Efficacy in diet-induced obese mice of the hepatotropic, peripheral cannabinoid 1 receptor inverse agonist TM38837
Cooper, Martin E, Nørregaard, Pia K, Högberg, Thomas, Andersson, Gunnar, Receveur, Jean-Marie, Linget, Jean-Michel, Elling, Christian E
Published in British journal of pharmacology (01.10.2024)
Published in British journal of pharmacology (01.10.2024)
Get more information
Journal Article
Optimizing and characterizing 4-methyl substituted pyrazol-3-carboxamides leading to the peripheral cannabinoid 1 receptor inverse agonist TM38837
Högberg, Thomas, Receveur, Jean-Marie, Murray, Anthony, Linget, Jean-Michel, Nørregaard, Pia K., Little, Paul B., Cooper, Martin
Published in Bioorganic & medicinal chemistry letters (15.01.2024)
Published in Bioorganic & medicinal chemistry letters (15.01.2024)
Get full text
Journal Article
Application of the Tissue Composition–Based Model to Minipig for Predicting the Volume of Distribution at Steady State and Dermis-to-Plasma Partition Coefficients of Drugs Used in the Physiologically Based Pharmacokinetics Model in Dermatology
Poulin, Patrick, Collet, Severine H., Atrux-Tallau, Nicolas, Linget, Jean-Michel, Hennequin, Laurent, Wilson, Claire E.
Published in Journal of pharmaceutical sciences (01.01.2019)
Published in Journal of pharmaceutical sciences (01.01.2019)
Get full text
Journal Article
Pretreatment of skin using an abrasive skin preparation pad, a microneedling device or iontophoresis improves absorption of methyl aminolevulinate in ex vivo human skin
Osman-Ponchet, Hanan, Gaborit, Alexandre, Sevin, Karine, Bianchi, Christophe, Linget, Jean-Michel, Wilson, Claire E., Bouvier, Guy
Published in Photodiagnosis and photodynamic therapy (01.12.2017)
Published in Photodiagnosis and photodynamic therapy (01.12.2017)
Get full text
Journal Article
Conversion of 4-cyanomethyl-pyrazole-3-carboxamides into CB1 antagonists with lowered propensity to pass the blood–brain-barrier
Receveur, Jean-Marie, Murray, Anthony, Linget, Jean-Michel, Nørregaard, Pia K., Cooper, Martin, Bjurling, Emelie, Nielsen, Peter Aadal, Högberg, Thomas
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
Get full text
Journal Article
Comparison of the Effect of Skin Preparation Pads on Transepidermal Water Loss in Ex Vivo Human Skin
Osman-Ponchet, Hanan, Gaborit, Alexandre, Kouidhi, Magali, Anglars, Sandrine, Marceau-Suissa, Jeanne, Duffy-Roger, Orla, Linget, Jean-Michel, Wilson, Claire E.
