Dabigatran etexilate--a novel, reversible, oral direct thrombin inhibitor: interpretation of coagulation assays and reversal of anticoagulant activity
van Ryn, Joanne, Stangier, Joachim, Haertter, Sebastian, Liesenfeld, Karl-Heinz, Wienen, Wolfgang, Feuring, Martin, Clemens, Andreas
Published in Thrombosis and haemostasis (01.06.2010)
Published in Thrombosis and haemostasis (01.06.2010)
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Dabigatran etexilate in atrial fibrillation patients with severe renal impairment: dose identification using pharmacokinetic modeling and simulation
Lehr, Thorsten, Haertter, Sebastian, Liesenfeld, Karl-Heinz, Staab, Alexander, Clemens, Andreas, Reilly, Paul A, Friedman, Jeffrey
Published in Journal of clinical pharmacology (01.09.2012)
Published in Journal of clinical pharmacology (01.09.2012)
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Population pharmacokinetics of adalimumab biosimilar adalimumab‐adbm and reference product in healthy subjects and patients with rheumatoid arthritis to assess pharmacokinetic similarity
Kang, Jia, Eudy‐Byrne, Rena J., Mondick, John, Knebel, William, Jayadeva, Girish, Liesenfeld, Karl‐Heinz
Published in British journal of clinical pharmacology (01.11.2020)
Published in British journal of clinical pharmacology (01.11.2020)
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Enhanced elimination of dabigatran: Identifying the appropriate patient for the use of continuous venovenous hemodialysis instead of intermittent hemodialysis-A simulation analysis
Liesenfeld, Karl-Heinz, Gruenenfelder, Fredrik, Clemens, Andreas
Published in Journal of clinical pharmacology (01.05.2016)
Published in Journal of clinical pharmacology (01.05.2016)
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Low‐dose empagliflozin as adjunct‐to‐insulin therapy in type 1 diabetes: A valid modelling and simulation analysis to confirm efficacy
Perkins, Bruce A., Soleymanlou, Nima, Rosenstock, Julio, Skyler, Jay S., Laffel, Lori M., Liesenfeld, Karl‐Heinz, Neubacher, Dietmar, Riggs, Matthew M., Johnston, Curtis K., Eudy‐Byrne, Rena J., Elmokadem, Ahmed, George, Jyothis T., Marquard, Jan, Nock, Valerie
Published in Diabetes, obesity & metabolism (01.03.2020)
Published in Diabetes, obesity & metabolism (01.03.2020)
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Evaluation of Pharmacokinetics and Pharmacodynamics of BI 425809, a Novel GlyT1 Inhibitor: Translational Studies
Rosenbrock, Holger, Desch, Michael, Kleiner, Oliver, Dorner‐Ciossek, Cornelia, Schmid, Bernhard, Keller, Sascha, Schlecker, Christina, Moschetti, Viktoria, Goetz, Sophia, Liesenfeld, Karl‐Heinz, Fillon, Gwenaelle, Giovannini, Riccardo, Ramael, Steven, Wunderlich, Glen, Wind, Sven
Published in Clinical and translational science (01.11.2018)
Published in Clinical and translational science (01.11.2018)
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Population pharmacokinetic analysis of the new oral thrombin inhibitor dabigatran etexilate (BIBR 1048) in patients undergoing primary elective total hip replacement surgery
Trocóniz, Iñaki F, Tillmann, Christiane, Liesenfeld, Karl-Heinz, Schäfer, Hans-Günter, Stangier, Joachim
Published in Journal of clinical pharmacology (01.03.2007)
Published in Journal of clinical pharmacology (01.03.2007)
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A Model-Informed Drug Development (MIDD) Approach for a Low Dose of Empagliflozin in Patients with Type 1 Diabetes
Johnston, Curtis K, Eudy-Byrne, Rena J, Elmokadem, Ahmed, Nock, Valerie, Marquard, Jan, Soleymanlou, Nima, Riggs, Matthew M, Liesenfeld, Karl-Heinz
Published in Pharmaceutics (02.04.2021)
Published in Pharmaceutics (02.04.2021)
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Effects of the direct thrombin inhibitor dabigatran on ex vivo coagulation time in orthopaedic surgery patients: a population model analysis
Liesenfeld, Karl‐Heinz, Schäfer, Hans G., Trocóniz, Iñaki F., Tillmann, Christiane, Eriksson, Bengt I., Stangier, Joachim
Published in British journal of clinical pharmacology (01.11.2006)
Published in British journal of clinical pharmacology (01.11.2006)
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Effective elimination of dabigatran by haemodialysis. A phase I single-centre study in patients with end-stage renal disease
Khadzhynov, Dmytro, Wagner, Frank, Formella, Stephan, Wiegert, Erol, Moschetti, Viktoria, Slowinski, Torsten, Neumayer, Hans-H, Liesenfeld, Karl-Heinz, Lehr, Thorsten, Härtter, Sebastian, Friedman, Jeffrey, Peters, Harm, Clemens, Andreas
