Cobalt-Catalyzed Diastereoselective Synthesis of C‑Furanosides. Total Synthesis of (−)-Isoaltholactone
Nicolas, Lionel, Izquierdo, Eva, Angibaud, Patrick, Stansfield, Ian, Meerpoel, Lieven, Reymond, Sébastien, Cossy, Janine
Published in Journal of organic chemistry (06.12.2013)
Published in Journal of organic chemistry (06.12.2013)
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Journal Article
Tandem Suzuki-Miyaura Coupling/Acid-Catalyzed Cyclization between Vinyl Ether Boronates and Vinyl Halides: A Concise Approach to Polysubstituted Furans
Butkevich, Alexey N, Meerpoel, Lieven, Stansfield, Ian, Angibaud, Patrick, Corbu, Andrei, Cossy, Janine
Published in Organic letters (02.08.2013)
Published in Organic letters (02.08.2013)
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Journal Article
C-2 Arylation of Piperidines through Directed Transition-Metal-Catalyzed sp3 CH Activation
Prokopcová, Hana, Bergman, Sheba D., Aelvoet, Karel, Smout, Veerle, Herrebout, Wouter, Van der Veken, Benjamin, Meerpoel, Lieven, Maes, Bert U. W.
Published in Chemistry : a European journal (22.11.2010)
Published in Chemistry : a European journal (22.11.2010)
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Journal Article
The Novel Azole R126638 Is a Selective Inhibitor of Ergosterol Synthesis in Candida albicans, Trichophyton spp., and Microsporum canis
VANDEN BOSSCHE, Hugo, AUSMA, Jannie, BOHETS, Hilde, VERMUYTEN, Karen, WILLEMSENS, Gustaaf, MARICHAL, Patrick, MEERPOEL, Lieven, ODDS, Frank, BORGERS, Marcel
Published in Antimicrobial Agents and Chemotherapy (01.09.2004)
Published in Antimicrobial Agents and Chemotherapy (01.09.2004)
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Journal Article
Direct α-Functionalization of Saturated Cyclic Amines
Mitchell, Emily A., Peschiulli, Aldo, Lefevre, Nicolas, Meerpoel, Lieven, Maes, Bert U. W.
Published in Chemistry : a European journal (13.08.2012)
Published in Chemistry : a European journal (13.08.2012)
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Journal Article
Minisci-Photoredox-Mediated α‑Heteroarylation of N‑Protected Secondary Amines: Remarkable Selectivity of Azetidines
Bosset, Cyril, Beucher, Hélène, Bretel, Guillaume, Pasquier, Elisabeth, Queguiner, Laurence, Henry, Cyril, Vos, Ann, Edwards, James P, Meerpoel, Lieven, Berthelot, Didier
Published in Organic letters (05.10.2018)
Published in Organic letters (05.10.2018)
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Journal Article
Stereodivergent Synthesis of Biologically Active Spironucleoside Scaffolds via Catalytic Cyclopropanation of 4-exo-Methylene Furanosides
Neouchy, Zeina, Verhoeven, Jonas, Kong, Hanchu, Zhao, Yongbin, Wang, Wenbin, Brambilla, Marta, Van Hecke, Kristof, Meerpoel, Lieven, Thuring, Jan Willem, Verniest, Guido, Winne, Johan
Published in Journal of organic chemistry (03.12.2021)
Published in Journal of organic chemistry (03.12.2021)
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Journal Article
Regio- and Stereoselective Synthesis of C‑4′ Spirocyclobutyl Ribofuranose Scaffolds and Their Use as Biologically Active Nucleoside Analogues
Jouffroy, Lucile, Verhoeven, Jonas, Brambilla, Marta, Verniest, Guido, Kong, Hanchu, Zhao, Yongbin, Wang, Wenbin, Meerpoel, Lieven, Thuring, Jan Willem, Winne, Johan M
Published in Organic letters (19.11.2021)
Published in Organic letters (19.11.2021)
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Journal Article