Published in Dermatology and therapy (01.09.2017)
Published in Dermatology and therapy (01.09.2017)
Get full text
Journal Article
PHENOL DERIVATIVES AND PHARMACEUTICAL OR COSMETIC USE THEREOF
RETHORE SANDRINE, COLLETTE PASCAL, MAUVAIS PASCALE, POINSARD CEDRIC, LINGET JEAN MICHEL
Year of Publication 07.09.2012
Get full text
Year of Publication 07.09.2012
Patent
PHENOL DERIVATIVES AND PHARMACEUTICAL OR COSMETIC USE THEREOF
RETHORE SANDRINE, COLLETTE PASCAL, MAUVAIS PASCALE, POINSARD CEDRIC, LINGET JEAN MICHEL
Year of Publication 29.08.2012
Get full text
Year of Publication 29.08.2012
Patent
PHENOL DERIVATIVES AND THE PHARMACEUTICAL OR COSMETIC USE THEREOF
RETHORE SANDRINE, COLLETTE PASCAL, MAUVAIS PASCALE, POINSARD CEDRIC, LINGET JEAN MICHEL
Year of Publication 29.08.2012
Get full text
Year of Publication 29.08.2012
Patent
CANNABINOID RECEPTOR MODULATORS
NIELSEN PETER AADAL, ALMHOLT DORTHE, MURRAY ANTHONY, NOERREGAARD PIA KARINA, BJURLING EMELIE, HOEGBERG THOMAS, RECEVEUR JEAN MARIE, LINGET JEAN MICHEL
Year of Publication 18.08.2010
Get full text
Year of Publication 18.08.2010
Patent
The Discovery of Tadalafil: A Novel and Highly Selective PDE5 Inhibitor. 2: 2,3,6,7,12,12a-hexahydropyrazino[1‘,2‘:1,6]pyrido[3,4-b]indole-1,4-dione Analogues
Daugan, Alain, Grondin, Pascal, Ruault, Cécile, Le Monnier de Gouville, Anne-Charlotte, Coste, Hervé, Linget, Jean Michel, Kirilovsky, Jorge, Hyafil, François, Labaudinière, Richard
Published in Journal of medicinal chemistry (09.10.2003)
Published in Journal of medicinal chemistry (09.10.2003)
Get full text
Journal Article
Substituted 2-[(4-Aminomethyl)phenoxy]-2-methylpropionic Acid PPARα Agonists. 1. Discovery of a Novel Series of Potent HDLc Raising Agents
Sierra, Michael L, Beneton, Véronique, Boullay, Anne-Bénédict, Boyer, Thierry, Brewster, Andrew G, Donche, Frédéric, Forest, Marie-Claire, Fouchet, Marie-Hélène, Gellibert, Françoise J, Grillot, Didier A, Lambert, Millard H, Laroze, Alain, Le Grumelec, Christelle, Linget, Jean Michel, Montana, Valerie G, Nguyen, Van-Loc, Nicodème, Edwige, Patel, Vipul, Penfornis, Annie, Pineau, Olivier, Pohin, Danig, Potvain, Florent, Poulain, Géraldine, Ruault, Cécile Bertho, Saunders, Michael, Toum, Jérôme, Xu, H. Eric, Xu, Robert X, Pianetti, Pascal M
Published in Journal of medicinal chemistry (22.02.2007)
Published in Journal of medicinal chemistry (22.02.2007)
Get full text
Journal Article
ChemInform Abstract: Conversion of 4-Cyanomethyl-pyrazole-3-carboxamides into CB1 Antagonists with Lowered Propensity to Pass the Blood-Brain-Barrier
Receveur, Jean-Marie, Murray, Anthony, Linget, Jean-Michel, Noerregaard, Pia K., Cooper, Martin, Bjurling, Emelie, Nielsen, Peter Aadal, Hoegberg, Thomas
Published in ChemInform (08.06.2010)
Published in ChemInform (08.06.2010)
Get full text
Journal Article
Substituted 2-[(4-aminomethyl)phenoxy]-2-methylpropionic acid PPARalpha agonists. 1. Discovery of a novel series of potent HDLc raising agents
Sierra, Michael L, Beneton, Véronique, Boullay, Anne-Bénédict, Boyer, Thierry, Brewster, Andrew G, Donche, Frédéric, Forest, Marie-Claire, Fouchet, Marie-Hélène, Gellibert, Françoise J, Grillot, Didier A, Lambert, Millard H, Laroze, Alain, Le Grumelec, Christelle, Linget, Jean Michel, Montana, Valerie G, Nguyen, Van-Loc, Nicodème, Edwige, Patel, Vipul, Penfornis, Annie, Pineau, Olivier, Pohin, Danig, Potvain, Florent, Poulain, Géraldine, Ruault, Cécile Bertho, Saunders, Michael, Toum, Jérôme, Xu, H Eric, Xu, Robert X, Pianetti, Pascal M
Published in Journal of medicinal chemistry (22.02.2007)
Get full text
Published in Journal of medicinal chemistry (22.02.2007)
Journal Article