The Interleukin‐1 Receptor–Associated Kinase 4 Inhibitor PF‐06650833 Blocks Inflammation in Preclinical Models of Rheumatic Disease and in Humans Enrolled in a Randomized Clinical Trial
Winkler, Aaron, Sun, Weiyong, De, Saurav, Jiao, Aiping, Sharif, M. Nusrat, Symanowicz, Peter T., Athale, Shruti, Shin, Julia H., Wang, Ju, Jacobson, Bruce A., Ramsey, Simeon J., Dower, Ken, Andreyeva, Tatyana, Liu, Heng, Hegen, Martin, Homer, Bruce L., Brodfuehrer, Joanne, Tilley, Mera, Gilbert, Steven A., Danto, Spencer I., Beebe, Jean J., Barnes, Betsy J., Pascual, Virginia, Lin, Lih‐Ling, Kilty, Iain, Fleming, Margaret, Rao, Vikram R.
Published in Arthritis & rheumatology (Hoboken, N.J.) (01.12.2021)
Published in Arthritis & rheumatology (Hoboken, N.J.) (01.12.2021)
Get full text
Journal Article
Efficacy and Pharmacology of the NLRP3 Inflammasome Inhibitor CP-456,773 (CRID3) in Murine Models of Dermal and Pulmonary Inflammation
Primiano, Michael J, Lefker, Bruce A, Bowman, Michael R, Bree, Andrea G, Hubeau, Cedric, Bonin, Paul D, Mangan, Matthew, Dower, Ken, Monks, Brian G, Cushing, Leah, Wang, Stephen, Guzova, Julia, Jiao, Aiping, Lin, Lih-Ling, Latz, Eicke, Hepworth, David, Hall, J Perry
Published in The Journal of immunology (1950) (15.09.2016)
Published in The Journal of immunology (1950) (15.09.2016)
Get full text
Journal Article
The bromodomain protein inhibitor I-BET151 suppresses expression of inflammatory genes and matrix degrading enzymes in rheumatoid arthritis synovial fibroblasts
Klein, Kerstin, Kabala, Pawel A, Grabiec, Aleksander M, Gay, Renate E, Kolling, Christoph, Lin, Lih-Ling, Gay, Steffen, Tak, Paul P, Prinjha, Rab K, Ospelt, Caroline, Reedquist, Kris A
Published in Annals of the rheumatic diseases (01.02.2016)
Published in Annals of the rheumatic diseases (01.02.2016)
Get full text
Journal Article
Discovery of PF-06928215 as a high affinity inhibitor of cGAS enabled by a novel fluorescence polarization assay
Hall, Justin, Brault, Amy, Vincent, Fabien, Weng, Shawn, Wang, Hong, Dumlao, Darren, Aulabaugh, Ann, Aivazian, Dikran, Castro, Dana, Chen, Ming, Culp, Jeffrey, Dower, Ken, Gardner, Joseph, Hawrylik, Steven, Golenbock, Douglas, Hepworth, David, Horn, Mark, Jones, Lyn, Jones, Peter, Latz, Eicke, Li, Jing, Lin, Lih-Ling, Lin, Wen, Lin, David, Lovering, Frank, Niljanskul, Nootaree, Nistler, Ryan, Pierce, Betsy, Plotnikova, Olga, Schmitt, Daniel, Shanker, Suman, Smith, James, Snyder, William, Subashi, Timothy, Trujillo, John, Tyminski, Edyta, Wang, Guoxing, Wong, Jimson, Lefker, Bruce, Dakin, Leslie, Leach, Karen
Published in PloS one (21.09.2017)
Published in PloS one (21.09.2017)
Get full text
Journal Article
IRAK4 kinase activity controls Toll-like receptor–induced inflammation through the transcription factor IRF5 in primary human monocytes
Cushing, Leah, Winkler, Aaron, Jelinsky, Scott A., Lee, Katherine, Korver, Wouter, Hawtin, Rachael, Rao, Vikram R., Fleming, Margaret, Lin, Lih-Ling
Published in The Journal of biological chemistry (10.11.2017)
Published in The Journal of biological chemistry (10.11.2017)
