Potency Comparison of Peptidomimetic Inhibitors against HIV-1 and HIV-2 Proteinases: Design of Equipotent Lead Compounds
Weber, Jan, Majer, Pavel, Litera, Jaroslav, Urban, Jan, Souček, Milan, Vondrášek, Jiřı́, Konvalinka, Jan, Novek, Petr, Sedláček, Juraj, Štrop, Petr, Kräusslich, Hans-Georg, Pichová, Iva
Published in Archives of biochemistry and biophysics (01.05.1997)
Published in Archives of biochemistry and biophysics (01.05.1997)
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Peptide inhibitors of aspartic proteinases with hydroxyethylene isostere replacement of peptide bond. I. Preparation of four diastereoisomeric (2R or 2S,4R or 4S,5S)-2-benzyl-5-[(tert-butoxycarbonyl)amino]-4-hydroxy-6-phenylhexanoic acids
Litera, J, Budesinsky, M, Urban, J, Soucek, M
Published in Collection of Czechoslovak chemical communications (1998)
Published in Collection of Czechoslovak chemical communications (1998)
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Configurations of Diastereomeric Hydroxyethylene Isosteres Strongly Affect Biological Activities of a Series of Specific Inhibitors of Human‐Immunodeficiency‐Virus Proteinase
Konvalinka, Jan, Litera, Jaroslav, Weber, Jan, Vondrášek, Jiří, Hradílek, Martin, Souček, Milan, Pichová, Iva, Majer, Pavel, Štrop, Petr, Sedlácek, Juraj, Heuser, Anke‐Mareil, Kottler, Hubert, Kräusslich, Hans‐Georg
Published in European journal of biochemistry (01.12.1997)
Published in European journal of biochemistry (01.12.1997)
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Peptide inhibitors of aspartic proteinases with hydroxyethylene isostere replacement of peptide bond. II. Preparation of pseudotetrapeptides derived from diastereoisomeric 5-amino-2-benzyl-4-hydroxy-6-phenylhexanoic acids
Litera, J, Weber, J, Krizova, Pichova, Konvalinka, J, Fusek, M, Soucek, M
Published in Collection of Czechoslovak chemical communications (1998)
Published in Collection of Czechoslovak chemical communications (1998)
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