Pharmacology of L-754,142, a highly potent, orally active, nonpeptidyl endothelin antagonist
D L Williams, Jr, K L Murphy, N A Nolan, J A O'Brien, D J Pettibone, S D Kivlighn, S M Krause, E V Lis, Jr, G J Zingaro, R A Gabel
Published in The Journal of pharmacology and experimental therapeutics (01.12.1995)
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Published in The Journal of pharmacology and experimental therapeutics (01.12.1995)
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A peripherally acting alpha-2 adrenoceptor antagonist: L-659,066
CLINESCHMIDT, B. V, PETTIBONE, D. J, LOTTI, V. J, HUCKER, H. B, SWEENEY, B. M, REISS, D. R, LIS, E. V, HUFF, J. R, VACCA, J
Published in The Journal of pharmacology and experimental therapeutics (01.04.1988)
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Published in The Journal of pharmacology and experimental therapeutics (01.04.1988)
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Identification of an orally active, nonpeptidyl oxytocin antagonist
PETTIBONE, D. J, CLINESCHMIDT, B. V, HALUSKA, G. J, NOVY, M. J, LOWENSOHN, R. I, KISHEL, M. T, LIS, E. V, REISS, D. R, WOYDEN, C. J, EVANS, B. E, FREIDINGER, R. M, VEBER, D. F, COOK, M. J
Published in The Journal of pharmacology and experimental therapeutics (01.01.1993)
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Published in The Journal of pharmacology and experimental therapeutics (01.01.1993)
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Nonpeptide oxytocin antagonists: Analogs of L-371,257 with improved potency
Williams, Peter D., Bock, Mark G., Evans, Ben E., Freidinger, Roger M., Gallicchio, Steven N., Guidotti, Maribeth T., Jacobson, Marlene A., Kuo, Michelle S., Levy, Michelle R., Lis, Edward V., Michelson, Stuart R., Pawluczyk, Joseph M., Perlow, Debra S., Pettibone, Douglas J., Quigley, Amy G., Reiss, Duane R., Salvatore, Christopher, Stauffer, Kenneth J., Woyden, Carla J.
Published in Bioorganic & medicinal chemistry letters (03.05.1999)
Published in Bioorganic & medicinal chemistry letters (03.05.1999)
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Nonpeptide oxytocin antagonists: Potent, orally bioavailable analogs of L-371,257 containing A 1- R-(pyridyl)ethyl ether terminus
Kuo, Michelle S., Bock, Mark G., Freidinger, Roger M., Guidotti, Maribeth T., Lis, Edward V., Pawluczyk, Joseph M., Perlow, Debra S., Pettibone, Douglas J., Quigley, Amy G., Reiss, Duane R., Williams, Peter D., Woyden, Carla J.
Published in Bioorganic & medicinal chemistry letters (03.11.1998)
Published in Bioorganic & medicinal chemistry letters (03.11.1998)
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Journal Article
In vitro pharmacological profile of a novel structural class of oxytocin antagonists
PETTIBONE, D. J, CLINESCHMIDT, B. V, WILLIAMS, P. D, LOWENSOHN, R. I, LIS, E. V, REISS, D. R, TOTARO, J. A, WOYDEN, C. J, BOCK, M. G, FREIDINGER, R. M, TUNG, R. D, VEBER, D. F
Published in The Journal of pharmacology and experimental therapeutics (01.01.1991)
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Published in The Journal of pharmacology and experimental therapeutics (01.01.1991)
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Antagonism of oxytocin in rats and pregnant rhesus monkeys by the novel cyclic hexapeptides, L-366,682 and L-366,948
CLINESCHMIDT, B. V, PETTIBONE, D. J, FREIDINGER, R. M, VEBER, D. F, WILLIAMS, P. D, REISS, D. R, LIS, E. V, HALUSKA, G. J, NOVY, M. J, COOK, M. J, CUKIERSKI, M. A, KAUFMAN, M. J, BOCK, M. G
Published in The Journal of pharmacology and experimental therapeutics (01.03.1991)
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Published in The Journal of pharmacology and experimental therapeutics (01.03.1991)
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Pharmacology of L-744,453, a novel nonpeptidyl endothelin antagonist
Williams, David L, Murphy, Kathryn L, Nolan, Nancy A, O'Brien, Julie A, Lis, Edward V, Pettibone, Douglas J, Clineschmidt, Bradley V, Krause, Stephen M, Veber, Daniel F, Naylor, Elizabeth M, Chakravarty, Prasun K, Walsh, Thomas F, Dhanoa, Dale M, Chent, Anna, Bagley, Scott W, Fitch, Kenneth J, Greenlee, William J
Published in Life sciences (1973) (01.03.1996)
Published in Life sciences (1973) (01.03.1996)
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Journal Article
Bradykinin agonist activity of a novel, potent oxytocin antagonist
