The identification of novel acid isostere based inhibitors of the VPS10P family sorting receptor Sortilin
Andersen, Jacob Lauwring, Lindberg, Samsa, Langgård, Morten, Maltas, Philip J., Rønn, Lars Christian Biilmann, Bundgaard, Christoffer, Strandbygaard, Dorthe, Thirup, Søren, Watson, Stephen P
Published in Bioorganic & medicinal chemistry letters (01.06.2017)
Published in Bioorganic & medicinal chemistry letters (01.06.2017)
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The identification of AF38469: An orally bioavailable inhibitor of the VPS10P family sorting receptor Sortilin
Schroder, Tenna Juul, Christensen, Soren, Lindberg, Samsa, Langgard, Morten, David, Laurent, Maltas, Philip J., Eskildsen, Jorgen, Jacobsen, Jan, Tagmose, Lena, Simonsen, Klaus Baek, Ronn, Lars Christian Biilmann, de Jong, Inge E. M., Malik, Ibrahim J., Karlsson, Jens-Jakob, Bundgaard, Christoffer, Egebjerg, Jan, Stavenhagen, Jeffrey B., Strandbygard, Dorthe, Thirup, Soren, Andersen, Jacob Lauwring, Uppalanchi, Srinivas, Pervaram, Sridhar, Kasturi, Shiva Prasad, Eradi, Pradheep, Sakumudi, Durga Rao, Watson, Stephen P.
Published in Bioorganic & medicinal chemistry letters (01.01.2014)
Published in Bioorganic & medicinal chemistry letters (01.01.2014)
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Identification of the first small-molecule ligand of the neuronal receptor sortilin and structure determination of the receptor-ligand complex
Andersen, Jacob Lauwring, Schrøder, Tenna Juul, Christensen, Søren, Strandbygård, Dorthe, Pallesen, Lone Tjener, García-Alai, Maria Marta, Lindberg, Samsa, Langgård, Morten, Eskildsen, Jørgen Calí, David, Laurent, Tagmose, Lena, Simonsen, Klaus Baek, Maltas, Philip James, Rønn, Lars Christian Biilmann, de Jong, Inge E. M., Malik, Ibrahim John, Egebjerg, Jan, Karlsson, Jens-Jacob, Uppalanchi, Srinivas, Sakumudi, Durga Rao, Eradi, Pradheep, Watson, Steven P., Thirup, Søren
Published in Acta crystallographica. Section D, Biological crystallography. (01.02.2014)
Published in Acta crystallographica. Section D, Biological crystallography. (01.02.2014)
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