Broad-Spectrum Antimalarial Activity of Peptido Sulfonyl Fluorides, a New Class of Proteasome Inhibitors
TSCHAN, Serena, BROUWER, Arwin J, MORDMÜLLER, Benjamin, WERKHOVEN, Paul R, JONKER, Anika M, WAGNER, Lena, KNITTEL, Sarah, AMINAKE, Makoah Nigel, PRADEL, Gabriele, JOANNY, Fanny, LISKAMP, Rob M. J
Published in Antimicrobial Agents and Chemotherapy (01.08.2013)
Published in Antimicrobial Agents and Chemotherapy (01.08.2013)
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Polar Hinges as Functionalized Conformational Constraints in (Bi)cyclic Peptides
van de Langemheen, Helmus, Korotkovs, Valerijs, Bijl, Joachim, Wilson, Claire, Kale, Sangram S., Heinis, Christian, Liskamp, Rob M. J.
Published in Chembiochem : a European journal of chemical biology (16.02.2017)
Published in Chembiochem : a European journal of chemical biology (16.02.2017)
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The Vancomycin−Nisin(1−12) Hybrid Restores Activity against Vancomycin Resistant Enterococci
Arnusch, Christopher J, Bonvin, Alexandre M. J. J, Verel, Anne Marie, Jansen, Wouter T. M, Liskamp, Rob M. J, de Kruijff, Ben, Pieters, Roland J, Breukink, Eefjan
Published in Biochemistry (Easton) (02.12.2008)
Published in Biochemistry (Easton) (02.12.2008)
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Potent and Highly Selective Inhibitors of the Proteasome Trypsin-like Site by Incorporation of Basic Side Chain Containing Amino Acid Derived Sulfonyl Fluorides
Artschwager, Raik, Ward, David J, Gannon, Susan, Brouwer, Arwin J, van de Langemheen, Helmus, Kowalski, Hubert, Liskamp, Rob M. J
Published in Journal of medicinal chemistry (28.06.2018)
Published in Journal of medicinal chemistry (28.06.2018)
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Synthesis and biological evaluation of novel irreversible serine protease inhibitors using amino acid based sulfonyl fluorides as an electrophilic trap
Brouwer, Arwin J., Ceylan, Tarik, Jonker, Anika M., Linden, Tima van der, Liskamp, Rob M.J.
Published in Bioorganic & medicinal chemistry (01.04.2011)
Published in Bioorganic & medicinal chemistry (01.04.2011)
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Synthesis, Antimicrobial Activity, and Membrane Permeabilizing Properties of C‑Terminally Modified Nisin Conjugates Accessed by CuAAC
Slootweg, Jack C, van der Wal, Steffen, Quarles van Ufford, H. C, Breukink, Eefjan, Liskamp, Rob M. J, Rijkers, Dirk T. S
Published in Bioconjugate chemistry (18.12.2013)
Published in Bioconjugate chemistry (18.12.2013)
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Targeted Covalent Inhibition of Prolyl Oligopeptidase (POP): Discovery of Sulfonylfluoride Peptidomimetics
Guardiola, Salvador, Prades, Roger, Mendieta, Laura, Brouwer, Arwin J., Streefkerk, Jelle, Nevola, Laura, Tarragó, Teresa, Liskamp, Rob M.J., Giralt, Ernest
Published in Cell chemical biology (16.08.2018)
Published in Cell chemical biology (16.08.2018)
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A proteinaceous fraction of wheat bran may interfere in the attachment of enterotoxigenic E. coli K88 (F4+) to porcine epithelial cells
González-Ortiz, Gemma, Bronsoms, Sílvia, Quarles Van Ufford, H C, Halkes, S Bart A, Virkola, Ritva, Liskamp, Rob M J, Beukelman, Cees J, Pieters, Roland J, Pérez, José Francisco, Martín-Orúe, Susana María
Published in PloS one (13.08.2014)
Published in PloS one (13.08.2014)
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New properties of wheat bran: anti‐biofilm activity and interference with bacteria quorum‐sensing systems
González‐Ortiz, Gemma, Quarles Van Ufford, H. C, Halkes, S. Bart A, Cerd ‐Cuéllar, Marta, Beukelman, Cees J, Pieters, Roland J, Liskamp, Rob M. J, Pérez, José F, Martín‐Orue, Susana M
Published in Environmental microbiology (01.05.2014)
Published in Environmental microbiology (01.05.2014)
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Specific N-terminal attachment of TMTHSI linkers to native peptides and proteins for strain-promoted azide alkyne cycloaddition
Timmers, Matt, Peeters, Wouter, Hauwert, Niels J, Rijcken, Cristianne J. F, Vermonden, Tina, Dijkgraaf, Ingrid, Liskamp, Rob M. J
Published in Chemical communications (Cambridge, England) (21.09.2023)
Published in Chemical communications (Cambridge, England) (21.09.2023)
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TMTHSI, a superior 7-membered ring alkyne containing reagent for strain-promoted azide-alkyne cycloaddition reactions
Weterings, Jimmy, Rijcken, Cristianne J. F, Veldhuis, Harald, Meulemans, Tommi, Hadavi, Darya, Timmers, Matt, Honing, Maarten, Ippel, Hans, Liskamp, Rob M. J
Published in Chemical science (Cambridge) (07.09.2020)
Published in Chemical science (Cambridge) (07.09.2020)
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Versatile convergent synthesis of a three peptide loop containing protein mimic of whooping cough pertactin by successive Cu(I)-catalyzed azide alkyne cycloaddition on an orthogonal alkyne functionalized TAC-scaffold
Werkhoven, Paul R., van de Langemheen, Helmus, van der Wal, Steffen, Kruijtzer, John A. W., Liskamp, Rob M. J.
Published in Journal of peptide science (01.04.2014)
Published in Journal of peptide science (01.04.2014)
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Journal Article
Inhibition of Streptococcus suis Adhesion by Dendritic Galabiose Compounds at Low Nanomolar Concentration
JOOSTEN, John A. F., LOIMARANTA, Vuokko, APPELDOORN, Chantal C. M., HAATAJA, Sauli, EL MAATE, Fatna Ait, LISKAMP, Rob M. J., FINNE, Jukka, PIETERS, Roland J.
Published in Journal of medicinal chemistry (16.12.2004)
Published in Journal of medicinal chemistry (16.12.2004)
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Molecular Construction of Sulfonamide Antisense Oligonucleotides
Korotkovs, Valerijs, Reichenbach, Linus F, Pescheteau, Clémentine, Burley, Glenn A, Liskamp, Rob M. J
Published in Journal of organic chemistry (06.09.2019)
Published in Journal of organic chemistry (06.09.2019)
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