Pettibone, D J, Clineschmidt, B V, Lis, E V, Ransom, R W, Totaro, J A, Young, G S, Bock, M G, Freidinger, R M, Veber, D F, Williams, P D
Published in European journal of pharmacology (24.04.1991)
Published in European journal of pharmacology (24.04.1991)
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Journal Article
Development of Orally Active Oxytocin Antagonists: Studies on 1-(1-{4-[1-(2-Methyl-1-oxidopyridin-3-ylmethyl)piperidin-4-yloxy]-2- methoxybenzoyl}piperidin-4-yl)-1,4-dihydrobenz[d][1,3]oxazin-2-one (L-372,662) and Related Pyridines
Bell, Ian M, Erb, Jill M, Freidinger, Roger M, Gallicchio, Steven N, Guare, James P, Guidotti, Maribeth T, Halpin, Rita A, Hobbs, Doug W, Homnick, Carl F, Kuo, Michelle S, Lis, Edward V, Mathre, David J, Michelson, Stuart R, Pawluczyk, Joseph M, Pettibone, Douglas J, Reiss, Duane R, Vickers, Stanley, Williams, Peter D, Woyden, Carla J
Published in Journal of medicinal chemistry (04.06.1998)
Published in Journal of medicinal chemistry (04.06.1998)
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The Effects of Deleting the Mouse Neurotensin Receptor NTR1 on Central and Peripheral Responses to Neurotensin
Pettibone, Douglas J, Hess, J Fred, Hey, Patricia J, Jacobson, Marlene A, Leviten, Michael, Lis, Edward V, Mallorga, Pierre J, Pascarella, Danette M, Snyder, Melissa A, Williams, Jacinta B, Zeng, Zhizhen
Published in The Journal of pharmacology and experimental therapeutics (01.01.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.01.2002)
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Journal Article
1-{1-[4-[(N-acetyl-4-piperidinyl)oxy]-2-methoxybenzoyl]piperidin-4-yl}-4H-3,1-benzoxazin-2(1H)-one (L-371,257) : a new, orally bioavailable, non-peptide oxytocin antagonist
WILLIAMS, P. D, CLINESCHMIDT, B. V, WOYDEN, C. J, ERB, J. M, FREIDINGER, R. M, GUIDOTTI, M. T, LIS, E. V, PAWLUCZYK, J. M, PETTIBONE, D. J, REISS, D. R, VEBER, D. F
Published in Journal of medicinal chemistry (01.11.1995)
Published in Journal of medicinal chemistry (01.11.1995)
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Journal Article
Benzodiazepines as potent and selective bradykinin B-1 antagonists
Wood, MR, Kim, JJ, Han, W, Dorsey, BD, Homnick, CF, DiPardo, RM, Kuduk, SD, MacNeil, T, Murphy, KL, Lis, EV, Ransom, RW, Stump, GL, Lynch, JJ, O'Malley, SS, Miller, PJ, Chen, TB, Harrell, CM, Chang, RSL, Sandhu, P, Ellis, JD, Bondiskey, PJ, Pettibone, DJ, Freidinger, RM, Bock, MG
Published in Journal of medicinal chemistry (08.05.2003)
Published in Journal of medicinal chemistry (08.05.2003)
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Development of orally active oxytocin antagonists : Studies on 1-(1-{4-[1-(2-methyl-1-oxidopyridin-3-ylmethyl)piperidin-4-yloxy]-2-methoxybenzo yl}piperidin-4-yl)-1,4-dihydrobenz[d][1,3]oxazin-2-one (L-372,662) and related pyridines
BELL, I. M, ERB, J. M, LIS, E. V, MATHRE, D. J, MICHELSON, S. R, PAWLUCZYK, J. M, PETTIBONE, D. J, REISS, D. R, VICKERS, S, WILLIAMS, P. D, WOYDEN, C. J, FREIDINGER, R. M, GALLICCHIO, S. N, GUARE, J. P, GUIDOTTI, M. T, HALPIN, R. A, HOBBS, D. W, HOMNICK, C. F, KUO, M. S
Published in Journal of medicinal chemistry (1998)
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Published in Journal of medicinal chemistry (1998)
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1-(1-[4-[(N-acetyl-4-piperidinyl)oxy]-2-methoxybenzoyl]piperidin-4- yl)-4H-3,1-benzoxazin-2(1H)-one (L-371,257): a new, orally bioavailable, non-peptide oxytocin antagonist
Williams, P D, Clineschmidt, B V, Erb, J M, Freidinger, R M, Guidotti, M T, Lis, E V, Pawluczyk, J M, Pettibone, D J, Reiss, D R, Veber, D F
Published in Journal of medicinal chemistry (10.11.1995)
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Published in Journal of medicinal chemistry (10.11.1995)
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Benzodiazepines as Potent and Selective Bradykinin B1 Antagonists
Wood, Michael R, Kim, June J, Han, Wei, Dorsey, Bruce D, Homnick, Carl F, DiPardo, Robert M, Kuduk, Scott D, MacNeil, Tanya, Murphy, Kathy L, Lis, Edward V, Ransom, Richard W, Stump, Gary L, Lynch, Joseph J, O'Malley, Stacey S, Miller, Patricia J, Chen, Tsing-Bau, Harrell, Charles M, Chang, Raymond S. L, Sandhu, Punam, Ellis, Joan D, Bondiskey, Peter J, Pettibone, Douglas J, Freidinger, Roger M, Bock, Mark G
Published in Journal of medicinal chemistry (08.05.2003)
Published in Journal of medicinal chemistry (08.05.2003)
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