith, Graham L., Sun, Shaoxian, Wang, Haitao, Yang, Anle, Yuan, Jing, Zou, Aihua
Published in Bioorganic & medicinal chemistry letters (15.10.2010)
Published in Bioorganic & medicinal chemistry letters (15.10.2010)
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Design and synthesis of orally-active and selective azaindane 5HT2c agonist for the treatment of obesity
Liu, Kevin K.-C., Cornelius, Peter, Patterson, Terrell A., Zeng, Yuan, Santucci, Stephanie, Tomlinson, Elizabeth, Gibbons, Colleen, Maurer, Tristan S., Marala, Ravi, Brown, Janice, Kong, Jimmy X., Lee, Eunsun, Werner, Wendy, Wenzel, Zane, Vage, Chandra
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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