Get full text
Journal Article
Microbial dysbiosis and childhood asthma development: Integrated role of the airway and gut microbiome, environmental exposures, and host metabolic and immune response
Liu, Conglin, Makrinioti, Heidi, Saglani, Sejal, Bowman, Michael, Lin, Lih-Ling, Camargo, Carlos A., Hasegawa, Kohei, Zhu, Zhaozhong
Published in Frontiers in immunology (30.09.2022)
Published in Frontiers in immunology (30.09.2022)
Get full text
Journal Article
Subsets of ILC3-ILC1-like cells generate a diversity spectrum of innate lymphoid cells in human mucosal tissues
Cella, Marina, Gamini, Ramya, Sécca, Cristiane, Collins, Patrick L, Zhao, Shanrong, Peng, Vincent, Robinette, Michelle L, Schettini, Jorge, Zaitsev, Konstantin, Gordon, William, Bando, Jennifer K, Yomogida, Kentaro, Cortez, Victor, Fronick, Catrina, Fulton, Robert, Lin, Lih-Ling, Gilfillan, Susan, Flavell, Richard A, Shan, Liang, Artyomov, Maxim N, Bowman, Michael, Oltz, Eugene M, Jelinsky, Scott A, Colonna, Marco
Published in Nature immunology (01.08.2019)
Published in Nature immunology (01.08.2019)
Get full text
Journal Article
Computational identification and validation of alternative splicing in ZSF1 rat RNA-seq data, a preclinical model for type 2 diabetic nephropathy
Zhang, Chi, Dower, Ken, Zhang, Baohong, Martinez, Robert V, Lin, Lih-Ling, Zhao, Shanrong
Published in Scientific reports (16.05.2018)
Published in Scientific reports (16.05.2018)
Get full text
Journal Article
Novel biomarkers of a peripheral blood interferon signature associated with drug-naïve early arthritis patients distinguish persistent from self-limiting disease course
Seyhan, Attila A, Gregory, Bernard, Cribbs, Adam P, Bhalara, Sundeept, Li, Yizheng, Loreth, Christine, Zhang, Ying, Guo, Yongjing, Lin, Lih-Ling, Feldmann, Marc, Williams, Lynn M, Brennan, Fionula M, Taylor, Peter C
Published in Scientific reports (01.06.2020)
Published in Scientific reports (01.06.2020)
Get full text
Journal Article
MAPKAP Kinase 2-Deficient Mice Are Resistant to Collagen-Induced Arthritis
Hegen, Martin, Gaestel, Matthias, Nickerson-Nutter, Cheryl L, Lin, Lih-Ling, Telliez, Jean-Baptiste
Published in Journal of Immunology (01.08.2006)
Published in Journal of Immunology (01.08.2006)
Get full text
Journal Article
Mice lacking Tbk1 activity exhibit immune cell infiltrates in multiple tissues and increased susceptibility to LPS-induced lethality
Marchlik, Erica, Thakker, Paresh, Carlson, Thaddeus, Jiang, Zhaozhao, Ryan, Mark, Marusic, Suzana, Goutagny, Nadege, Kuang, Wen, Askew, G. Roger, Roberts, Victoria, Benoit, Stephen, Zhou, Tianhui, Ling, Vincent, Pfeifer, Richard, Stedman, Nancy, Fitzgerald, Katherine A., Lin, Lih‐Ling, Hall, J. Perry
Published in Journal of leukocyte biology (01.12.2010)
Published in Journal of leukocyte biology (01.12.2010)
Get full text
Journal Article
Publisher Correction: Subsets of ILC3-ILC1-like cells generate a diversity spectrum of innate lymphoid cells in human mucosal tissues