Published in Thrombosis and haemostasis (01.04.2013)
Published in Thrombosis and haemostasis (01.04.2013)
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Population pharmacokinetics of tamsulosin hydrochloride in paediatric patients with neuropathic and non‐neuropathic bladder
Tsuda, Yasuhiro, Tatami, Shinji, Yamamura, Norio, Tadayasu, Yusuke, Sarashina, Akiko, Liesenfeld, Karl‐Heinz, Staab, Alexander, Schäfer, Hans‐Günter, Ieiri, Ichiro, Higuchi, Shun
Published in British journal of clinical pharmacology (01.07.2010)
Published in British journal of clinical pharmacology (01.07.2010)
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Pharmacokinetic-Interactions of BI 425809, a Novel Glycine Transporter 1 Inhibitor, With Cytochrome P450 and P-Glycoprotein Substrates: Findings From In Vitro Analyses and an Open-Label, Single-Sequence Phase I Study
Desch, Michael, Schlecker, Christina, Hohl, Kathrin, Liesenfeld, Karl-Heinz, Chan, Tom, Müller, Fabian, Wunderlich, Glen, Keller, Sascha, Ishiguro, Naoki, Wind, Sven
Published in Journal of clinical psychopharmacology (01.03.2023)
Published in Journal of clinical psychopharmacology (01.03.2023)
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Population pharmacokinetics of nintedanib, an inhibitor of tyrosine kinases, in patients with non-small cell lung cancer or idiopathic pulmonary fibrosis
Schmid, Ulrike, Liesenfeld, Karl-Heinz, Fleury, Angele, Dallinger, Claudia, Freiwald, Matthias
Published in Cancer chemotherapy and pharmacology (01.01.2018)
Published in Cancer chemotherapy and pharmacology (01.01.2018)
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Switching Between Adalimumab Reference Product and BI 695501 in Patients with Chronic Plaque Psoriasis (VOLTAIRE-X): A Randomized Controlled Trial
Menter, Alan, Cohen, Stanley, Kay, Jonathan, Strand, Vibeke, Gottlieb, Alice, Hanauer, Stephen, Eduru, Sravan Kumar, Buschke, Susanne, Lang, Benjamin, Liesenfeld, Karl-Heinz, Schaible, Jennifer, McCabe, Dorothy
Published in American journal of clinical dermatology (01.09.2022)
Published in American journal of clinical dermatology (01.09.2022)
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Pharmacometric Characterization of Dabigatran Hemodialysis
Liesenfeld, Karl-Heinz, Staab, Alexander, Härtter, Sebastian, Formella, Stephan, Clemens, Andreas, Lehr, Thorsten
Published in Clinical pharmacokinetics (01.06.2013)
Published in Clinical pharmacokinetics (01.06.2013)
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Multiple Rising Doses of Oral BI 425809, a GlyT1 Inhibitor, in Young and Elderly Healthy Volunteers: A Randomised, Double-Blind, Phase I Study Investigating Safety and Pharmacokinetics
Moschetti, Viktoria, Schlecker, Christina, Wind, Sven, Goetz, Sophia, Schmitt, Holger, Schultz, Armin, Liesenfeld, Karl-Heinz, Wunderlich, Glen, Desch, Michael
Published in Clinical drug investigation (01.08.2018)
Published in Clinical drug investigation (01.08.2018)
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Safety, Tolerability and Pharmacokinetics of Oral BI 425809, a Glycine Transporter 1 Inhibitor, in Healthy Male Volunteers: A Partially Randomised, Single-Blind, Placebo-Controlled, First-in-Human Study
Moschetti, Viktoria, Desch, Michael, Goetz, Sophia, Liesenfeld, Karl-Heinz, Rosenbrock, Holger, Kammerer, Klaus-Peter, Wunderlich, Glen, Wind, Sven
Published in European journal of drug metabolism and pharmacokinetics (01.04.2018)
Published in European journal of drug metabolism and pharmacokinetics (01.04.2018)
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Effects of Cytochrome P450 3A4 Induction and Inhibition on the Pharmacokinetics of BI 425809, a Novel Glycine Transporter 1 Inhibitor
Desch, Michael, Wunderlich, Glen, Goettel, Markus, Goetz, Sophia, Liesenfeld, Karl-Heinz, Chan, Tom S., Rosenbrock, Holger, Sennewald, Regina, Link, Jasmin, Keller, Sascha, Wind, Sven
Published in European journal of drug metabolism and pharmacokinetics (01.01.2022)
Published in European journal of drug metabolism and pharmacokinetics (01.01.2022)
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A combined pharmacometric analysis of dabigatran etexilate in healthy volunteers and patients with atrial fibrillation or undergoing orthopaedic surgery
Dansirikul, C, Lehr, T, Liesenfeld, K-H, Haertter, S, Staab, A
Published in Thrombosis and haemostasis (01.04.2012)
Published in Thrombosis and haemostasis (01.04.2012)
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