Novel, Achiral 1,3,4-Benzotriazepine Analogues of 1,4-Benzodiazepine-Based CCK2 Antagonists That Display High Selectivity over CCK1 Receptors
McDonald, Iain M, Austin, Carol, Buck, Ildiko M, Dunstone, David J, Griffin, Eric, Harper, Elaine A, Hull, Robert A. D, Kalindjian, S. Barret, Linney, Ian D, Low, Caroline M. R, Pether, Michael J, Spencer, John, Wright, Paul T, Adatia, Trushar, Bashall, Alan
Published in Journal of medicinal chemistry (06.04.2006)
Published in Journal of medicinal chemistry (06.04.2006)
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Optimization of the in Vitro and in Vivo Properties of a Novel Series of 2,4,5-Trisubstituted Imidazoles as Potent Cholecystokinin-2 (CCK2) Antagonists
Buck, Ildiko M, Black, James W, Cooke, Tracey, Dunstone, David J, Gaffen, John D, Griffin, Eric P, Harper, Elaine A, Hull, Robert A. D, Kalindjian, S. Barret, Lilley, Elliot J, Linney, Ian D, Low, Caroline M. R, McDonald, Iain M, Pether, Michael J, Roberts, Sonia P, Shankley, Nigel P, Shaxted, Mark E, Steel, Katherine I. M, Sykes, David A, Tozer, Matthew J, Watt, Gillian F, Walker, Martin K, Wright, Laurence, Wright, Paul T
Published in Journal of medicinal chemistry (03.11.2005)
Published in Journal of medicinal chemistry (03.11.2005)
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2,7-Dioxo-2,3,4,5,6,7-hexahydro-1H-benzo[h][1,4]diazonine as a New Template for the Design of CCK2 Receptor Antagonists
McDonald, Iain M, Dunstone, David J, Kalindjian, S. Barret, Linney, Ian D, Low, Caroline M. R, Pether, Michael J, Steel, Katherine I. M, Tozer, Matthew J, Vinter, J. G
Published in Journal of medicinal chemistry (21.09.2000)
Published in Journal of medicinal chemistry (21.09.2000)
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Synthesis of Enantiopure Dihydropyranones: Aldol-Based Ring Expansion of Dihydrofurans
Donohoe, Timothy J, Raoof, Ali, Freestone, Graeme C, Linney, Ian D, Cowley, Andrew, Helliwell, Madeleine
Published in Organic letters (05.09.2002)
Published in Organic letters (05.09.2002)
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Recoverable chiral sulfoxides for asymmetric synthesis: Application to stereoselective carbonyl reduction and the asymmetric synthesis of allylic alcohols
Butlin, RJ, Linney, ID, Mahon, MF, Tye, H, Wills, M
Published in Journal of the Chemical Society, Perkin Transactions 1 (07.01.1996)
Published in Journal of the Chemical Society, Perkin Transactions 1 (07.01.1996)
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Recoverable chiral sulfoxides for asymmetric synthesis : preparation, regeneration and application to the asymmetric aldol reaction
BUTLIN, R. J, LINNEY, I. D, CRITCHER, D. J, MAHON, M. F, MOLLOY, K. C, WILLS, M
Published in Journal of the Chemical Society, Perkin Transactions 1 (1993)
Published in Journal of the Chemical Society, Perkin Transactions 1 (1993)
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DEPENDENCE OF RING-CLOSURE STEREOSELECTIVITY ON THE NATURE OF THE LEAVING GROUP - APPLICATION TO THE SYNTHESIS OF A NEW CLASS OF CHIRAL SULFOXIDE FOR THE CONTROL OF ASYMMETRIC ALDOL REACTIONS
WILLS, M, BUTLIN, RJ, LINNEY, ID, GIBSON, RW
Published in Journal of the Chemical Society, Perkin Transactions 1 (1991)
Published in Journal of the Chemical Society, Perkin Transactions 1 (1991)
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THE TOTAL SYNTHESIS OF EPIBATIDINE
KO, SY, LERPINIERE, J, LINNEY, ID, WRIGGLESWORTH, R
Published in Journal of the Chemical Society. Chemical communications (1994)
Published in Journal of the Chemical Society. Chemical communications (1994)
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