Cella, Marina, Gamini, Ramya, Sécca, Cristiane, Collins, Patrick L, Zhao, Shanrong, Peng, Vincent, Robinette, Michelle L, Schettini, Jorge, Zaitsev, Konstantin, Gordon, William, Bando, Jennifer K, Yomogida, Kentaro, Cortez, Victor, Fronick, Catrina, Fulton, Robert, Lin, Lih-Ling, Gilfillan, Susan, Flavell, Richard A, Shan, Liang, Artyomov, Maxim N, Bowman, Michael, Oltz, Eugene M, Jelinsky, Scott A, Colonna, Marco
Published in Nature immunology (01.10.2019)
Published in Nature immunology (01.10.2019)
Get full text
Journal Article
CD47 antibody blockade suppresses microglia-dependent phagocytosis and monocyte transition to macrophages, impairing recovery in EAE
Wang, Huan, Newton, Gail, Wu, Liguo, Lin, Lih-Ling, Miracco, Amy S, Natesan, Sridaran, Luscinskas, Francis W
Published in JCI insight (08.11.2021)
Published in JCI insight (08.11.2021)
Get full text
Journal Article
Distinct Cellular Functions of MK2
Kotlyarov, Alexey, Yannoni, Yvonne, Fritz, Susann, Laaß, Kathrin, Telliez, Jean-Baptiste, Pitman, Deborah, Lin, Lih-Ling, Gaestel, Matthias
Published in Molecular and Cellular Biology (01.07.2002)
Published in Molecular and Cellular Biology (01.07.2002)
Get full text
Journal Article
Identification and SAR of a new series of thieno[3,2- d]pyrimidines as Tpl2 kinase inhibitors
Ni, Yike, Gopalsamy, Ariamala, Cole, Derek, Hu, Yonghan, Denny, Rajiah, Ipek, Manus, Liu, Julie, Lee, Julie, Hall, J. Perry, Luong, Michael, Telliez, Jean-Baptiste, Lin, Lih-Ling
Published in Bioorganic & medicinal chemistry letters (01.10.2011)
Published in Bioorganic & medicinal chemistry letters (01.10.2011)
Get full text
Journal Article
Pharmacologic Inhibition of Tpl2 Blocks Inflammatory Responses in Primary Human Monocytes, Synoviocytes, and Blood
Hall, J. Perry, Kurdi, Yahya, Hsu, Sang, Cuozzo, John, Liu, Julie, Telliez, Jean-Baptiste, Seidl, Katherine J., Winkler, Aaron, Hu, Yonghan, Green, Neal, Askew, G. Roger, Tam, Steve, Clark, James D., Lin, Lih-Ling
Published in The Journal of biological chemistry (16.11.2007)
Published in The Journal of biological chemistry (16.11.2007)
Get full text
Journal Article
TRIL, a Functional Component of the TLR4 Signaling Complex, Highly Expressed in Brain
Carpenter, Susan, Carlson, Thaddeus, Dellacasagrande, Jerome, Garcia, Amaya, Gibbons, Sharon, Hertzog, Paul, Lyons, Anthony, Lin, Lih-Ling, Lynch, Marina, Monie, Tom, Murphy, Caroline, Seidl, Katherine J, Wells, Christine, Dunne, Aisling, O'Neill, Luke A. J
Published in The Journal of immunology (1950) (15.09.2009)
Published in The Journal of immunology (1950) (15.09.2009)
Get full text
Journal Article
Identification of Pathogenic Immune Cell Subsets Associated With Checkpoint Inhibitor-Induced Myocarditis
Zhu, Han, Galdos, Francisco X, Lee, Daniel, Waliany, Sarah, Huang, Yuhsin Vivian, Ryan, Julia, Dang, Katherine, Neal, Joel W, Wakelee, Heather A, Reddy, Sunil A, Srinivas, Sandy, Lin, Lih-Ling, Witteles, Ronald M, Maecker, Holden T, Davis, Mark M, Nguyen, Patricia K, Wu, Sean M
Published in Circulation (New York, N.Y.) (26.07.2022)
Published in Circulation (New York, N.Y.) (26.07.2022)
Get full text
Journal Article