Synthesis and Reactivity of Spirocarbocycles as Scaffolds for Nucleoside Analogues
Verhoeven, Jonas, Deraet, Xavier, Pande, Vineet, Sun, Weimei, Alonso, Mercedes, De Proft, Frank, Meerpoel, Lieven, Thuring, Jan Willem, Verniest, Guido
Published in Journal of organic chemistry (04.12.2020)
Published in Journal of organic chemistry (04.12.2020)
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Journal Article
Discovery and Pharmacological Characterization of JNJ-64619178, a Novel Small-Molecule Inhibitor of PRMT5 with Potent Antitumor Activity
Brehmer, Dirk, Beke, Lijs, Wu, Tongfei, Millar, Hillary J, Moy, Christopher, Sun, Weimei, Mannens, Geert, Pande, Vineet, Boeckx, An, van Heerde, Erika, Nys, Thomas, Gustin, Emmanuel M, Verbist, Bie, Zhou, Longen, Fan, Yue, Bhargava, Vipul, Safabakhsh, Pegah, Vinken, Petra, Verhulst, Tinne, Gilbert, Angelique, Rai, Sumit, Graubert, Timothy A, Pastore, Friederike, Fiore, Danilo, Gu, Junchen, Johnson, Amy, Philippar, Ulrike, Morschhäuser, Barbara, Walker, David, De Lange, Desiree, Keersmaekers, Vikki, Viellevoye, Marcel, Diels, Gaston, Schepens, Wim, Thuring, Jan Willem, Meerpoel, Lieven, Packman, Kathryn, Lorenzi, Matthew V, Laquerre, Sylvie
Published in Molecular cancer therapeutics (01.12.2021)
Published in Molecular cancer therapeutics (01.12.2021)
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Journal Article
Synthesis and transformations of pyrrolo[1,2-a][1,3,5]-triazines
Verhoeven, Jonas, Reddy, B. Narendraprasad, Meerpoel, Lieven, Thuring, Jan Willem, Verniest, Guido
Published in Tetrahedron letters (26.12.2018)
Published in Tetrahedron letters (26.12.2018)
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Journal Article
Correction to “Regio- and Stereoselective Synthesis of C‑4′ Spirocyclobutyl Ribofuranose Scaffolds and Their Use as Biologically Active Nucleoside Analogues”
Jouffroy, Lucile, Verhoeven, Jonas, Brambilla, Marta, Verniest, Guido, Kong, Hanchu, Zhao, Yongbin, Wang, Wenbin, Meerpoel, Lieven, Thuring, Jan Willem, Winne, Johan M
Published in Organic letters (21.01.2022)
Published in Organic letters (21.01.2022)
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Journal Article
Iron-Catalyzed Synthesis of Sulfur-Containing Heterocycles
Bosset, Cyril, Lefebvre, Gauthier, Angibaud, Patrick, Stansfield, Ian, Meerpoel, Lieven, Berthelot, Didier, Guérinot, Amandine, Cossy, Janine
Published in Journal of organic chemistry (21.04.2017)
Published in Journal of organic chemistry (21.04.2017)
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Journal Article
Preparation of Novel 4 '-Spirocyclopropyl Nucleoside Analogues
Verhoeven, Jonas, Kong, Hanchu, Zhao, Yongbin, Wang, Wenbin, Pande, Vineet, Brambilla, Marta, Van Hecke, Kristof, Meerpoel, Lieven, Thuring, Jan Willem, Verniest, Guido
Published in Synlett (02.06.2021)
Published in Synlett (02.06.2021)
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Journal Article
Pd(0)-Catalyzed Direct Inter- and Intramolecular C-H Functionalization of 4-Carboxyimidazoles
Frippiat, Steven, Peresson, Antoine, Perse, Thibaut, Ramondenc, Yvan, Schneider, Cedric, Querolle, Olivier, Angibaud, Patrick, Poncelet, Virginie, Meerpoel, Lieven, Levacher, Vincent, Bischoff, Laurent, Baudequin, Christine, Hoarau, Christophe
Published in Synlett (17.06.2020)
Published in Synlett (17.06.2020)
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